| Title : Novel neuroprotective 5,6-dihydropyrido[2',1':2,3]imidazo[4,5-c]quinoline derivatives acting through cholinesterase inhibition and CB2 signaling modulation - Jena_2024_Eur.J.Med.Chem_276_116592 |
| Author(s) : Jena S , Gonzalez G , Vitek D , Kvasnicova M , Stepankova S , Strnad M , Voller J , Chanda K |
| Ref : Eur Journal of Medicinal Chemistry , 276 :116592 , 2024 |
| Abstract : |
| PubMedSearch : Jena_2024_Eur.J.Med.Chem_276_116592 |
| PubMedID: 39013357 |
| Title : New biologically active sulfonamides as potential drugs for Alzheimer's disease - Nevyhostena_2024_Arch.Pharm.(Weinheim)__e2400191 |
| Author(s) : Nevyhostena M , Komersova A , Pejchal V , Stepankova S , Cesla P , Matzick K , Machackova J , Svoboda R |
| Ref : Arch Pharm (Weinheim) , :e2400191 , 2024 |
| Abstract : |
| PubMedSearch : Nevyhostena_2024_Arch.Pharm.(Weinheim)__e2400191 |
| PubMedID: 38941614 |
| Title : Synthesis and neuroprotective activity of 3-aryl-3-azetidinyl acetic acid methyl ester derivatives - Sachleviciute_2023_Arch.Pharm.(Weinheim)__e2300378 |
| Author(s) : Sachleviciute U , Gonzalez G , Kvasnicova M , Stepankova S , Kleizien N , Bieliauskas A , Zatloukal M , Strnad M , Slok FA , Kvasnica M , Sackus A , zukauskait A |
| Ref : Arch Pharm (Weinheim) , :e2300378 , 2023 |
| Abstract : |
| PubMedSearch : Sachleviciute_2023_Arch.Pharm.(Weinheim)__e2300378 |
| PubMedID: 37797174 |
| Title : New 3-amino-2-thioxothiazolidin-4-one-based inhibitors of acetyl- and butyryl-cholinesterase: synthesis and activity - Kratky_2023_Future.Med.Chem__ |
| Author(s) : Kratky M , Novackova K , Svrckova K , Svarcova M , Stepankova S |
| Ref : Future Med Chem , : , 2023 |
| Abstract : |
| PubMedSearch : Kratky_2023_Future.Med.Chem__ |
| PubMedID: 38047370 |
| Title : Novel Inhibitors of Acetyl- and Butyrylcholinesterase Derived from Benzohydrazides: Synthesis, Evaluation and Docking Study - Houngbedji_2023_Pharmaceuticals.(Basel)_16_ |
| Author(s) : Houngbedji NH , Stepankova S , Pflegr V , Svrckova K , Svarcova M , Vinsova J , Kratky M |
| Ref : Pharmaceuticals (Basel) , 16 : , 2023 |
| Abstract : |
| PubMedSearch : Houngbedji_2023_Pharmaceuticals.(Basel)_16_ |
| PubMedID: 37259322 |
| Title : 5-Aryl-1,3,4-oxadiazol-2-amines Decorated with Long Alkyl and Their Analogues: Synthesis, Acetyl- and Butyrylcholinesterase Inhibition and Docking Study - Pflegr_2022_Pharmaceuticals.(Basel)_15_400 |
| Author(s) : Pflegr V , Stepankova S , Svrckova K , Svarcova M , Vinsova J , Kratky M |
| Ref : Pharmaceuticals (Basel) , 15 :400 , 2022 |
| Abstract : |
| PubMedSearch : Pflegr_2022_Pharmaceuticals.(Basel)_15_400 |
| PubMedID: 35455397 |
| Title : Ring-fused 3beta-acetoxyandrost-5-enes as novel neuroprotective agents with cholinesterase inhibitory properties - Gonzalez_2022_J.Steroid.Biochem.Mol.Biol__106194 |
| Author(s) : Gonzalez G , Kvasnica M , Svrckova K , Stepankova S , Santos JRC , Perina M , Jorda R , Lopes SMM , Melo T |
| Ref : J Steroid Biochem Mol Biol , :106194 , 2022 |
| Abstract : |
| PubMedSearch : Gonzalez_2022_J.Steroid.Biochem.Mol.Biol__106194 |
| PubMedID: 36162631 |
| Title : Synthesis and Hybrid SAR Property Modeling of Novel Cholinesterase Inhibitors - Kos_2021_Int.J.Mol.Sci_22_ |
| Author(s) : Kos J , Kozik V , Pindjakova D , Jankech T , Smolinski A , Stepankova S , Hosek J , Oravec M , Jampilek J , Bak A |
| Ref : Int J Mol Sci , 22 : , 2021 |
| Abstract : |
| PubMedSearch : Kos_2021_Int.J.Mol.Sci_22_ |
| PubMedID: 33810550 |
| Title : Novel Sulfonamide-Based Carbamates as Selective Inhibitors of BChE - Magar_2021_Int.J.Mol.Sci_22_ |
| Author(s) : Magar P , Parravicini O , Stepankova S , Svrckova K , Garro AD , Jendrzejewska I , Pauk K , Hosek J , Jampilek J , Enriz RD , Imramovsky A |
| Ref : Int J Mol Sci , 22 : , 2021 |
| Abstract : |
| PubMedSearch : Magar_2021_Int.J.Mol.Sci_22_ |
