Title : [(18)F]FNDP PET neuroimaging test-retest repeatability and whole-body dosimetry in humans - Du_2023_Eur.J.Nucl.Med.Mol.Imaging__ |
Author(s) : Du Y , Coughlin JM , Amindarolzarbi A , Sweeney SE , Harrington CK , Brosnan MK , Zandi A , Shinehouse LK , Sanchez ANR , Abdallah R , Holt DP , Fan H , Lesniak WG , Nandi A , Rowe SP , Solnes LB , Dannals RF , Horti AG , Lodge MA , Pomper MG |
Ref : Eur J Nucl Med Mol Imaging , : , 2023 |
Abstract : |
PubMedSearch : Du_2023_Eur.J.Nucl.Med.Mol.Imaging__ |
PubMedID: 37458759 |
Title : First-in-human neuroimaging of soluble epoxide hydrolase using [(18)F]FNDP PET - Coughlin_2021_Eur.J.Nucl.Med.Mol.Imaging__ |
Author(s) : Coughlin JM , Slania S , Du Y , Shinehouse LK , Brosnan MK , Azad BB , Holt DP , Fan H , Lesniak WG , Minn I , Rowe SP , Dannals RF , Horti AG , Pomper MG |
Ref : Eur J Nucl Med Mol Imaging , : , 2021 |
Abstract : |
PubMedSearch : Coughlin_2021_Eur.J.Nucl.Med.Mol.Imaging__ |
PubMedID: 33585963 |
Title : PET imaging of soluble epoxide hydrolase in non-human primate brain with [(18)F]FNDP - Du_2020_EJNMMI.Res_10_67 |
Author(s) : Du Y , Minn I , Foss C , Lesniak WG , Hu F , Dannals RF , Pomper MG , Horti AG |
Ref : EJNMMI Res , 10 :67 , 2020 |
Abstract : |
PubMedSearch : Du_2020_EJNMMI.Res_10_67 |
PubMedID: 32572592 |
Title : An optimized radiosynthesis of [(18) F]FNDP, a positron emission tomography radiotracer for imaging soluble epoxide hydrolase (sEH) - Azad_2018_J.Labelled.Comp.Radiopharm_61_567 |
Author(s) : Azad BB , Holt DP , Ravert HT , Horti AG , Dannals RF |
Ref : J Labelled Comp Radiopharm , 61 :567 , 2018 |
Abstract : |
PubMedSearch : Azad_2018_J.Labelled.Comp.Radiopharm_61_567 |
PubMedID: 29529708 |
Title : 18F-FNDP for PET Imaging of Soluble Epoxide Hydrolase - Horti_2016_J.Nucl.Med_57_1817 |
Author(s) : Horti AG , Wang Y , Minn I , Lan X , Wang J , Koehler RC , Alkayed NJ , Dannals RF , Pomper MG |
Ref : J Nucl Med , 57 :1817 , 2016 |
Abstract : |
PubMedSearch : Horti_2016_J.Nucl.Med_57_1817 |
PubMedID: 27417650 |
Title : Development of [(18)F]ASEM, a specific radiotracer for quantification of the alpha7-nAChR with positron-emission tomography - Horti_2015_Biochem.Pharmacol_97(4)_566 |
Author(s) : Horti AG |
Ref : Biochemical Pharmacology , 97 :566 , 2015 |
Abstract : |
PubMedSearch : Horti_2015_Biochem.Pharmacol_97(4)_566 |
PubMedID: 26232729 |
Title : AT-1001 Is a Partial Agonist with High Affinity and Selectivity at Human and Rat alpha3beta4 Nicotinic Cholinergic Receptors - Tuan_2015_Mol.Pharmacol_88_640 |
Author(s) : Tuan EW , Horti AG , Olson TT , Gao Y , Stockmeier CA , Al-Muhtasib N , Bowman Dalley C , Lewin AE , Wolfe BB , Sahibzada N , Xiao Y , Kellar KJ |
Ref : Molecular Pharmacology , 88 :640 , 2015 |
Abstract : |
PubMedSearch : Tuan_2015_Mol.Pharmacol_88_640 |
PubMedID: 26162864 |
