| Title : A Phenotypic Screen Identifies Potent DPP9 Inhibitors Capable of Killing HIV-1 Infected Cells - Moore_2022_ACS.Chem.Biol_17_2595 |
| Author(s) : Moore KP , Schwaid AG , Tudor M , Park S , Beshore DC , Converso A , Shipe WD , Anand R , Lan P , Moningka R , Rothman DM , Sun W , Chi A , Cornella-Taracido I , Adam GC , Bahnck-Teets C , Carroll SS , Fay JF , Goh SL , Lusen J , Quan S , Rodriguez S , Xu M , Andrews CL , Song C , Filzen T , Li J , Hollenstein K , Klein DJ , Lammens A , Lim UM , Fang Z , McHale C , Li Y , Lu M , Diamond TL , Howell BJ , Zuck P , Balibar CJ |
| Ref : ACS Chemical Biology , 17 :2595 , 2022 |
| Abstract : |
| PubMedSearch : Moore_2022_ACS.Chem.Biol_17_2595 |
| PubMedID: 36044633 |
| Gene_locus related to this paper: human-DPP8 , human-DPP9 |
| Title : Identification of potent, highly constrained CGRP receptor antagonists - Stump_2010_Bioorg.Med.Chem.Lett_20_2572 |
| Author(s) : Stump CA , Bell IM , Bednar RA , Fay JF , Gallicchio SN , Hershey JC , Jelley R , Kreatsoulas C , Moore EL , Mosser SD , Quigley AG , Roller SA , Salvatore CA , Sharik SS , Theberge CR , Zartman CB , Kane SA , Graham SL , Selnick HG , Vacca JP , Williams TM |
| Ref : Bioorganic & Medicinal Chemistry Lett , 20 :2572 , 2010 |
| Abstract : |
| PubMedSearch : Stump_2010_Bioorg.Med.Chem.Lett_20_2572 |
| PubMedID: 20299218 |
| Title : The discovery of highly potent CGRP receptor antagonists - Stump_2009_Bioorg.Med.Chem.Lett_19_214 |
| Author(s) : Stump CA , Bell IM , Bednar RA , Bruno JG , Fay JF , Gallicchio SN , Johnston VK , Moore EL , Mosser SD , Quigley AG , Salvatore CA , Theberge CR , Blair Zartman C , Zhang XF , Kane SA , Graham SL , Vacca JP , Williams TM |
| Ref : Bioorganic & Medicinal Chemistry Lett , 19 :214 , 2009 |
| Abstract : |
| PubMedSearch : Stump_2009_Bioorg.Med.Chem.Lett_19_214 |
| PubMedID: 19010673 |
| Title : Novel CGRP receptor antagonists through a design strategy of target simplification with addition of molecular flexibility - Wood_2009_Bioorg.Med.Chem.Lett_19_5787 |
| Author(s) : Wood MR , Schirripa KM , Kim JJ , Quigley AG , Stump CA , Bell IM , Bednar RA , Fay JF , Bruno JG , Moore EL , Mosser SD , Roller S , Salvatore CA , Kane SA , Vacca JP , Selnick HG |
| Ref : Bioorganic & Medicinal Chemistry Lett , 19 :5787 , 2009 |
| Abstract : |
| PubMedSearch : Wood_2009_Bioorg.Med.Chem.Lett_19_5787 |
| PubMedID: 19703767 |
| Title : Potent benzimidazolone-based CGRP receptor antagonists - Theberge_2008_Bioorg.Med.Chem.Lett_18_6122 |
| Author(s) : Theberge CR , Bednar RA , Bell IM , Corcoran HA , Fay JF , Hershey JC , Johnston VK , Kane SA , Mosser S , Salvatore CA , Williams TM , Zartman CB , Zhang XF , Graham SL , Vacca JP |
| Ref : Bioorganic & Medicinal Chemistry Lett , 18 :6122 , 2008 |
| Abstract : |
| PubMedSearch : Theberge_2008_Bioorg.Med.Chem.Lett_18_6122 |
| PubMedID: 18947992 |