Title : Design, Synthesis, and In Vitro Biological Activities of a Bio-Oxidizable Prodrug to Deliver Both ChEs and DYRK1A Inhibitors for AD Therapy - Barre_2019_Molecules_24_ |
Author(s) : Barre A , Azzouz R , Gembus V , Papamicael C , Levacher V |
Ref : Molecules , 24 : , 2019 |
Abstract : |
PubMedSearch : Barre_2019_Molecules_24_ |
PubMedID: 30939771 |
Title : Donepezil-Based Central Acetylcholinesterase Inhibitors by Means of a Bio-Oxidizable Prodrug Strategy: Design, Synthesis, and in Vitro Biological Evaluation - Peauger_2017_J.Med.Chem_60_5909 |
Author(s) : Peauger L , Azzouz R , Gembus V , Tintas ML , Sopkova-de Oliveira Santos J , Bohn P , Papamicael C , Levacher V |
Ref : Journal of Medicinal Chemistry , 60 :5909 , 2017 |
Abstract : |
PubMedSearch : Peauger_2017_J.Med.Chem_60_5909 |
PubMedID: 28613859 |
Title : Dihydroquinoline Carbamate Derivatives as Bio-oxidizable Prodrugs for Brain Delivery of Acetylcholinesterase Inhibitors: [(11)C] Radiosynthesis and Biological Evaluation - Bohn_2015_ACS.Chem.Neurosci_6_737 |
Author(s) : Bohn P , Gourand F , Papamicael C , Ibazizene M , Dhilly M , Gembus V , Alix F , Tintas ML , Marsais F , Barre L , Levacher V |
Ref : ACS Chem Neurosci , 6 :737 , 2015 |
Abstract : |
PubMedSearch : Bohn_2015_ACS.Chem.Neurosci_6_737 |
PubMedID: 25695305 |
Title : New developments in redox chemical delivery systems by means of 1,4-dihydroquinoline-based targetor: Application to galantamine delivery to the brain - Tintas_2014_Eur.J.Med.Chem_81C_218 |
Author(s) : Tintas ML , Foucout L , Petit S , Oudeyer S , Gourand F , Barre L , Papamicael C , Levacher V |
Ref : Eur Journal of Medicinal Chemistry , 81C :218 , 2014 |
Abstract : |
PubMedSearch : Tintas_2014_Eur.J.Med.Chem_81C_218 |
PubMedID: 24852273 |
Title : Rational design of central selective acetylcholinesterase inhibitors by means of a bio-oxidisable prodrug strategy - Bohn_2009_Org.Biomol.Chem_7_2612 |
Author(s) : Bohn P , Le Fur N , Hagues G , Costentin J , Torquet N , Papamicael C , Marsais F , Levacher V |
Ref : Org Biomol Chem , 7 :2612 , 2009 |
Abstract : |
PubMedSearch : Bohn_2009_Org.Biomol.Chem_7_2612 |
PubMedID: 19503937 |