Title : 18F-ASEM, a radiolabeled antagonist for imaging the alpha7-nicotinic acetylcholine receptor with PET - Horti_2014_J.Nucl.Med_55_672 |
Author(s) : Horti AG , Gao Y , Kuwabara H , Wang Y , Abazyan S , Yasuda RP , Tran T , Xiao Y , Sahibzada N , Holt DP , Kellar KJ , Pletnikov MV , Pomper MG , Wong DF , Dannals RF |
Ref : J Nucl Med , 55 :672 , 2014 |
Abstract : |
PubMedSearch : Horti_2014_J.Nucl.Med_55_672 |
PubMedID: 24556591 |
Title : Derivatives of dibenzothiophene for positron emission tomography imaging of alpha7-nicotinic acetylcholine receptors - Gao_2013_J.Med.Chem_56_7574 |
Author(s) : Gao Y , Kellar KJ , Yasuda RP , Tran T , Xiao Y , Dannals RF , Horti AG |
Ref : Journal of Medicinal Chemistry , 56 :7574 , 2013 |
Abstract : |
PubMedSearch : Gao_2013_J.Med.Chem_56_7574 |
PubMedID: 24050653 |
Title : Discovery of (-)-7-methyl-2-exo-[3'-(6-[18F]fluoropyridin-2-yl)-5'-pyridinyl]-7-azabicyclo[2.2 .1]heptane, a radiolabeled antagonist for cerebral nicotinic acetylcholine receptor (alpha4beta2-nAChR) with optimal positron emission tomography imaging properties - Gao_2008_J.Med.Chem_51_4751 |
Author(s) : Gao Y , Kuwabara H , Spivak CE , Xiao Y , Kellar K , Ravert HT , Kumar A , Alexander M , Hilton J , Wong DF , Dannals RF , Horti AG |
Ref : Journal of Medicinal Chemistry , 51 :4751 , 2008 |
Abstract : |
PubMedSearch : Gao_2008_J.Med.Chem_51_4751 |
PubMedID: 18605717 |
Title : In vitro characterization of 6-[18F]fluoro-A-85380, a high-affinity ligand for alpha4beta2* nicotinic acetylcholine receptors - Gundisch_2005_Synapse_55_89 |
Author(s) : Gundisch D , Koren AO , Horti AG , Pavlova OA , Kimes AS , Mukhin AG , London ED |
Ref : Synapse , 55 :89 , 2005 |
Abstract : |
PubMedSearch : Gundisch_2005_Synapse_55_89 |
PubMedID: 15529332 |
Title : Pharmacological and toxicological evaluation of 2-fluoro-3-(2(S)-azetidinylmethoxy)pyridine (2-F-A-85380), a ligand for imaging cerebral nicotinic acetylcholine receptors with positron emission tomography - Vaupel_2005_J.Pharmacol.Exp.Ther_312_355 |
Author(s) : Vaupel DB , Tella SR , Huso DL , Wagner VO, 3rd , Mukhin AG , Chefer SI , Horti AG , London ED , Koren AO , Kimes AS |
Ref : Journal of Pharmacology & Experimental Therapeutics , 312 :355 , 2005 |
Abstract : |
PubMedSearch : Vaupel_2005_J.Pharmacol.Exp.Ther_312_355 |
PubMedID: 15331657 |
Title : Graphical analysis of 2-[18F]FA binding to nicotinic acetylcholine receptors in rhesus monkey brain - Chefer_2003_Synapse_48_25 |
Author(s) : Chefer SI , London ED , Koren AO , Pavlova OA , Kurian V , Kimes AS , Horti AG , Mukhin AG |
Ref : Synapse , 48 :25 , 2003 |
Abstract : |
PubMedSearch : Chefer_2003_Synapse_48_25 |
PubMedID: 12557269 |
Title : 2-[18F]F-A-85380: PET imaging of brain nicotinic acetylcholine receptors and whole body distribution in humans - Kimes_2003_FASEB.J_17_1331 |
