Title : Discovery of beta-homophenylalanine based pyrrolidin-2-ylmethyl amides and sulfonamides as highly potent and selective inhibitors of dipeptidyl peptidase IV - Nordhoff_2009_Bioorg.Med.Chem.Lett_19_4201 |
Author(s) : Nordhoff S , Cerezo-Galvez S , Deppe H , Hill O , Lopez-Canet M , Rummey C , Thiemann M , Matassa VG , Edwards PJ , Feurer A |
Ref : Bioorganic & Medicinal Chemistry Lett , 19 :4201 , 2009 |
Abstract : |
PubMedSearch : Nordhoff_2009_Bioorg.Med.Chem.Lett_19_4201 |
PubMedID: 19515557 |
Gene_locus related to this paper: human-DPP4 |
Title : Homology models of dipeptidyl peptidases 8 and 9 with a focus on loop predictions near the active site - Rummey_2007_Proteins_66_160 |
Author(s) : Rummey C , Metz G |
Ref : Proteins , 66 :160 , 2007 |
Abstract : |
PubMedSearch : Rummey_2007_Proteins_66_160 |
PubMedID: 17068815 |
Title : The reversed binding of beta-phenethylamine inhibitors of DPP-IV: X-ray structures and properties of novel fragment and elaborated inhibitors - Nordhoff_2006_Bioorg.Med.Chem.Lett_16_1744 |
Author(s) : Nordhoff S , Cerezo-Galvez S , Feurer A , Hill O , Matassa VG , Metz G , Rummey C , Thiemann M , Edwards PJ |
Ref : Bioorganic & Medicinal Chemistry Lett , 16 :1744 , 2006 |
Abstract : |
PubMedSearch : Nordhoff_2006_Bioorg.Med.Chem.Lett_16_1744 |
PubMedID: 16376544 |
Gene_locus related to this paper: pig-dpp4 |
Title : In silico fragment-based discovery of DPP-IV S1 pocket binders - Rummey_2006_Bioorg.Med.Chem.Lett_16_1405 |
Author(s) : Rummey C , Nordhoff S , Thiemann M , Metz G |
Ref : Bioorganic & Medicinal Chemistry Lett , 16 :1405 , 2006 |
Abstract : |
PubMedSearch : Rummey_2006_Bioorg.Med.Chem.Lett_16_1405 |
PubMedID: 16321524 |