5T4B

Name : Human DPP4 in complex with a ligand 34a

Revelation date : 05-Oct-2016

Family : DPP4N_Peptidase_S9

Gene_locus : human-DPP4

PDB file : ESTHER: header of PDB entry RCSB: Full entry

Comment
Pissarnitski, D.A., Zhao, Z., Cole, D., Wu, W.L., Domalski, M., Clader, J.W., Scapin, G., Voigt, J., Soriano, A., Kelly, T., Powles, M.A., Yao, Z., Burnett, D.A.

Ligand :

References (1)

Title : Scaffold-hopping from xanthines to tricyclic guanines: A case study of dipeptidyl peptidase 4 (DPP4) inhibitors - Pissarnitski_2016_Bioorg.Med.Chem_24_5534
Author(s) : Pissarnitski DA , Zhao Z , Cole D , Wu WL , Domalski M , Clader JW , Scapin G , Voigt J , Soriano A , Kelly T , Powles MA , Yao Z , Burnett DA
Ref : Bioorganic & Medicinal Chemistry , 24 :5534 , 2016
PubMedID: 27670099
Gene_locus related to this paper: human-DPP4

Representative scheme of Prolylcarboxypeptidase structure and an image from PDBsum server

Databases

PDB-Sum : 5T4B Previously Class, Architecture, Topology and Homologous superfamily - PDB-Sum server

FSSP : 5T4B Fold classification based on Structure-Structure alignment of Proteins - FSSP server

SCOP : 5T4B Structural Classification Of Protein - SCOP server

PROTEOPEDIA : 5T4B 3D, interactive encyclopedia of proteins - PROTEOPEDIA server