Author(s) : Kimes AS , Horti AG , London ED , Chefer SI , Contoreggi C , Ernst M , Friello P , Koren AO , Kurian V , Matochik JA , Pavlova O , Vaupel DB , Mukhin AG |
Ref : FASEB Journal , 17 :1331 , 2003 |
Abstract : |
PubMedSearch : Kimes_2003_FASEB.J_17_1331 |
PubMedID: 12759330 |
Title : Quantification of nicotinic acetylcholine receptors in human brain using [123I]5-I-A-85380 SPET - Fujita_2003_Eur.J.Nucl.Med.Mol.Imaging_30_1620 |
Author(s) : Fujita M , Ichise M , van Dyck CH , Zoghbi SS , Tamagnan G , Mukhin AG , Bozkurt A , Seneca N , Tipre D , DeNucci CC , Iida H , Vaupel DB , Horti AG , Koren AO , Kimes AS , London ED , Seibyl JP , Baldwin RM , Innis RB |
Ref : Eur J Nucl Med Mol Imaging , 30 :1620 , 2003 |
Abstract : |
PubMedSearch : Fujita_2003_Eur.J.Nucl.Med.Mol.Imaging_30_1620 |
PubMedID: 14523584 |
Title : Whole-body biodistribution, radiation absorbed dose, and brain SPET imaging with [123i]5-i-A-85380 in healthy human subjects - Fujita_2002_Eur.J.Nucl.Med.Mol.Imaging_29_183 |
Author(s) : Fujita M , Seibyl JP , Vaupel DB , Tamagnan G , Early M , Zoghbi SS , Baldwin RM , Horti AG , Kore NA , Mukhin AG , Khan S , Bozkurt A , Kimes AS , London ED , Innis RB |
Ref : Eur J Nucl Med Mol Imaging , 29 :183 , 2002 |
Abstract : |
PubMedSearch : Fujita_2002_Eur.J.Nucl.Med.Mol.Imaging_29_183 |
PubMedID: 11926380 |
Title : 6-[18F]Fluoro-A-85380: an in vivo tracer for the nicotinic acetylcholine receptor - Scheffel_2000_Nucl.Med.Biol_27_51 |
Author(s) : Scheffel U , Horti AG , Koren AO , Ravert HT , Banta JP , Finley PA , London ED , Dannals RF |
Ref : Nucl Med Biol , 27 :51 , 2000 |
Abstract : |
PubMedSearch : Scheffel_2000_Nucl.Med.Biol_27_51 |
PubMedID: 10755645 |
Title : 6-[18F]fluoro-A-85380, a novel radioligand for in vivo imaging of central nicotinic acetylcholine receptors - Horti_2000_Life.Sci_67_463 |
Author(s) : Horti AG , Chefer SI , Mukhin AG , Koren AO , Gundisch D , Links JM , Kurian V , Dannals RF , London ED |
Ref : Life Sciences , 67 :463 , 2000 |
Abstract : |
PubMedSearch : Horti_2000_Life.Sci_67_463 |
PubMedID: 11003056 |
Title : 5-Iodo-A-85380, an alpha4beta2 subtype-selective ligand for nicotinic acetylcholine receptors - Mukhin_2000_Mol.Pharmacol_57_642 |
Author(s) : Mukhin AG , Gundisch D , Horti AG , Koren AO , Tamagnan G , Kimes AS , Chambers J , Vaupel DB , King SL , Picciotto MR , Innis RB , London ED |
Ref : Molecular Pharmacology , 57 :642 , 2000 |
Abstract : |
PubMedSearch : Mukhin_2000_Mol.Pharmacol_57_642 |
PubMedID: 10692507 |
Title : Synthesis and characterization of binding of 5-[76Br]bromo-3-[[2(S)-azetidinyl]methoxy]pyridine, a novel nicotinic acetylcholine receptor ligand, in rat brain - Sihver_1999_J.Neurochem_73_1264 |
Author(s) : Sihver W , Fasth KJ , Horti AG , Koren AO , Bergstrom M , Lu L , Hagberg G , Lundqvist H , Dannals RF , London ED , Nordberg A , Langstrom B |
Ref : Journal of Neurochemistry , 73 :1264 , 1999 |
Abstract : |
