Full name : Kellar Kenneth J
First name : Kenneth J
Mail : Department of Pharmacology and Physiology, Georgetown University School of Medicine, Washington, D. C. 20057
Zip Code :
City :
Country : USA
Email : kellark@georgetown.edu
Phone : 202-687-1032
Fax :
Website :
Directory :
Comment
| Title : Poster: Nicotinic treatments not only for tobacco, but also other addictions - |
| Author(s) : Levin ED , Rezvani AH , Xiao Y , Yenugonda VM , Brown ML , Kellar KJ |
| Ref : Biochemical Pharmacology , 97 :635 , 2015 |
| PubMedID: |
| Title : AT-1001 Is a Partial Agonist with High Affinity and Selectivity at Human and Rat alpha3beta4 Nicotinic Cholinergic Receptors - Tuan_2015_Mol.Pharmacol_88_640 |
| Author(s) : Tuan EW , Horti AG , Olson TT , Gao Y , Stockmeier CA , Al-Muhtasib N , Bowman Dalley C , Lewin AE , Wolfe BB , Sahibzada N , Xiao Y , Kellar KJ |
| Ref : Molecular Pharmacology , 88 :640 , 2015 |
| Abstract : |
| PubMedSearch : Tuan_2015_Mol.Pharmacol_88_640 |
| PubMedID: 26162864 |
| Title : Chronic sazetidine-A maintains anxiolytic effects and slower weight gain following chronic nicotine without maintaining increased density of nicotinic receptors in rodent brain - Hussmann_2014_J.Neurochem_129_721 |
| Author(s) : Hussmann GP , DeDominicis KE , Turner JR , Yasuda RP , Klehm J , Forcelli PA , Xiao Y , Richardson JR , Sahibzada N , Wolfe BB , Lindstrom JM , Blendy JA , Kellar KJ |
| Ref : Journal of Neurochemistry , 129 :721 , 2014 |
| Abstract : |
| PubMedSearch : Hussmann_2014_J.Neurochem_129_721 |
| PubMedID: 24422997 |
| Title : 18F-ASEM, a radiolabeled antagonist for imaging the alpha7-nicotinic acetylcholine receptor with PET - Horti_2014_J.Nucl.Med_55_672 |
| Author(s) : Horti AG , Gao Y , Kuwabara H , Wang Y , Abazyan S , Yasuda RP , Tran T , Xiao Y , Sahibzada N , Holt DP , Kellar KJ , Pletnikov MV , Pomper MG , Wong DF , Dannals RF |
| Ref : J Nucl Med , 55 :672 , 2014 |
| Abstract : |
| PubMedSearch : Horti_2014_J.Nucl.Med_55_672 |
| PubMedID: 24556591 |
| Title : Synthesis and pharmacological characterization of new neuronal nicotinic acetylcholine receptor ligands derived from Sazetidine-A - Liu_2014_Bioorg.Med.Chem.Lett_24_2954 |
| Author(s) : Liu Y , Paige M , Olson TT , Al-Muhtasib N , Xie T , Hou S , White MP , Cordova A , Guo JL , Kellar KJ , Xiao Y , Brown ML |
| Ref : Bioorganic & Medicinal Chemistry Lett , 24 :2954 , 2014 |
| Abstract : |
| PubMedSearch : Liu_2014_Bioorg.Med.Chem.Lett_24_2954 |
| PubMedID: 24844195 |
| Title : Design, synthesis and discovery of picomolar selective alpha4beta2 nicotinic acetylcholine receptor ligands - Yenugonda_2013_J.Med.Chem_56_8404 |
| Author(s) : Yenugonda VM , Xiao Y , Levin ED , Rezvani AH , Tran T , Al-Muhtasib N , Sahibzada N , Xie T , Wells C , Slade S , Johnson JE , Dakshanamurthy S , Kong HS , Tomita Y , Liu Y , Paige M , Kellar KJ , Brown ML |
| Ref : Journal of Medicinal Chemistry , 56 :8404 , 2013 |
| Abstract : |
| PubMedSearch : Yenugonda_2013_J.Med.Chem_56_8404 |
| PubMedID: 24047231 |
| Title : Derivatives of dibenzothiophene for positron emission tomography imaging of alpha7-nicotinic acetylcholine receptors - Gao_2013_J.Med.Chem_56_7574 |
| Author(s) : Gao Y , Kellar KJ , Yasuda RP , Tran T , Xiao Y , Dannals RF , Horti AG |
| Ref : Journal of Medicinal Chemistry , 56 :7574 , 2013 |
| Abstract : |
| PubMedSearch : Gao_2013_J.Med.Chem_56_7574 |
| PubMedID: 24050653 |
| Title : Effects of the sazetidine-a family of compounds on the body temperature in wildtype, nicotinic receptor beta2-\/- and alpha7-\/- mice - Levin_2013_Eur.J.Pharmacol_718_167 |
| Author(s) : Levin ED , Sexton HG , Gordon K , Gordon CJ , Xiao Y , Kellar KJ , Yenugonda VM , Liu Y , White MP , Paige M , Brown ML , Rezvani AH |
| Ref : European Journal of Pharmacology , 718 :167 , 2013 |
