| Title : Synthesis of imidazopyridines and purines as potent inhibitors of leukotriene A4 hydrolase - Penning_2003_Bioorg.Med.Chem.Lett_13_1137 |
| Author(s) : Penning TD , Chandrakumar NS , Desai BN , Djuric SW , Gasiecki AF , Malecha JW , Miyashiro JM , Russell MA , Askonas LJ , Gierse JK , Harding EI , Highkin MK , Kachur JF , Kim SH , Villani-Price D , Pyla EY , Ghoreishi-Haack NS , Smith WG |
| Ref : Bioorganic & Medicinal Chemistry Lett , 13 :1137 , 2003 |
| Abstract : |
| PubMedSearch : Penning_2003_Bioorg.Med.Chem.Lett_13_1137 |
| PubMedID: 12643929 |
| Title : Pharmacological characterization of SC-57461A (3-[methyl[3-[4-(phenylmethyl)phenoxy]propyl]amino]propanoic acid HCl), a potent and selective inhibitor of leukotriene A(4) hydrolase I: in vitro studies - Askonas_2002_J.Pharmacol.Exp.Ther_300_577 |
| Author(s) : Askonas LJ , Kachur JF , Villani-Price D , Liang CD , Russell MA , Smith WG |
| Ref : Journal of Pharmacology & Experimental Therapeutics , 300 :577 , 2002 |
| Abstract : |
| PubMedSearch : Askonas_2002_J.Pharmacol.Exp.Ther_300_577 |
| PubMedID: 11805219 |
| Title : Pyrrolidine and piperidine analogues of SC-57461A as potent, orally active inhibitors of leukotriene A(4) hydrolase - Penning_2002_Bioorg.Med.Chem.Lett_12_3383 |
| Author(s) : Penning TD , Chandrakumar NS , Desai BN , Djuric SW , Gasiecki AF , Liang CD , Miyashiro JM , Russell MA , Askonas LJ , Gierse JK , Harding EI , Highkin MK , Kachur JF , Kim SH , Villani-Price D , Pyla EY , Ghoreishi-Haack NS , Smith WG |
| Ref : Bioorganic & Medicinal Chemistry Lett , 12 :3383 , 2002 |
| Abstract : |
| PubMedSearch : Penning_2002_Bioorg.Med.Chem.Lett_12_3383 |
| PubMedID: 12419366 |
| Title : Synthesis of potent leukotriene A(4) hydrolase inhibitors. Identification of 3-[methyl[3-[4-(phenylmethyl)phenoxy]propyl]amino]propanoic acid - Penning_2002_J.Med.Chem_45_3482 |
| Author(s) : Penning TD , Russell MA , Chen BB , Chen HY , Liang CD , Mahoney MW , Malecha JW , Miyashiro JM , Yu SS , Askonas LJ , Gierse JK , Harding EI , Highkin MK , Kachur JF , Kim SH , Villani-Price D , Pyla EY , Ghoreishi-Haack NS , Smith WG |
| Ref : Journal of Medicinal Chemistry , 45 :3482 , 2002 |
| Abstract : |
| PubMedSearch : Penning_2002_J.Med.Chem_45_3482 |
| PubMedID: 12139459 |
| Title : Pharmacological characterization of SC-57461A (3-[methyl[3-[4-(phenylmethyl)phenoxy]propyl]amino]propanoic acid HCl), a potent and selective inhibitor of leukotriene A(4) hydrolase II: in vivo studies - Kachur_2002_J.Pharmacol.Exp.Ther_300_583 |
| Author(s) : Kachur JF , Askonas LJ , Villani-Price D , Ghoreishi-Haack N , Won-Kim S , Liang CD , Russell MA , Smith WG |
| Ref : Journal of Pharmacology & Experimental Therapeutics , 300 :583 , 2002 |
| Abstract : |
| PubMedSearch : Kachur_2002_J.Pharmacol.Exp.Ther_300_583 |
| PubMedID: 11805220 |
| Title : Structure-activity relationship studies on 1-[2-(4-Phenylphenoxy)ethyl]pyrrolidine (SC-22716), a potent inhibitor of leukotriene A(4) (LTA(4)) hydrolase - Penning_2000_J.Med.Chem_43_721 |
| Author(s) : Penning TD , Chandrakumar NS , Chen BB , Chen HY , Desai BN , Djuric SW , Docter SH , Gasiecki AF , Haack RA , Miyashiro JM , Russell MA , Yu SS , Corley DG , Durley RC , Kilpatrick BF , Parnas BL , Askonas LJ , Gierse JK , Harding EI , Highkin MK , Kachur JF , Kim SH , Krivi GG , Villani-Price D , Pyla EY , Smith WG |
| Ref : Journal of Medicinal Chemistry , 43 :721 , 2000 |
| Abstract : |
| PubMedSearch : Penning_2000_J.Med.Chem_43_721 |
| PubMedID: 10691697 |