2QT9
Name : Human dipeptidyl peptidase IV\/CD26 in complex with 4-aryl cyclohexylanine inhibitor 2
Revelation date : 06-Nov-2007
Family : DPP4N_Peptidase_S9
Gene_locus : human-DPP4
PDB file : ESTHER: header of PDB entry RCSB: Full entry
Comment
Kaelin, D.E., Smetin, A.L, Eiermann, G.J., He, H., Leiting, B., Lyons, K.A., Patel, R.A, Patel, S.B, Petrov, A., Scapin, G., Wu, J.K., Thornberry, N.A, Weber, A.E, Duffy, J.L.
Ligand :
References (1)
| Title : 4-arylcyclohexylalanine analogs as potent, selective, and orally active inhibitors of dipeptidyl peptidase IV - Kaelin_2007_Bioorg.Med.Chem.Lett_17_5806 |
| Author(s) : Kaelin DE , Smenton AL , Eiermann GJ , He H , Leiting B , Lyons KA , Patel RA , Patel SB , Petrov A , Scapin G , Wu JK , Thornberry NA , Weber AE , Duffy JL |
| Ref : Bioorganic & Medicinal Chemistry Lett , 17 :5806 , 2007 |
| Abstract : Kaelin_2007_Bioorg.Med.Chem.Lett_17_5806 |
| ESTHER : Kaelin_2007_Bioorg.Med.Chem.Lett_17_5806 |
| PubMedSearch : Kaelin_2007_Bioorg.Med.Chem.Lett_17_5806 |
| PubMedID: 17851076 |
| Gene_locus related to this paper: human-DPP4 |
Representative scheme of Prolylcarboxypeptidase structure and an image from PDBsum server
Databases
PDB-Sum : 2QT9 Previously Class, Architecture, Topology and Homologous superfamily - PDB-Sum server
FSSP : 2QT9 Fold classification based on Structure-Structure alignment of Proteins - FSSP server
SCOP : 2QT9 Structural Classification Of Protein - SCOP server
PROTEOPEDIA : 2QT9 3D, interactive encyclopedia of proteins - PROTEOPEDIA server