| Abstract : |
| PubMedSearch : Levin_2013_Eur.J.Pharmacol_718_167 |
| PubMedID: 24036108 |
| Title : Chemistry and pharmacological studies of 3-alkoxy-2,5-disubstituted-pyridinyl compounds as novel selective alpha4beta2 nicotinic acetylcholine receptor ligands that reduce alcohol intake in rats - Liu_2013_J.Med.Chem_56_3000 |
| Author(s) : Liu Y , Richardson J , Tran T , Al-Muhtasib N , Xie T , Yenugonda VM , Sexton HG , Rezvani AH , Levin ED , Sahibzada N , Kellar KJ , Brown ML , Xiao Y , Paige M |
| Ref : Journal of Medicinal Chemistry , 56 :3000 , 2013 |
| Abstract : |
| PubMedSearch : Liu_2013_J.Med.Chem_56_3000 |
| PubMedID: 23540678 |
| Title : Effects of chronic sazetidine-A, a selective alpha4beta2 neuronal nicotinic acetylcholine receptors desensitizing agent on pharmacologically-induced impaired attention in rats - Rezvani_2013_Psychopharmacology.(Berl)_226_35 |
| Author(s) : Rezvani AH , Cauley M , Xiao Y , Kellar KJ , Levin ED |
| Ref : Psychopharmacology (Berl) , 226 :35 , 2013 |
| Abstract : |
| PubMedSearch : Rezvani_2013_Psychopharmacology.(Berl)_226_35 |
| PubMedID: 23100170 |
| Title : Chronic sazetidine-A at behaviorally active doses does not increase nicotinic cholinergic receptors in rodent brain - Hussmann_2012_J.Pharmacol.Exp.Ther_343_441 |
| Author(s) : Hussmann GP , Turner JR , Lomazzo E , Venkatesh R , Cousins V , Xiao Y , Yasuda RP , Wolfe BB , Perry DC , Rezvani AH , Levin ED , Blendy JA , Kellar KJ |
| Ref : Journal of Pharmacology & Experimental Therapeutics , 343 :441 , 2012 |
| Abstract : |
| PubMedSearch : Hussmann_2012_J.Pharmacol.Exp.Ther_343_441 |
| PubMedID: 22899752 |
| Title : Assessing the effects of chronic sazetidine-A delivery on nicotine self-administration in both male and female rats - Johnson_2012_Psychopharmacology.(Berl)_222_269 |
| Author(s) : Johnson JE , Slade S , Wells C , Petro A , Sexton H , Rezvani AH , Brown ML , Paige MA , McDowell BE , Xiao Y , Kellar KJ , Levin ED |
| Ref : Psychopharmacology (Berl) , 222 :269 , 2012 |
| Abstract : |
| PubMedSearch : Johnson_2012_Psychopharmacology.(Berl)_222_269 |
| PubMedID: 22297831 |
| Title : Effects of sazetidine-A, a selective alpha4beta2* nicotinic receptor desensitizing agent, on body temperature regulation in mice and rats - Rezvani_2012_Eur.J.Pharmacol_682_110 |
| Author(s) : Rezvani AH , Timofeeva O , Sexton HG , DeCuir D , Xiao Y , Gordon CJ , Kellar KJ , Levin ED |
| Ref : European Journal of Pharmacology , 682 :110 , 2012 |
| Abstract : |
| PubMedSearch : Rezvani_2012_Eur.J.Pharmacol_682_110 |
| PubMedID: 22387853 |
| Title : Effects of chronic nicotine on heteromeric neuronal nicotinic receptors in rat primary cultured neurons - Lomazzo_2011_J.Neurochem_119_153 |
| Author(s) : Lomazzo E , Hussmann GP , Wolfe BB , Yasuda RP , Perry DC , Kellar KJ |
| Ref : Journal of Neurochemistry , 119 :153 , 2011 |
| Abstract : |
| PubMedSearch : Lomazzo_2011_J.Neurochem_119_153 |
| PubMedID: 21806615 |
| Title : Poster: Pharmacological properties of sazetidine A, a selective ligand of alpha4\/beta2 nicotinic acetylcholine receptors - |
| Author(s) : Xiao Y , Tuan E , Yasuda RP , Sahibzada N , Wolfe BB , Horton L , Tran T , Al-Muhtasib N , Iwueze AF , Dipietro JR , Xie T , Paige M , Brown ML , Kellar KJ |
| Ref : Biochemical Pharmacology , 82 :1029 , 2011 |
| PubMedID: |
| Title : Endogenously expressed muscarinic receptors in HEK293 cells augment up-regulation of stably expressed alpha4beta2 nicotinic receptors - Hussmann_2011_J.Biol.Chem_286_39726 |
| Author(s) : Hussmann GP , Yasuda RP , Xiao Y , Wolfe BB , Kellar KJ |
| Ref : Journal of Biological Chemistry , 286 :39726 , 2011 |
| Abstract : |
| PubMedSearch : Hussmann_2011_J.Biol.Chem_286_39726 |
| PubMedID: 21940627 |
