| Title : Sensitive quantification of fibroblast activation protein and high-throughput screening for inhibition by FDA-approved compounds - Cermakova_2024_Eur.J.Med.Chem_280_116948 |
| Author(s) : Cermakova K , Simkova A , Wichterle F , Krystufek R , Stanurova J , Vanickova Z , Busek P , Konvalinka J , Sacha P |
| Ref : Eur Journal of Medicinal Chemistry , 280 :116948 , 2024 |
| Abstract : |
| PubMedSearch : Cermakova_2024_Eur.J.Med.Chem_280_116948 |
| PubMedID: 39437576 |
| Gene_locus related to this paper: human-FAP |
| Title : Sensitive quantification of fibroblast activation protein and high-throughput screening for inhibition by FDA-approved compounds - Cermakova_2024_Eur.J.Med.Chem_280_116948 |
| Author(s) : Cermakova K , Simkova A , Wichterle F , Krystufek R , Stanurova J , Vanickova Z , Busek P , Konvalinka J , Sacha P |
| Ref : Eur Journal of Medicinal Chemistry , 280 :116948 , 2024 |
| Abstract : |
| PubMedSearch : Cermakova_2024_Eur.J.Med.Chem_280_116948 |
| PubMedID: 39437576 |
| Gene_locus related to this paper: human-FAP |
| Title : Sensitive quantification of fibroblast activation protein and high-throughput screening for inhibition by FDA-approved compounds - Cermakova_2024_Eur.J.Med.Chem_280_116948 |
| Author(s) : Cermakova K , Simkova A , Wichterle F , Krystufek R , Stanurova J , Vanickova Z , Busek P , Konvalinka J , Sacha P |
| Ref : Eur Journal of Medicinal Chemistry , 280 :116948 , 2024 |
| Abstract : |
| PubMedSearch : Cermakova_2024_Eur.J.Med.Chem_280_116948 |
| PubMedID: 39437576 |
| Gene_locus related to this paper: human-FAP |
| Title : Structure-activity relationship and biochemical evaluation of novel fibroblast activation protein and prolyl endopeptidase inhibitors with alpha-ketoamide warheads - Simkova_2021_Eur.J.Med.Chem_224_113717 |
| Author(s) : Simkova A , Ormsby T , Sidej N , Slavetinska LP , Brynda J , Beranova J , Sacha P , Majer P , Konvalinka J |
| Ref : Eur Journal of Medicinal Chemistry , 224 :113717 , 2021 |
| Abstract : |
| PubMedSearch : Simkova_2021_Eur.J.Med.Chem_224_113717 |
| PubMedID: 34371463 |
| Gene_locus related to this paper: human-FAP |
| Title : Structure-activity relationship and biochemical evaluation of novel fibroblast activation protein and prolyl endopeptidase inhibitors with alpha-ketoamide warheads - Simkova_2021_Eur.J.Med.Chem_224_113717 |
| Author(s) : Simkova A , Ormsby T , Sidej N , Slavetinska LP , Brynda J , Beranova J , Sacha P , Majer P , Konvalinka J |
| Ref : Eur Journal of Medicinal Chemistry , 224 :113717 , 2021 |
| Abstract : |
| PubMedSearch : Simkova_2021_Eur.J.Med.Chem_224_113717 |
| PubMedID: 34371463 |
| Gene_locus related to this paper: human-FAP |
| Title : Structure-activity relationship and biochemical evaluation of novel fibroblast activation protein and prolyl endopeptidase inhibitors with alpha-ketoamide warheads - Simkova_2021_Eur.J.Med.Chem_224_113717 |
| Author(s) : Simkova A , Ormsby T , Sidej N , Slavetinska LP , Brynda J , Beranova J , Sacha P , Majer P , Konvalinka J |
| Ref : Eur Journal of Medicinal Chemistry , 224 :113717 , 2021 |
| Abstract : |
| PubMedSearch : Simkova_2021_Eur.J.Med.Chem_224_113717 |
| PubMedID: 34371463 |
| Gene_locus related to this paper: human-FAP |
| Title : Molecular recognition of fibroblast activation protein for diagnostic and therapeutic applications - Simkova_2020_Biochim.Biophys.Acta.Proteins.Proteom_1868_140409 |
| Author(s) : Simkova A , Busek P , Sedo A , Konvalinka J |
| Ref : Biochimica & Biophysica Acta Proteins Proteom , 1868 :140409 , 2020 |
| Abstract : |
| PubMedSearch : Simkova_2020_Biochim.Biophys.Acta.Proteins.Proteom_1868_140409 |
| PubMedID: 32171757 |
| Gene_locus related to this paper: human-FAP |
| Title : Molecular recognition of fibroblast activation protein for diagnostic and therapeutic applications - Simkova_2020_Biochim.Biophys.Acta.Proteins.Proteom_1868_140409 |
| Author(s) : Simkova A , Busek P , Sedo A , Konvalinka J |
| Ref : Biochimica & Biophysica Acta Proteins Proteom , 1868 :140409 , 2020 |
| Abstract : |
| PubMedSearch : Simkova_2020_Biochim.Biophys.Acta.Proteins.Proteom_1868_140409 |
| PubMedID: 32171757 |
| Gene_locus related to this paper: human-FAP |
| Title : Molecular recognition of fibroblast activation protein for diagnostic and therapeutic applications - Simkova_2020_Biochim.Biophys.Acta.Proteins.Proteom_1868_140409 |
| Author(s) : Simkova A , Busek P , Sedo A , Konvalinka J |
| Ref : Biochimica & Biophysica Acta Proteins Proteom , 1868 :140409 , 2020 |
| Abstract : |
| PubMedSearch : Simkova_2020_Biochim.Biophys.Acta.Proteins.Proteom_1868_140409 |
| PubMedID: 32171757 |
| Gene_locus related to this paper: human-FAP |