Title : Identification of selective and potent inhibitors of fibroblast activation protein and prolyl oligopeptidase - Poplawski_2013_J.Med.Chem_56_3467 |
Author(s) : Poplawski SE , Lai JH , Li Y , Jin Z , Liu Y , Wu W , Wu Y , Zhou Y , Sudmeier JL , Sanford DG , Bachovchin WW |
Ref : Journal of Medicinal Chemistry , 56 :3467 , 2013 |
Abstract : |
PubMedSearch : Poplawski_2013_J.Med.Chem_56_3467 |
PubMedID: 23594271 |
Title : 4-Substituted boro-proline dipeptides: synthesis, characterization, and dipeptidyl peptidase IV, 8, and 9 activities - Wu_2012_Bioorg.Med.Chem.Lett_22_5536 |
Author(s) : Wu W , Liu Y , Milo LJ, Jr. , Shu Y , Zhao P , Li Y , Woznica I , Yu G , Sanford DG , Zhou Y , Poplawski SE , Connolly BA , Sudmeier JL , Bachovchin WW , Lai JH |
Ref : Bioorganic & Medicinal Chemistry Lett , 22 :5536 , 2012 |
Abstract : |
PubMedSearch : Wu_2012_Bioorg.Med.Chem.Lett_22_5536 |
PubMedID: 22853995 |
Title : Pro-soft Val-boroPro: a strategy for enhancing in vivo performance of boronic acid inhibitors of serine proteases - Poplawski_2011_J.Med.Chem_54_2022 |
Author(s) : Poplawski SE , Lai JH , Sanford DG , Sudmeier JL , Wu W , Bachovchin WW |
Ref : Journal of Medicinal Chemistry , 54 :2022 , 2011 |
Abstract : |
PubMedSearch : Poplawski_2011_J.Med.Chem_54_2022 |
PubMedID: 21388136 |
Title : Dipeptide boronic acid inhibitors of dipeptidyl peptidase IV: determinants of potency and in vivo efficacy and safety - Connolly_2008_J.Med.Chem_51_6005 |
Author(s) : Connolly BA , Sanford DG , Chiluwal AK , Healey SE , Peters DE , Dimare MT , Wu W , Liu Y , Maw H , Zhou Y , Li Y , Jin Z , Sudmeier JL , Lai JH , Bachovchin WW |
Ref : Journal of Medicinal Chemistry , 51 :6005 , 2008 |
Abstract : |
PubMedSearch : Connolly_2008_J.Med.Chem_51_6005 |
PubMedID: 18783201 |
Title : Synthesis and characterization of constrained peptidomimetic dipeptidyl peptidase IV inhibitors: amino-lactam boroalanines - Lai_2007_J.Med.Chem_50_2391 |
Author(s) : Lai JH , Wu W , Zhou Y , Maw HH , Liu Y , Milo LJ, Jr. , Poplawski SE , Henry GD , Sudmeier JL , Sanford DG , Bachovchin WW |
Ref : Journal of Medicinal Chemistry , 50 :2391 , 2007 |
Abstract : |
PubMedSearch : Lai_2007_J.Med.Chem_50_2391 |
PubMedID: 17458948 |
Title : Solution structures of active and inactive forms of the DP IV (CD26) inhibitor Pro-boroPro determined by NMR spectroscopy - Sudmeier_1994_Biochemistry_33_12427 |
Author(s) : Sudmeier JL , Gunther UL , Gutheil WG , Coutts SJ , Snow RJ , Barton RW , Bachovchin WW |
Ref : Biochemistry , 33 :12427 , 1994 |
Abstract : |
PubMedSearch : Sudmeier_1994_Biochemistry_33_12427 |
PubMedID: 7918465 |