| Title : Sazetidine-A, a selective alpha4beta2 nicotinic acetylcholine receptor ligand: effects on dizocilpine and scopolamine-induced attentional impairments in female Sprague-Dawley rats - Rezvani_2011_Psychopharmacology.(Berl)_215_621 |
| Author(s) : Rezvani AH , Cauley M , Sexton H , Xiao Y , Brown ML , Paige MA , McDowell BE , Kellar KJ , Levin ED |
| Ref : Psychopharmacology (Berl) , 215 :621 , 2011 |
| Abstract : |
| PubMedSearch : Rezvani_2011_Psychopharmacology.(Berl)_215_621 |
| PubMedID: 21274704 |
| Title : Quantitative analysis of the heteromeric neuronal nicotinic receptors in the rat hippocampus - Lomazzo_2010_J.Neurochem_115_625 |
| Author(s) : Lomazzo E , MacArthur L , Yasuda RP , Wolfe BB , Kellar KJ |
| Ref : Journal of Neurochemistry , 115 :625 , 2010 |
| Abstract : |
| PubMedSearch : Lomazzo_2010_J.Neurochem_115_625 |
| PubMedID: 20796176 |
| Title : Sazetidine-A, a selective alpha4beta2 nicotinic receptor desensitizing agent and partial agonist, reduces nicotine self-administration in rats - Levin_2010_J.Pharmacol.Exp.Ther_332_933 |
| Author(s) : Levin ED , Rezvani AH , Xiao Y , Slade S , Cauley M , Wells C , Hampton D , Petro A , Rose JE , Brown ML , Paige MA , McDowell BE , Kellar KJ |
| Ref : Journal of Pharmacology & Experimental Therapeutics , 332 :933 , 2010 |
| Abstract : |
| PubMedSearch : Levin_2010_J.Pharmacol.Exp.Ther_332_933 |
| PubMedID: 20007754 |
| Title : Effects of sazetidine-A, a selective alpha4beta2 nicotinic acetylcholine receptor desensitizing agent on alcohol and nicotine self-administration in selectively bred alcohol-preferring (P) rats - Rezvani_2010_Psychopharmacology.(Berl)_211_161 |
| Author(s) : Rezvani AH , Slade S , Wells C , Petro A , Lumeng L , Li TK , Xiao Y , Brown ML , Paige MA , McDowell BE , Rose JE , Kellar KJ , Levin ED |
| Ref : Psychopharmacology (Berl) , 211 :161 , 2010 |
| Abstract : |
| PubMedSearch : Rezvani_2010_Psychopharmacology.(Berl)_211_161 |
| PubMedID: 20535453 |
| Title : Rat neuronal nicotinic acetylcholine receptors containing alpha7 subunit: pharmacological properties of ligand binding and function - Xiao_2009_Acta.Pharmacol.Sin_30_842 |
| Author(s) : Xiao Y , Abdrakhmanova GR , Baydyuk M , Hernandez S , Kellar KJ |
| Ref : Acta Pharmacol Sin , 30 :842 , 2009 |
| Abstract : |
| PubMedSearch : Xiao_2009_Acta.Pharmacol.Sin_30_842 |
| PubMedID: 19448648 |
| Title : 18F-ZW-104: a new radioligand for imaging neuronal nicotinic acetylcholine receptors--in vitro binding properties and PET studies in baboons - Valette_2009_J.Nucl.Med_50_1349 |
| Author(s) : Valette H , Xiao Y , Peyronneau MA , Damont A , Kozikowski AP , Wei ZL , Kassiou M , Kellar KJ , Dolle F , Bottlaender M |
| Ref : J Nucl Med , 50 :1349 , 2009 |
| Abstract : |
| PubMedSearch : Valette_2009_J.Nucl.Med_50_1349 |
| PubMedID: 19652217 |
| Title : The alpha4beta2alpha5 nicotinic cholinergic receptor in rat brain is resistant to up-regulation by nicotine in vivo - Mao_2008_J.Neurochem_104_446 |
| Author(s) : Mao D , Perry DC , Yasuda RP , Wolfe BB , Kellar KJ |
| Ref : Journal of Neurochemistry , 104 :446 , 2008 |
| Abstract : |
| PubMedSearch : Mao_2008_J.Neurochem_104_446 |
| PubMedID: 17961152 |
| Title : Toxicological analysis of low-nicotine and nicotine-free cigarettes - Chen_2008_Toxicology_249_194 |
| Author(s) : Chen J , Higby R , Tian D , Tan D , Johnson MD , Xiao Y , Kellar KJ , Feng S , Shields PG |
| Ref : Toxicology , 249 :194 , 2008 |
| Abstract : |
| PubMedSearch : Chen_2008_Toxicology_249_194 |
| PubMedID: 18599178 |
| Title : Analgesic effects of Sazetidine-A, a new nicotinic cholinergic drug - Cucchiaro_2008_Anesthesiology_109_512 |
| Author(s) : Cucchiaro G , Xiao Y , Gonzalez-Sulser A , Kellar KJ |
| Ref : Anesthesiology , 109 :512 , 2008 |
| Abstract : |
