Title : New 3-amino-2-thioxothiazolidin-4-one-based inhibitors of acetyl- and butyryl-cholinesterase: synthesis and activity - Kratky_2023_Future.Med.Chem__ |
Author(s) : Kratky M , Novackova K , Svrckova K , Svarcova M , Stepankova S |
Ref : Future Med Chem , : , 2023 |
Abstract : |
PubMedSearch : Kratky_2023_Future.Med.Chem__ |
PubMedID: 38047370 |
Title : Novel Inhibitors of Acetyl- and Butyrylcholinesterase Derived from Benzohydrazides: Synthesis, Evaluation and Docking Study - Houngbedji_2023_Pharmaceuticals.(Basel)_16_ |
Author(s) : Houngbedji NH , Stepankova S , Pflegr V , Svrckova K , Svarcova M , Vinsova J , Kratky M |
Ref : Pharmaceuticals (Basel) , 16 : , 2023 |
Abstract : |
PubMedSearch : Houngbedji_2023_Pharmaceuticals.(Basel)_16_ |
PubMedID: 37259322 |
Title : 5-Aryl-1,3,4-oxadiazol-2-amines Decorated with Long Alkyl and Their Analogues: Synthesis, Acetyl- and Butyrylcholinesterase Inhibition and Docking Study - Pflegr_2022_Pharmaceuticals.(Basel)_15_400 |
Author(s) : Pflegr V , Stepankova S , Svrckova K , Svarcova M , Vinsova J , Kratky M |
Ref : Pharmaceuticals (Basel) , 15 :400 , 2022 |
Abstract : |
PubMedSearch : Pflegr_2022_Pharmaceuticals.(Basel)_15_400 |
PubMedID: 35455397 |
Title : Ring-fused 3beta-acetoxyandrost-5-enes as novel neuroprotective agents with cholinesterase inhibitory properties - Gonzalez_2022_J.Steroid.Biochem.Mol.Biol__106194 |
Author(s) : Gonzalez G , Kvasnica M , Svrckova K , Stepankova S , Santos JRC , Perina M , Jorda R , Lopes SMM , Melo T |
Ref : J Steroid Biochem Mol Biol , :106194 , 2022 |
Abstract : |
PubMedSearch : Gonzalez_2022_J.Steroid.Biochem.Mol.Biol__106194 |
PubMedID: 36162631 |
Title : Novel propargylamine-based inhibitors of cholinesterases and monoamine oxidases: Synthesis, biological evaluation and docking study - Kratky_2021_Bioorg.Chem_116_105301 |
Author(s) : Kratky M , Vu QA , Stepankova S , Maruca A , Silva TB , Ambroz M , Pflegr V , Rocca R , Svrckova K , Alcaro S , Borges F , Vinsova J |
Ref : Bioorg Chem , 116 :105301 , 2021 |
Abstract : |
PubMedSearch : Kratky_2021_Bioorg.Chem_116_105301 |
PubMedID: 34492558 |
Title : Hydrazones of 4-(Trifluoromethyl)benzohydrazide as New Inhibitors of Acetyl- and Butyrylcholinesterase - Kratky_2021_Molecules_26_ |
Author(s) : Kratky M , Svrckova K , Vu QA , Stpankova S , Vinsova J |
Ref : Molecules , 26 : , 2021 |
Abstract : |
PubMedSearch : Kratky_2021_Molecules_26_ |
PubMedID: 33668452 |
Title : Novel Aminoguanidine Hydrazone Analogues: From Potential Antimicrobial Agents to Potent Cholinesterase Inhibitors - Kratky_2021_Pharmaceuticals.(Basel)_14_ |
Author(s) : Kratky M , Stepankova S , Konecna K , Svrckova K , Maixnerova J , Svarcova M , Janourek O , Trejtnar F , Vinsova J |
Ref : Pharmaceuticals (Basel) , 14 : , 2021 |
Abstract : |
PubMedSearch : Kratky_2021_Pharmaceuticals.(Basel)_14_ |
PubMedID: 34959630 |
Title : Novel Sulfonamide-Based Carbamates as Selective Inhibitors of BChE - Magar_2021_Int.J.Mol.Sci_22_ |
Author(s) : Magar P , Parravicini O , Stepankova S , Svrckova K , Garro AD , Jendrzejewska I , Pauk K , Hosek J , Jampilek J , Enriz RD , Imramovsky A |
Ref : Int J Mol Sci , 22 : , 2021 |
Abstract : |
PubMedSearch : Magar_2021_Int.J.Mol.Sci_22_ |
PubMedID: 34502357 |
Title : N-[3,5-Bis(trifluoromethyl)phenyl]-5-bromo-2-hydroxybenzamide Analogues: Novel Acetyl- and Butyrylcholinesterase Inhibitors - Kratky_2020_Curr.Top.Med.Chem_20_2094 |
Author(s) : Kratky M , Jaklova K , Stepankova S , Svrckova K , Pflegr V , Vinsova J |
Ref : Curr Top Med Chem , 20 :2094 , 2020 |
Abstract : |
PubMedSearch : Kratky_2020_Curr.Top.Med.Chem_20_2094 |
PubMedID: 32814530 |
Title : Novel Iodinated Hydrazide-hydrazones and their Analogues as Acetyl- and Butyrylcholinesterase Inhibitors - Kratky_2020_Curr.Top.Med.Chem_20_2106 |
Author(s) : Kratky M , Stepankova S , Brablikova M , Svrckova K , Svarcova M , Vinsova J |
Ref : Curr Top Med Chem , 20 :2106 , 2020 |
Abstract : |
PubMedSearch : Kratky_2020_Curr.Top.Med.Chem_20_2106 |
PubMedID: 32814531 |
Title : N-Alkyl-2-[4-(trifluoromethyl)benzoyl]hydrazine-1-carboxamides and Their Analogues: Synthesis and Multitarget Biological Activity - Kratky_2020_Molecules_25_ |
Author(s) : Kratky M , Baranyai Z , Stepankova S , Svrckova K , Svarcova M , Stolarikova J , Horvath L , Bosze S , Vinsova J |
Ref : Molecules , 25 : , 2020 |
Abstract : |
PubMedSearch : Kratky_2020_Molecules_25_ |
PubMedID: 32408517 |
Title : The synthesis and cholinesterase inhibitory activities of solasodine analogues with seven-membered F ring - Kielczewska_2020_J.Steroid.Biochem.Mol.Biol__105776 |
Author(s) : Kielczewska U , Jorda R , Gonzalez G , Morzycki JW , Ajani H , Svrckova K , Stepankova S , Wojtkielewicz A |
Ref : J Steroid Biochem Mol Biol , :105776 , 2020 |
Abstract : |
PubMedSearch : Kielczewska_2020_J.Steroid.Biochem.Mol.Biol__105776 |
PubMedID: 33130020 |