Title : Synthesis and Anti-Diabetic Activity of an 8-Purine Derivative as a Novel DPP-4 Inhibitor in Obese Diabetic Zucker Rats - Chayah_2024_Drug.Des.Devel.Ther_18_1133 |
Author(s) : Chayah M , Luque-Gonzalez A , Gomez-Perez V , Salagre D , Al-Shdaifat A , Campos JM , Conejo-Garcia A , Agil A |
Ref : Drug Des Devel Ther , 18 :1133 , 2024 |
Abstract : |
PubMedSearch : Chayah_2024_Drug.Des.Devel.Ther_18_1133 |
PubMedID: 38618281 |
Title : Galantamine Based Novel Acetylcholinesterase Enzyme Inhibitors: A Molecular Modeling Design Approach - Silva_2023_Molecules_28_:1035 |
Author(s) : Silva LB , Ferreira EFB , Maryam , Espejo-Roman JM , Costa GV , Cruz JV , Kimani NM , Costa JS , Bittencourt J , Cruz JN , Campos JM , Santos CBR |
Ref : Molecules , 28 :1035 , 2023 |
Abstract : |
PubMedSearch : Silva_2023_Molecules_28_:1035 |
PubMedID: 36770702 |
Title : Development of Potential Multi-Target Inhibitors for Human Cholinesterases and Beta-Secretase 1: A Computational Approach - Barbosa_2023_Pharmaceuticals.(Basel)_16_ |
Author(s) : Barbosa DB , do Bomfim MR , de Oliveira TA , da Silva AM , Taranto AG , Cruz JN , de Carvalho PB , Campos JM , Santos CBR , Leite FHA |
Ref : Pharmaceuticals (Basel) , 16 : , 2023 |
Abstract : |
PubMedSearch : Barbosa_2023_Pharmaceuticals.(Basel)_16_ |
PubMedID: 38139784 |
Title : Identification of a Novel Dual Inhibitor of Acetylcholinesterase and Butyrylcholinesterase: In Vitro and In Silico Studies - de Almeida_2023_Pharmaceuticals.(Basel)_16_ |
Author(s) : de Almeida RBM , Barbosa DB , do Bomfim MR , Amparo JAO , Andrade BS , Costa SL , Campos JM , Cruz JN , Santos CBR , Leite FHA , Botura MB |
Ref : Pharmaceuticals (Basel) , 16 : , 2023 |
Abstract : |
PubMedSearch : de Almeida_2023_Pharmaceuticals.(Basel)_16_ |
PubMedID: 36678592 |
Title : Homodimeric bis-quaternary heterocyclic ammonium salts as potent acetyl- and butyrylcholinesterase inhibitors: a systematic investigation of the influence of linker and cationic heads over affinity and selectivity - Conejo-Garcia_2011_J.Med.Chem_54_2627 |
Author(s) : Conejo-Garcia A , Pisani L , Nunez Mdel C , Catto M , Nicolotti O , Leonetti F , Campos JM , Gallo MA , Espinosa A , Carotti A |
Ref : Journal of Medicinal Chemistry , 54 :2627 , 2011 |
Abstract : |
PubMedSearch : Conejo-Garcia_2011_J.Med.Chem_54_2627 |
PubMedID: 21417225 |