| PubMedSearch : Cucchiaro_2008_Anesthesiology_109_512 |
| PubMedID: 18719450 |
| Title : Initial synthesis and characterization of an alpha7 nicotinic receptor cellular membrane affinity chromatography column: effect of receptor subtype and cell type - Moaddel_2008_Anal.Chem_80_48 |
| Author(s) : Moaddel R , Oliveira RV , Kimura T , Hyppolite P , Juhaszova M , Xiao Y , Kellar KJ , Bernier M , Wainer IW |
| Ref : Analytical Chemistry , 80 :48 , 2008 |
| Abstract : |
| PubMedSearch : Moaddel_2008_Anal.Chem_80_48 |
| PubMedID: 18062706 |
| Title : Chronic nicotine differentially regulates alpha6- and beta3-containing nicotinic cholinergic receptors in rat brain - Perry_2007_J.Pharmacol.Exp.Ther_322_306 |
| Author(s) : Perry DC , Mao D , Gold AB , McIntosh JM , Pezzullo JC , Kellar KJ |
| Ref : Journal of Pharmacology & Experimental Therapeutics , 322 :306 , 2007 |
| Abstract : |
| PubMedSearch : Perry_2007_J.Pharmacol.Exp.Ther_322_306 |
| PubMedID: 17446303 |
| Title : Acetylenic pyridines for use in PET imaging of nicotinic receptors - |
| Author(s) : Kozikowski AP , Chellappan SK , Henderson D , Fulton R , Giboureau N , Xiao Y , Wei ZL , Guilloteau D , Emond P , Dolle F , Kellar KJ , Kassiou M |
| Ref : ChemMedChem , 2 :54 , 2007 |
| PubMedID: 17096450 |
| Title : Chemical medicine: novel 10-substituted cytisine derivatives with increased selectivity for alpha4beta2 nicotinic acetylcholine receptors - |
| Author(s) : Kozikowski AP , Chellappan SK , Xiao Y , Bajjuri KM , Yuan H , Kellar KJ , Petukhov PA |
| Ref : ChemMedChem , 2 :1157 , 2007 |
| PubMedID: 17530728 |
| Title : Heterogeneity of nicotinic cholinergic receptors in rat superior cervical and nodose Ganglia - Mao_2006_Mol.Pharmacol_70_1693 |
| Author(s) : Mao D , Yasuda RP , Fan H , Wolfe BB , Kellar KJ |
| Ref : Molecular Pharmacology , 70 :1693 , 2006 |
| Abstract : |
| PubMedSearch : Mao_2006_Mol.Pharmacol_70_1693 |
| PubMedID: 16882879 |
| Title : Synthesis and pharmacological evaluation of novel 9- and 10-substituted cytisine derivatives. Nicotinic ligands of enhanced subtype selectivity - Chellappan_2006_J.Med.Chem_49_2673 |
| Author(s) : Chellappan SK , Xiao Y , Tueckmantel W , Kellar KJ , Kozikowski AP |
| Ref : Journal of Medicinal Chemistry , 49 :2673 , 2006 |
| Abstract : |
| PubMedSearch : Chellappan_2006_J.Med.Chem_49_2673 |
| PubMedID: 16640326 |
| Title : Mouse beta-TC6 insulinoma cells: high expression of functional alpha3beta4 nicotinic receptors mediating membrane potential, intracellular calcium, and insulin release - Ohtani_2006_Mol.Pharmacol_69_899 |
| Author(s) : Ohtani M , Oka T , Badyuk M , Xiao Y , Kellar KJ , Daly JW |
| Ref : Molecular Pharmacology , 69 :899 , 2006 |
| Abstract : |
| PubMedSearch : Ohtani_2006_Mol.Pharmacol_69_899 |
| PubMedID: 16332988 |
| Title : Sazetidine-A, a novel ligand that desensitizes alpha4beta2 nicotinic acetylcholine receptors without activating them - Xiao_2006_Mol.Pharmacol_70_1454 |
| Author(s) : Xiao Y , Fan H , Musachio JL , Wei ZL , Chellappan SK , Kozikowski AP , Kellar KJ |
| Ref : Molecular Pharmacology , 70 :1454 , 2006 |
| Abstract : |
| PubMedSearch : Xiao_2006_Mol.Pharmacol_70_1454 |
| PubMedID: 16857741 |
| Title : Novel pyridyl ring C5 substituted analogues of epibatidine and 3-(1-methyl-2(S)-pyrrolidinylmethoxy)pyridine (A-84543) as highly selective agents for neuronal nicotinic acetylcholine receptors containing beta2 subunits - Wei_2005_J.Med.Chem_48_1721 |
| Author(s) : Wei ZL , Xiao Y , Yuan H , Baydyuk M , Petukhov PA , Musachio JL , Kellar KJ , Kozikowski AP |
| Ref : Journal of Medicinal Chemistry , 48 :1721 , 2005 |
| Abstract : |
| PubMedSearch : Wei_2005_J.Med.Chem_48_1721 |
| PubMedID: 15771418 |
