Title : AT-1001 Is a Partial Agonist with High Affinity and Selectivity at Human and Rat alpha3beta4 Nicotinic Cholinergic Receptors - Tuan_2015_Mol.Pharmacol_88_640 |
Author(s) : Tuan EW , Horti AG , Olson TT , Gao Y , Stockmeier CA , Al-Muhtasib N , Bowman Dalley C , Lewin AE , Wolfe BB , Sahibzada N , Xiao Y , Kellar KJ |
Ref : Molecular Pharmacology , 88 :640 , 2015 |
Abstract : |
PubMedSearch : Tuan_2015_Mol.Pharmacol_88_640 |
PubMedID: 26162864 |
Title : Structure-activity relationship studies of SEN12333 analogues: determination of the optimal requirements for binding affinities at alpha7 nAChRs through incorporation of known structural motifs - Beinat_2015_Eur.J.Med.Chem_95_277 |
Author(s) : Beinat C , Reekie T , Banister SD , O'Brien-Brown J , Xie T , Olson TT , Xiao Y , Harvey A , O'Connor S , Coles C , Grishin A , Kolesik P , Tsanaktsidis J , Kassiou M |
Ref : Eur Journal of Medicinal Chemistry , 95 :277 , 2015 |
Abstract : |
PubMedSearch : Beinat_2015_Eur.J.Med.Chem_95_277 |
PubMedID: 25827398 |
Title : Synthesis and pharmacological characterization of new neuronal nicotinic acetylcholine receptor ligands derived from Sazetidine-A - Liu_2014_Bioorg.Med.Chem.Lett_24_2954 |
Author(s) : Liu Y , Paige M , Olson TT , Al-Muhtasib N , Xie T , Hou S , White MP , Cordova A , Guo JL , Kellar KJ , Xiao Y , Brown ML |
Ref : Bioorganic & Medicinal Chemistry Lett , 24 :2954 , 2014 |
Abstract : |
PubMedSearch : Liu_2014_Bioorg.Med.Chem.Lett_24_2954 |
PubMedID: 24844195 |
Title : Investigations of amide bond variation and biaryl modification in analogues of alpha7 nAChR agonist SEN12333 - Beinat_2014_Eur.J.Med.Chem_84C_200 |
Author(s) : Beinat C , Reekie T , Hibbs D , Xie T , Olson TT , Xiao Y , Harvey A , O'Connor S , Coles C , Tsanaktsidis J , Kassiou M |
Ref : Eur Journal of Medicinal Chemistry , 84C :200 , 2014 |
Abstract : |
PubMedSearch : Beinat_2014_Eur.J.Med.Chem_84C_200 |
PubMedID: 25019477 |