| Title : Discover the Power of Lithospermic Acid as Human Carbonic Anhydrase VA and Pancreatic Lipase Inhibitor Through In Silico and In Vitro Studies - Citriniti_2025_Arch.Pharm.(Weinheim)_358_e3128 |
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| Ref : Arch Pharm (Weinheim) , 358 :e3128 , 2025 |
| Abstract : |
| PubMedSearch : Citriniti_2025_Arch.Pharm.(Weinheim)_358_e3128 |
| PubMedID: 40257393 |
| Title : A Dynamic and Effective Peptide-Based Strategy for Promptly Addressing Emerging SARS-CoV-2 Variants of Concern - Murdocca_2024_Pharmaceuticals.(Basel)_17_ |
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| Ref : Pharmaceuticals (Basel) , 17 : , 2024 |
| Abstract : |
| PubMedSearch : Murdocca_2024_Pharmaceuticals.(Basel)_17_ |
| PubMedID: 39065742 |
| Title : Novel multifunctional tacrine-donepezil hybrids against Alzheimer's disease: Design synthesis and bioactivity studies - Bayraktar_2024_Arch.Pharm.(Weinheim)__e2300575 |
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| Ref : Arch Pharm (Weinheim) , :e2300575 , 2024 |
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| PubMedSearch : Bayraktar_2024_Arch.Pharm.(Weinheim)__e2300575 |
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| Title : Evaluating Quinolines: Molecular Dynamics Approach to Assess Their Potential as Acetylcholinesterase Inhibitors for Alzheimer's Disease - Prejano_2024_Chemphyschem__e202400653 |
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| Ref : Chemphyschem , :e202400653 , 2024 |
| Abstract : |
| PubMedSearch : Prejano_2024_Chemphyschem__e202400653 |
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| Title : Design, Synthesis, and In Vitro, In Silico and In Cellulo Evaluation of New Pyrimidine and Pyridine Amide and Carbamate Derivatives as Multi-Functional Cholinesterase Inhibitors - Bortolami_2022_Pharmaceuticals.(Basel)_15_ |
| Author(s) : Bortolami M , Pandolfi F , Tudino V , Messore A , Madia VN , De Vita D , Di Santo R , Costi R , Romeo I , Alcaro S , Colone M , Stringaro A , Espargaro A , Sabate R , Scipione L |
| Ref : Pharmaceuticals (Basel) , 15 : , 2022 |
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| PubMedSearch : Bortolami_2022_Pharmaceuticals.(Basel)_15_ |
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| Ref : Bioorganic & Medicinal Chemistry , 68 :116807 , 2022 |
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| PubMedSearch : Moutayakine_2022_Bioorg.Med.Chem_68_116807 |
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| Title : Novel propargylamine-based inhibitors of cholinesterases and monoamine oxidases: Synthesis, biological evaluation and docking study - Kratky_2021_Bioorg.Chem_116_105301 |
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| Title : New Pyrimidine and Pyridine Derivatives as Multitarget Cholinesterase Inhibitors: Design, Synthesis, and In Vitro and In Cellulo Evaluation - Bortolami_2021_ACS.Chem.Neurosci__ |
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| Ref : ACS Chem Neurosci , : , 2021 |
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| Title : N-1,2,3-triazole-isatin derivatives for cholinesterase and beta-amyloid aggregation inhibition: A comprehensive bioassay study - Marques_2020_Bioorg.Chem_98_103753 |
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| Ref : Eur Journal of Medicinal Chemistry , 198 :112350 , 2020 |
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| Ref : Eur Journal of Medicinal Chemistry , 174 :116 , 2019 |
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| Ref : Eur Journal of Medicinal Chemistry , 181 :111572 , 2019 |
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| Title : 4-(3-Nitrophenyl)thiazol-2-ylhydrazone derivatives as antioxidants and selective hMAO-B inhibitors: synthesis, biological activity and computational analysis - Secci_2019_J.Enzyme.Inhib.Med.Chem_34_597 |
| Author(s) : Secci D , Carradori S , Petzer A , Guglielmi P , D'Ascenzio M , Chimenti P , Bagetta D , Alcaro S , Zengin G , Petzer JP , Ortuso F |
| Ref : J Enzyme Inhib Med Chem , 34 :597 , 2019 |
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| Ref : Eur Journal of Medicinal Chemistry , 158 :781 , 2018 |
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| PubMedSearch : Reis_2018_Eur.J.Med.Chem_158_781 |
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| Ref : Eur Journal of Medicinal Chemistry , 143 :1543 , 2018 |
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| Ref : J Enzyme Inhib Med Chem , 30 :908 , 2015 |
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| PubMedSearch : D'Ascenzio_2015_J.Enzyme.Inhib.Med.Chem_30_908 |
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| PubMedSearch : Alcaro_2002_Bioorg.Med.Chem.Lett_12_2899 |
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