| Title : Nicotinic cholinergic receptors in the rat retina: simple and mixed heteromeric subtypes - Marritt_2005_Mol.Pharmacol_68_1656 |
| Author(s) : Marritt AM , Cox BC , Yasuda RP , McIntosh JM , Xiao Y , Wolfe BB , Kellar KJ |
| Ref : Molecular Pharmacology , 68 :1656 , 2005 |
| Abstract : |
| PubMedSearch : Marritt_2005_Mol.Pharmacol_68_1656 |
| PubMedID: 16129735 |
| Title : Nicotinic cholinergic receptors in the rat cerebellum: multiple heteromeric subtypes - Turner_2005_J.Neurosci_25_9258 |
| Author(s) : Turner JR , Kellar KJ |
| Ref : Journal of Neuroscience , 25 :9258 , 2005 |
| Abstract : |
| PubMedSearch : Turner_2005_J.Neurosci_25_9258 |
| PubMedID: 16207885 |
| Title : The biology of tobacco and nicotine: bench to bedside - Dennis_2005_Cancer.Epidemiol.Biomarkers.Prev_14_764 |
| Author(s) : Dennis PA , Van Waes C , Gutkind JS , Kellar KJ , Vinson C , Mukhin AG , Spitz MR , Bailey-Wilson JE , Yeh GC , Anderson LM , Wiest JS |
| Ref : Cancer Epidemiol Biomarkers Prev , 14 :764 , 2005 |
| Abstract : |
| PubMedSearch : Dennis_2005_Cancer.Epidemiol.Biomarkers.Prev_14_764 |
| PubMedID: 15824140 |
| Title : The nicotinic receptor in the rat pineal gland is an alpha3beta4 subtype - Hernandez_2004_Mol.Pharmacol_66_978 |
| Author(s) : Hernandez SC , Vicini S , Xiao Y , Davila-Garcia MI , Yasuda RP , Wolfe BB , Kellar KJ |
| Ref : Molecular Pharmacology , 66 :978 , 2004 |
| Abstract : |
| PubMedSearch : Hernandez_2004_Mol.Pharmacol_66_978 |
| PubMedID: 15247319 |
| Title : Synthesis and pharmacological characterization of bivalent ligands of epibatidine at neuronal nicotinic acetylcholine receptors - Wei_2004_Bioorg.Med.Chem.Lett_14_1855 |
| Author(s) : Wei ZL , Xiao Y , Kellar KJ , Kozikowski AP |
| Ref : Bioorganic & Medicinal Chemistry Lett , 14 :1855 , 2004 |
| Abstract : |
| PubMedSearch : Wei_2004_Bioorg.Med.Chem.Lett_14_1855 |
| PubMedID: 15050615 |
| Title : Pharmacology of the agonist binding sites of rat neuronal nicotinic receptor subtypes expressed in HEK 293 cells - Xiao_2004_Bioorg.Med.Chem.Lett_14_1845 |
| Author(s) : Xiao Y , Baydyuk M , Wang HP , Davis HE , Kellar KJ |
| Ref : Bioorganic & Medicinal Chemistry Lett , 14 :1845 , 2004 |
| Abstract : |
| PubMedSearch : Xiao_2004_Bioorg.Med.Chem.Lett_14_1845 |
| PubMedID: 15050613 |
| Title : The comparative pharmacology and up-regulation of rat neuronal nicotinic receptor subtype binding sites stably expressed in transfected mammalian cells - Xiao_2004_J.Pharmacol.Exp.Ther_310_98 |
| Author(s) : Xiao Y , Kellar KJ |
| Ref : Journal of Pharmacology & Experimental Therapeutics , 310 :98 , 2004 |
| Abstract : |
| PubMedSearch : Xiao_2004_J.Pharmacol.Exp.Ther_310_98 |
| PubMedID: 15016836 |
| Title : Differential regulation of nicotinic acetylcholine receptors in PC12 cells by nicotine and nerve growth factor - Avila_2003_Mol.Pharmacol_64_974 |
| Author(s) : Avila AM , Davila-Garcia MI , Ascarrunz VS , Xiao Y , Kellar KJ |
| Ref : Molecular Pharmacology , 64 :974 , 2003 |
| Abstract : |
| PubMedSearch : Avila_2003_Mol.Pharmacol_64_974 |
| PubMedID: 14500754 |
| Title : Membrane potential fluorescence: a rapid and highly sensitive assay for nicotinic receptor channel function - Fitch_2003_Proc.Natl.Acad.Sci.U.S.A_100_4909 |
| Author(s) : Fitch RW , Xiao Y , Kellar KJ , Daly JW |
| Ref : Proc Natl Acad Sci U S A , 100 :4909 , 2003 |
| Abstract : |
| PubMedSearch : Fitch_2003_Proc.Natl.Acad.Sci.U.S.A_100_4909 |
| PubMedID: 12657731 |
| Title : Enantioselective interactions of dextromethorphan and levomethorphan with the alpha 3 beta 4-nicotinic acetylcholine receptor: comparison of chromatographic and functional data - Jozwiak_2003_J.Chromatogr.B.Analyt.Technol.Biomed.Life.Sci_797_373 |
| Author(s) : Jozwiak K , Hernandez SC , Kellar KJ , Wainer IW |
| Ref : Journal of Chromatography B Analyt Technol Biomed Life Sciences , 797 :373 , 2003 |