PubMedSearch : Sihver_1999_J.Neurochem_73_1264 |
PubMedID: 10461920 |
Title : 2-[18F]F-A-85380: a PET radioligand for alpha4beta2 nicotinic acetylcholine receptors - Chefer_1999_Neuroreport_10_2715 |
Author(s) : Chefer SI , Horti AG , Koren AO , Gundisch D , Links JM , Kurian V , Dannals RF , Mukhin AG , London ED |
Ref : Neuroreport , 10 :2715 , 1999 |
Abstract : |
PubMedSearch : Chefer_1999_Neuroreport_10_2715 |
PubMedID: 10511429 |
Title : Radiosynthesis and preliminary evaluation of 5-[123\/125I]iodo-3-(2(S)-azetidinylmethoxy)pyridine: a radioligand for nicotinic acetylcholine receptors - Horti_1999_Nucl.Med.Biol_26_175 |
Author(s) : Horti AG , Koren AO , Lee KS , Mukhin AG , Vaupel DB , Kimes AS , Stratton M , London ED |
Ref : Nucl Med Biol , 26 :175 , 1999 |
Abstract : |
PubMedSearch : Horti_1999_Nucl.Med.Biol_26_175 |
PubMedID: 10100216 |
Title : In vivo studies with [125I]5-I-A-85380, a nicotinic acetylcholine receptor radioligand - Vaupel_1998_Neuroreport_9_2311 |
Author(s) : Vaupel DB , Mukhin AG , Kimes AS , Horti AG , Koren AO , London ED |
Ref : Neuroreport , 9 :2311 , 1998 |
Abstract : |
PubMedSearch : Vaupel_1998_Neuroreport_9_2311 |
PubMedID: 9694220 |
Title : In vivo imaging of brain nicotinic acetylcholine receptors with 5-[123I]iodo-A-85380 using single photon emission computed tomography - Chefer_1998_Life.Sci_63_PL355 |
Author(s) : Chefer SI , Horti AG , Lee KS , Koren AO , Jones DW , Gorey JG , Links JM , Mukhin AG , Weinberger DR , London ED |
Ref : Life Sciences , 63 :PL355 , 1998 |
Abstract : |
PubMedSearch : Chefer_1998_Life.Sci_63_PL355 |
PubMedID: 9870715 |
Title : Synthesis and evaluation of N-[11C]methylated analogues of epibatidine as tracers for positron emission tomographic studies of nicotinic acetylcholine receptors - Horti_1998_J.Med.Chem_41_4199 |
Author(s) : Horti AG , Scheffel U , Kimes AS , Musachio JL , Ravert HT , Mathews WB , Zhan Y , Finley PA , London ED , Dannals RF |
Ref : Journal of Medicinal Chemistry , 41 :4199 , 1998 |
Abstract : |
PubMedSearch : Horti_1998_J.Med.Chem_41_4199 |
PubMedID: 9784094 |
Title : 2-[18F]Fluoro-A-85380, an in vivo tracer for the nicotinic acetylcholine receptors - Horti_1998_Nucl.Med.Biol_25_599 |
Author(s) : Horti AG , Scheffel U , Koren AO , Ravert HT , Mathews WB , Musachio JL , Finley PA , London ED , Dannals RF |
Ref : Nucl Med Biol , 25 :599 , 1998 |
Abstract : |
PubMedSearch : Horti_1998_Nucl.Med.Biol_25_599 |
PubMedID: 9804040 |
Title : 2-, 5-, and 6-Halo-3-(2(S)-azetidinylmethoxy)pyridines: synthesis, affinity for nicotinic acetylcholine receptors, and molecular modeling - Koren_1998_J.Med.Chem_41_3690 |
Author(s) : Koren AO , Horti AG , Mukhin AG , Gundisch D , Kimes AS , Dannals RF , London ED |
Ref : Journal of Medicinal Chemistry , 41 :3690 , 1998 |
Abstract : |
PubMedSearch : Koren_1998_J.Med.Chem_41_3690 |
PubMedID: 9733494 |