Title : Tight-Binding Small-Molecule Carboxylesterase 2 Inhibitors Reduce Intracellular Irinotecan Activation - Kailass_2024_J.Med.Chem__ |
Author(s) : Kailass K , Casalena D , Jenane L , McEdwards G , Auld DS , Sadovski O , Kaye EG , Hudson E , Nettleton D , Currie MA , Beharry AA |
Ref : Journal of Medicinal Chemistry , : , 2024 |
Abstract : Kailass_2024_J.Med.Chem__ |
ESTHER : Kailass_2024_J.Med.Chem__ |
PubMedSearch : Kailass_2024_J.Med.Chem__ |
PubMedID: 38265364 |
Gene_locus related to this paper: human-CES2 |
Title : Two-Photon Photodynamic Therapy Targeting Cancers with Low Carboxylesterase 2 Activity Guided by Ratiometric Fluorescence - Kailass_2022_J.Med.Chem__ |
Author(s) : Kailass K , Sadovski O , Zipfel WR , Beharry AA |
Ref : Journal of Medicinal Chemistry , : , 2022 |
Abstract : Kailass_2022_J.Med.Chem__ |
ESTHER : Kailass_2022_J.Med.Chem__ |
PubMedSearch : Kailass_2022_J.Med.Chem__ |
PubMedID: 35700557 |
Title : Measuring human carboxylesterase 2 activity in pancreatic cancer patient-derived xenografts using a ratiometric fluorescent chemosensor - Kailass_2019_Chem.Sci_10_8428 |
Author(s) : Kailass K , Sadovski O , Capello M , Kang Y , Fleming JB , Hanash SM , Beharry AA |
Ref : Chem Sci , 10 :8428 , 2019 |
Abstract : Kailass_2019_Chem.Sci_10_8428 |
ESTHER : Kailass_2019_Chem.Sci_10_8428 |
PubMedSearch : Kailass_2019_Chem.Sci_10_8428 |
PubMedID: 31803422 |
Gene_locus related to this paper: human-CES2 |