| Abstract : |
| PubMedSearch : Jozwiak_2003_J.Chromatogr.B.Analyt.Technol.Biomed.Life.Sci_797_373 |
| PubMedID: 14630163 |
| Title : Synthesis, nicotinic acetylcholine receptor binding affinities, and molecular modeling of constrained epibatidine analogues - Wei_2003_J.Med.Chem_46_921 |
| Author(s) : Wei ZL , Petukhov PA , Xiao Y , Tuckmantel W , George C , Kellar KJ , Kozikowski AP |
| Ref : Journal of Medicinal Chemistry , 46 :921 , 2003 |
| Abstract : |
| PubMedSearch : Wei_2003_J.Med.Chem_46_921 |
| PubMedID: 12620069 |
| Title : Functionalization of the alicyclic skeleton of epibatidine: synthesis and nicotinic acetylcholine receptor binding affinities of epibatidine analogues - Wei_2003_Org.Biomol.Chem_1_3878 |
| Author(s) : Wei ZL , Xiao Y , George C , Kellar KJ , Kozikowski AP |
| Ref : Org Biomol Chem , 1 :3878 , 2003 |
| Abstract : |
| PubMedSearch : Wei_2003_Org.Biomol.Chem_1_3878 |
| PubMedID: 14664377 |
| Title : Measuring nicotinic receptors with characteristics of alpha4beta2, alpha3beta2 and alpha3beta4 subtypes in rat tissues by autoradiography - Perry_2002_J.Neurochem_82_468 |
| Author(s) : Perry DC , Xiao Y , Nguyen HN , Musachio JL , Davila-Garcia MI , Kellar KJ |
| Ref : Journal of Neurochemistry , 82 :468 , 2002 |
| Abstract : |
| PubMedSearch : Perry_2002_J.Neurochem_82_468 |
| PubMedID: 12153472 |
| Title : Axotomy and nerve growth factor regulate levels of neuronal nicotinic acetylcholine receptor alpha3 subunit protein in the rat superior cervical ganglion - Yeh_2001_J.Neurochem_79_258 |
| Author(s) : Yeh J , Ferreira M , Ebert S , Yasuda RP , Kellar KJ , Wolfe BB |
| Ref : Journal of Neurochemistry , 79 :258 , 2001 |
| Abstract : |
| PubMedSearch : Yeh_2001_J.Neurochem_79_258 |
| PubMedID: 11677253 |
| Title : Neuronal nicotinic acetylcholine receptor alpha3 subunit protein in rat brain and sympathetic ganglion measured using a subunit-specific antibody: regional and ontogenic expression - Yeh_2001_J.Neurochem_77_336 |
| Author(s) : Yeh JJ , Yasuda RP , Davila-Garcia MI , Xiao Y , Ebert S , Gupta T , Kellar KJ , Wolfe BB |
| Ref : Journal of Neurochemistry , 77 :336 , 2001 |
| Abstract : |
| PubMedSearch : Yeh_2001_J.Neurochem_77_336 |
| PubMedID: 11279289 |
| Title : Blockade of rat alpha3beta4 nicotinic receptor function by methadone, its metabolites, and structural analogs - Xiao_2001_J.Pharmacol.Exp.Ther_299_366 |
| Author(s) : Xiao Y , Smith RD , Caruso FS , Kellar KJ |
| Ref : Journal of Pharmacology & Experimental Therapeutics , 299 :366 , 2001 |
| Abstract : |
| PubMedSearch : Xiao_2001_J.Pharmacol.Exp.Ther_299_366 |
| PubMedID: 11561100 |
| Title : Agonist regulation of rat alpha 3 beta 4 nicotinic acetylcholine receptors stably expressed in human embryonic kidney 293 cells - Meyer_2001_Mol.Pharmacol_60_568 |
| Author(s) : Meyer EL , Xiao Y , Kellar KJ |
| Ref : Molecular Pharmacology , 60 :568 , 2001 |
| Abstract : |
| PubMedSearch : Meyer_2001_Mol.Pharmacol_60_568 |
| PubMedID: 11502889 |
| Title : [125\/123I] 5-Iodo-3-pyridyl ethers. syntheses and binding to neuronal nicotinic acetylcholine receptors - Fan_2001_Nucl.Med.Biol_28_911 |
| Author(s) : Fan H , Scheffel UA , Rauseo P , Xiao Y , Dogan AS , Yokoi F , Hilton J , Kellar KJ , Wong DF , Musachio JL |
| Ref : Nucl Med Biol , 28 :911 , 2001 |
| Abstract : |
| PubMedSearch : Fan_2001_Nucl.Med.Biol_28_911 |
| PubMedID: 11711310 |
| Title : Dextromethorphan and its metabolite dextrorphan block alpha3beta4 neuronal nicotinic receptors - Hernandez_2000_J.Pharmacol.Exp.Ther_293_962 |
| Author(s) : Hernandez SC , Bertolino M , Xiao Y , Pringle KE , Caruso FS , Kellar KJ |
| Ref : Journal of Pharmacology & Experimental Therapeutics , 293 :962 , 2000 |
| Abstract : |
