Title : Identification of covalent inhibitors of Staphylococcus aureus serine hydrolases important for virulence and biofilm formation - Upadhyay_2025_Nat.Commun_16_5046 |
Author(s) : Upadhyay T , Woods EC , Dela Ahator S , Julin K , Faucher FF , Uddin MJ , Hollander MJ , Pedowitz NJ , Abegg D , Hammond I , Eke IE , Wang S , Chen S , Bennett JM , Jo J , Lentz CS , Adibekian A , Fellner M , Bogyo M |
Ref : Nat Commun , 16 :5046 , 2025 |
Abstract : |
PubMedSearch : Upadhyay_2025_Nat.Commun_16_5046 |
PubMedID: 40447595 |
Title : Mixed alkyl\/aryl phosphonates identify metabolic serine hydrolases as antimalarial targets - Bennett_2024_Cell.Chem.Biol__ |
Author(s) : Bennett JM , Narwal SK , Kabeche S , Abegg D , Thathy V , Hackett F , Yeo T , Li VL , Muir R , Faucher F , Lovell S , Blackman MJ , Adibekian A , Yeh E , Fidock DA , Bogyo M |
Ref : Cell Chemical Biology , : , 2024 |
Abstract : |
PubMedSearch : Bennett_2024_Cell.Chem.Biol__ |
PubMedID: 39137783 |
Title : Mixed Alkyl\/Aryl Phosphonates Identify Metabolic Serine Hydrolases as Antimalarial Targets - Bennett_2024_bioRxiv__ |
Author(s) : Bennett JM , Narwal SK , Kabeche S , Abegg D , Hackett F , Yeo T , Li VL , Muir RK , Faucher FF , Lovell S , Blackman MJ , Adibekian A , Yeh E , Fidock DA , Bogyo M |
Ref : Biorxiv , : , 2024 |
Abstract : |
PubMedSearch : Bennett_2024_bioRxiv__ |
PubMedID: 38260474 |
Title : Covalent-fragment screening identifies selective inhibitors of multiple Staphylococcus aureus serine hydrolases important for growth and biofilm formation - Bogyo_2024_Res.Sq__ |
Author(s) : Bogyo M , Upadhyay T , Woods E , Ahator S , Julin K , Faucher F , Hollander M , Pedowitz N , Abegg D , Hammond I , Eke I , Wang S , Chen S , Bennett J , Jo J , Lentz C , Adibekian A , Fellner M |
Ref : Res Sq , : , 2024 |
Abstract : |
PubMedSearch : Bogyo_2024_Res.Sq__ |
PubMedID: 39711551 |
Title : Chemoproteomics-Enabled De Novo Discovery of Photoswitchable Carboxylesterase Inhibitors for Optically Controlled Drug Metabolism - Dwyer_2021_Angew.Chem.Int.Ed.Engl_60_3071 |
Author(s) : Dwyer BG , Wang C , Abegg D , Racioppo B , Qiu N , Zhao Z , Pechalrieu D , Shuster A , Hoch DG , Adibekian A |
Ref : Angew Chem Int Ed Engl , 60 :3071 , 2021 |
Abstract : |
PubMedSearch : Dwyer_2021_Angew.Chem.Int.Ed.Engl_60_3071 |
PubMedID: 33035395 |
Title : Combined Omics Approach Identifies Gambogic Acid and Related Xanthones as Covalent Inhibitors of the Serine Palmitoyltransferase Complex - Hoch_2020_Cell.Chem.Biol_27_586 |
Author(s) : Hoch DG , Abegg D , Hannich JT , Pechalrieu D , Shuster A , Dwyer BG , Wang C , Zhang X , You Q , Riezman H , Adibekian A |
Ref : Cell Chemical Biology , 27 :586 , 2020 |
Abstract : |
PubMedSearch : Hoch_2020_Cell.Chem.Biol_27_586 |
PubMedID: 32330443 |
Title : Discovery and Evaluation of New Activity-Based Probes for Serine Hydrolases - Wang_2019_Chembiochem_20_2212 |
Author(s) : Wang C , Abegg D , Dwyer BG , Adibekian A |
Ref : Chembiochem , 20 :2212 , 2019 |
Abstract : |
PubMedSearch : Wang_2019_Chembiochem_20_2212 |
PubMedID: 30968522 |
Title : Cysteine-reactive probes and their use in chemical proteomics - Hoch_2018_Chem.Commun.(Camb)_54_4501 |
Author(s) : Hoch DG , Abegg D , Adibekian A |
Ref : Chem Commun (Camb) , 54 :4501 , 2018 |
Abstract : |
PubMedSearch : Hoch_2018_Chem.Commun.(Camb)_54_4501 |
PubMedID: 29645055 |