Gembus V

References (5)

Title : Design, synthesis and preliminary biological evaluation of rivastigmine-INDY hybrids as multitarget ligands against Alzheimer's disease by targeting butyrylcholinesterase and DYRK1A\/CLK1 kinases - Tintas_2024_RSC.Med.Chem_15_963
Author(s) : Tintas ML , Peauger L , Barre A , Papamical C , Besson T , Sopkova-de Oliveira Santos J , Gembus V , Levacher V
Ref : RSC Med Chem , 15 :963 , 2024
Abstract :
PubMedSearch : Tintas_2024_RSC.Med.Chem_15_963
PubMedID: 38516603

Title : Design, Synthesis, and In Vitro Biological Activities of a Bio-Oxidizable Prodrug to Deliver Both ChEs and DYRK1A Inhibitors for AD Therapy - Barre_2019_Molecules_24_
Author(s) : Barre A , Azzouz R , Gembus V , Papamicael C , Levacher V
Ref : Molecules , 24 : , 2019
Abstract :
PubMedSearch : Barre_2019_Molecules_24_
PubMedID: 30939771

Title : Rational design of carbamate-based dual binding site and central AChE inhibitors by a 'biooxidisable' prodrug approach: Synthesis, invitro evaluation and docking studies - Tintas_2018_Eur.J.Med.Chem_155_171
Author(s) : Tintas ML , Gembus V , Alix F , Barre A , Coadou G , Truong L , Sebban M , Papamical C , Oulyadi H , Levacher V
Ref : Eur Journal of Medicinal Chemistry , 155 :171 , 2018
Abstract :
PubMedSearch : Tintas_2018_Eur.J.Med.Chem_155_171
PubMedID: 29886321

Title : Donepezil-Based Central Acetylcholinesterase Inhibitors by Means of a Bio-Oxidizable Prodrug Strategy: Design, Synthesis, and in Vitro Biological Evaluation - Peauger_2017_J.Med.Chem_60_5909
Author(s) : Peauger L , Azzouz R , Gembus V , Tintas ML , Sopkova-de Oliveira Santos J , Bohn P , Papamicael C , Levacher V
Ref : Journal of Medicinal Chemistry , 60 :5909 , 2017
Abstract :
PubMedSearch : Peauger_2017_J.Med.Chem_60_5909
PubMedID: 28613859

Title : Dihydroquinoline Carbamate Derivatives as Bio-oxidizable Prodrugs for Brain Delivery of Acetylcholinesterase Inhibitors: [(11)C] Radiosynthesis and Biological Evaluation - Bohn_2015_ACS.Chem.Neurosci_6_737
Author(s) : Bohn P , Gourand F , Papamicael C , Ibazizene M , Dhilly M , Gembus V , Alix F , Tintas ML , Marsais F , Barre L , Levacher V
Ref : ACS Chem Neurosci , 6 :737 , 2015
Abstract :
PubMedSearch : Bohn_2015_ACS.Chem.Neurosci_6_737
PubMedID: 25695305