| PubMedSearch : Hernandez_2000_J.Pharmacol.Exp.Ther_293_962 |
| PubMedID: 10869398 |
| Title : International Union of Pharmacology. XX. Current status of the nomenclature for nicotinic acetylcholine receptors and their subunits - |
| Author(s) : Lukas RJ , Changeux JP , Le Novere N , Albuquerque EX , Balfour DJ , Berg DK , Bertrand D , Chiappinelli VA , Clarke PB , Collins AC , Dani JA , Grady SR , Kellar KJ , Lindstrom JM , Marks MJ , Quik M , Taylor P , Wonnacott S |
| Ref : Pharmacol Rev , 51 :397 , 1999 |
| PubMedID: 10353988 |
| Title : Activation and Ca2+ permeation of stably transfected alpha3\/beta4 neuronal nicotinic acetylcholine receptor - Zhang_1999_Mol.Pharmacol_55_970 |
| Author(s) : Zhang J , Xiao Y , Abdrakhmanova G , Wang W , Cleemann L , Kellar KJ , Morad M |
| Ref : Molecular Pharmacology , 55 :970 , 1999 |
| Abstract : |
| PubMedSearch : Zhang_1999_Mol.Pharmacol_55_970 |
| PubMedID: 10347237 |
| Title : Pharmacology of neuronal nicotinic acetylcholine recceptors: effects of acute and chronic nicotine - Kellar_1999_Nicotine.Tob.Res_1 Suppl 2_S117 |
| Author(s) : Kellar KJ , Davila-Garcia MI , Xiao Y |
| Ref : Nicotine Tob Res , 1 Suppl 2 :S117 , 1999 |
| Abstract : |
| PubMedSearch : Kellar_1999_Nicotine.Tob.Res_1 Suppl 2_S117 |
| PubMedID: 11768167 |
| Title : Liquid chromatographic studies with immobilized neuronal nicotinic acetylcholine receptor stationary phases: effects of receptor subtypes, pH and ionic strength on drug-receptor interactions - Wainer_1999_J.Chromatogr.B.Biomed.Sci.Appl_724_65 |
| Author(s) : Wainer IW , Zhang Y , Xiao Y , Kellar KJ |
| Ref : Journal of Chromatography B Biomed Sci Appl , 724 :65 , 1999 |
| Abstract : |
| PubMedSearch : Wainer_1999_J.Chromatogr.B.Biomed.Sci.Appl_724_65 |
| PubMedID: 10202958 |
| Title : Immobilized nicotinic receptor stationary phase for on-line liquid chromatographic determination of drug-receptor affinities - Zhang_1998_Anal.Biochem_264_22 |
| Author(s) : Zhang Y , Xiao Y , Kellar KJ , Wainer IW |
| Ref : Analytical Biochemistry , 264 :22 , 1998 |
| Abstract : |
| PubMedSearch : Zhang_1998_Anal.Biochem_264_22 |
| PubMedID: 9784183 |
| Title : Rat alpha3\/beta4 subtype of neuronal nicotinic acetylcholine receptor stably expressed in a transfected cell line: pharmacology of ligand binding and function - Xiao_1998_Mol.Pharmacol_54_322 |
| Author(s) : Xiao Y , Meyer EL , Thompson JM , Surin A , Wroblewski J , Kellar KJ |
| Ref : Molecular Pharmacology , 54 :322 , 1998 |
| Abstract : |
| PubMedSearch : Xiao_1998_Mol.Pharmacol_54_322 |
| PubMedID: 9687574 |
| Title : Differential regulation of neuronal nicotinic receptor binding sites following chronic nicotine administration - Flores_1997_J.Neurochem_69_2216 |
| Author(s) : Flores CM , Davila-Garcia MI , Ulrich YM , Kellar KJ |
| Ref : Journal of Neurochemistry , 69 :2216 , 1997 |
| Abstract : |
| PubMedSearch : Flores_1997_J.Neurochem_69_2216 |
| PubMedID: 9349569 |
| Title : [125I]IPH, an epibatidine analog, binds with high affinity to neuronal nicotinic cholinergic receptors - Davila-Garcia_1997_J.Pharmacol.Exp.Ther_282_445 |
| Author(s) : Davila-Garcia MI , Musachio JL , Perry DC , Xiao Y , Horti A , London ED , Dannals RF , Kellar KJ |
| Ref : Journal of Pharmacology & Experimental Therapeutics , 282 :445 , 1997 |
| Abstract : |
| PubMedSearch : Davila-Garcia_1997_J.Pharmacol.Exp.Ther_282_445 |
| PubMedID: 9223586 |
| Title : Characterization of (+\/-)(-)[3H]epibatidine binding to nicotinic cholinergic receptors in rat and human brain - Houghtling_1995_Mol.Pharmacol_48_280 |
| Author(s) : Houghtling RA , Davila-Garcia MI , Kellar KJ |
| Ref : Molecular Pharmacology , 48 :280 , 1995 |
| Abstract : |
| PubMedSearch : Houghtling_1995_Mol.Pharmacol_48_280 |
| PubMedID: 7651361 |
| Title : In vivo labeling of nicotinic acetylcholine receptors in brain with [3H]epibatidine - London_1995_Eur.J.Pharmacol_278_R1 |
| Author(s) : London ED , Scheffel U , Kimes AS , Kellar KJ |
| Ref : European Journal of Pharmacology , 278 :R1 , 1995 |
| Abstract : |
| PubMedSearch : London_1995_Eur.J.Pharmacol_278_R1 |
| PubMedID: 7664806 |
| Title : A subtype of nicotinic cholinergic receptor in rat brain is composed of alpha 4 and beta 2 subunits and is up-regulated by chronic nicotine treatment - Flores_1992_Mol.Pharmacol_41_31 |
| Author(s) : Flores CM , Rogers SW , Pabreza LA , Wolfe BB , Kellar KJ |
| Ref : Molecular Pharmacology , 41 :31 , 1992 |
| Abstract : |
| PubMedSearch : Flores_1992_Mol.Pharmacol_41_31 |
| PubMedID: 1732720 |
| Title : [3H]cytisine binding to nicotinic cholinergic receptors in brain - Pabreza_1991_Mol.Pharmacol_39_9 |
| Author(s) : Pabreza LA , Dhawan S , Kellar KJ |
| Ref : Molecular Pharmacology , 39 :9 , 1991 |
| Abstract : |
| PubMedSearch : Pabreza_1991_Mol.Pharmacol_39_9 |
| PubMedID: 1987453 |
| Title : Naltrexone blocks nicotine-induced prolactin release - Flores_1989_Neuropharmacol_28_1287 |
| Author(s) : Flores CM , Hulihan-Giblin BA , Kellar KJ |
| Ref : Neuropharmacology , 28 :1287 , 1989 |
| Abstract : |
| PubMedSearch : Flores_1989_Neuropharmacol_28_1287 |
| PubMedID: 2594167 |
| Title : Nicotinic Cholinergic Receptors Labeled with [3H]Acetylcholine in Brain: Characterization, Localization and In Vivo Regulation - |
| Author(s) : Schwartz RD , Kellar KJ |
| Ref : Advances in Behavioral Biology , 30 :467 , 1986 |
| PubMedID: |
| Title : In vivo regulation of [3H]acetylcholine recognition sites in brain by nicotinic cholinergic drugs - Schwartz_1985_J.Neurochem_45_427 |
| Author(s) : Schwartz RD , Kellar KJ |
| Ref : Journal of Neurochemistry , 45 :427 , 1985 |
| Abstract : |
| PubMedSearch : Schwartz_1985_J.Neurochem_45_427 |
| PubMedID: 4009168 |
| Title : High-affinity binding of [3H]acetylcholine to muscarinic cholinergic receptors - Kellar_1985_J.Neurosci_5_1577 |
| Author(s) : Kellar KJ , Martino AM , Hall DP, Jr. , Schwartz RD , Taylor RL |
| Ref : Journal of Neuroscience , 5 :1577 , 1985 |
| Abstract : |
| PubMedSearch : Kellar_1985_J.Neurosci_5_1577 |
| PubMedID: 4009247 |
| Title : Quantitative autoradiography of nicotinic [3H]acetylcholine binding sites in rat brain - Rainbow_1984_Neurosci.Lett_50_193 |
| Author(s) : Rainbow TC , Schwartz RD , Parsons B , Kellar KJ |
| Ref : Neuroscience Letters , 50 :193 , 1984 |
| Abstract : |
| PubMedSearch : Rainbow_1984_Neurosci.Lett_50_193 |
| PubMedID: 6493626 |
| Title : Presynaptic nicotinic cholinergic receptors labeled by [3H]acetylcholine on catecholamine and serotonin axons in brain - Schwartz_1984_J.Neurochem_42_1495 |
| Author(s) : Schwartz RD , Lehmann J , Kellar KJ |
| Ref : Journal of Neurochemistry , 42 :1495 , 1984 |
| Abstract : |
| PubMedSearch : Schwartz_1984_J.Neurochem_42_1495 |
| PubMedID: 6707650 |
| Title : [3H]acetylcholine binding sites in brain. Effect of disulfide bond modification - Schwartz_1983_Mol.Pharmacol_24_387 |
| Author(s) : Schwartz RD , Kellar KJ |
| Ref : Molecular Pharmacology , 24 :387 , 1983 |
| Abstract : |
| PubMedSearch : Schwartz_1983_Mol.Pharmacol_24_387 |
| PubMedID: 6633505 |
| Title : Nicotinic cholinergic receptor binding sites in the brain: regulation in vivo - Schwartz_1983_Science_220_214 |
| Author(s) : Schwartz RD , Kellar KJ |
| Ref : Science , 220 :214 , 1983 |
| Abstract : |
| PubMedSearch : Schwartz_1983_Science_220_214 |
| PubMedID: 6828889 |
| Title : Nicotinic cholinergic receptors labeled by [3H]acetylcholine in rat brain - |
| Author(s) : Schwartz RD , McGee R, Jr. , Kellar KJ |
| Ref : Molecular Pharmacology , 22 :56 , 1982 |
| PubMedID: 7121451 |