| PubMedID: 34502357 |
| Title : Novel Aminoguanidine Hydrazone Analogues: From Potential Antimicrobial Agents to Potent Cholinesterase Inhibitors - Kratky_2021_Pharmaceuticals.(Basel)_14_ |
| Author(s) : Kratky M , Stepankova S , Konecna K , Svrckova K , Maixnerova J , Svarcova M , Janourek O , Trejtnar F , Vinsova J |
| Ref : Pharmaceuticals (Basel) , 14 : , 2021 |
| Abstract : |
| PubMedSearch : Kratky_2021_Pharmaceuticals.(Basel)_14_ |
| PubMedID: 34959630 |
| Title : Novel propargylamine-based inhibitors of cholinesterases and monoamine oxidases: Synthesis, biological evaluation and docking study - Kratky_2021_Bioorg.Chem_116_105301 |
| Author(s) : Kratky M , Vu QA , Stepankova S , Maruca A , Silva TB , Ambroz M , Pflegr V , Rocca R , Svrckova K , Alcaro S , Borges F , Vinsova J |
| Ref : Bioorg Chem , 116 :105301 , 2021 |
| Abstract : |
| PubMedSearch : Kratky_2021_Bioorg.Chem_116_105301 |
| PubMedID: 34492558 |
| Title : N-[3,5-Bis(trifluoromethyl)phenyl]-5-bromo-2-hydroxybenzamide Analogues: Novel Acetyl- and Butyrylcholinesterase Inhibitors - Kratky_2020_Curr.Top.Med.Chem_20_2094 |
| Author(s) : Kratky M , Jaklova K , Stepankova S , Svrckova K , Pflegr V , Vinsova J |
| Ref : Curr Top Med Chem , 20 :2094 , 2020 |
| Abstract : |
| PubMedSearch : Kratky_2020_Curr.Top.Med.Chem_20_2094 |
| PubMedID: 32814530 |
| Title : Novel Iodinated Hydrazide-hydrazones and their Analogues as Acetyl- and Butyrylcholinesterase Inhibitors - Kratky_2020_Curr.Top.Med.Chem_20_2106 |
| Author(s) : Kratky M , Stepankova S , Brablikova M , Svrckova K , Svarcova M , Vinsova J |
| Ref : Curr Top Med Chem , 20 :2106 , 2020 |
| Abstract : |
| PubMedSearch : Kratky_2020_Curr.Top.Med.Chem_20_2106 |
| PubMedID: 32814531 |
| Title : N-Alkyl-2-[4-(trifluoromethyl)benzoyl]hydrazine-1-carboxamides and Their Analogues: Synthesis and Multitarget Biological Activity - Kratky_2020_Molecules_25_ |
| Author(s) : Kratky M , Baranyai Z , Stepankova S , Svrckova K , Svarcova M , Stolarikova J , Horvath L , Bosze S , Vinsova J |
| Ref : Molecules , 25 : , 2020 |
| Abstract : |
| PubMedSearch : Kratky_2020_Molecules_25_ |
| PubMedID: 32408517 |
| Title : The synthesis and cholinesterase inhibitory activities of solasodine analogues with seven-membered F ring - Kielczewska_2020_J.Steroid.Biochem.Mol.Biol__105776 |
| Author(s) : Kielczewska U , Jorda R , Gonzalez G , Morzycki JW , Ajani H , Svrckova K , Stepankova S , Wojtkielewicz A |
| Ref : J Steroid Biochem Mol Biol , :105776 , 2020 |
| Abstract : |
| PubMedSearch : Kielczewska_2020_J.Steroid.Biochem.Mol.Biol__105776 |
| PubMedID: 33130020 |
| Title : 2-Hydroxy-N-phenylbenzamides and Their Esters Inhibit Acetylcholinesterase and Butyrylcholinesterase - Kratky_2019_Biomolecules_9_ |
| Author(s) : Kratky M , Stepankova S , Houngbedji NH , Vosatka R , Vorcakova K , Vinsova J |
| Ref : Biomolecules , 9 : , 2019 |
| Abstract : |
| PubMedSearch : Kratky_2019_Biomolecules_9_ |
| PubMedID: 31694272 |
| Title : Novel Benzene-Based Carbamates for AChE\/BChE Inhibition: Synthesis and Ligand\/Structure-Oriented SAR Study - Bak_2019_Int.J.Mol.Sci_20_1524 |
| Author(s) : Bak A , Kozik V , Kozakiewicz D , Gajcy K , Strub DJ , Swietlicka A , Stepankova S , Imramovsky A , Polanski J , Smolinski A , Jampilek J |
| Ref : Int J Mol Sci , 20 :1524 , 2019 |
| Abstract : |
| PubMedSearch : Bak_2019_Int.J.Mol.Sci_20_1524 |
| PubMedID: 30934674 |
| Title : In Vitro and In Silico Acetylcholinesterase Inhibitory Activity of Thalictricavine and Canadine and Their Predicted Penetration across the Blood-Brain Barrier - Chlebek_2019_Molecules_24_ |
| Author(s) : Chlebek J , Korabecny J , Dolezal R , Stepankova S , Perez DI , Hostalkova A , Opletal L , Cahlikova L , Macakova K , Kucera T , Hrabinova M , Jun D |
| Ref : Molecules , 24 : , 2019 |
| Abstract : |
| PubMedSearch : Chlebek_2019_Molecules_24_ |
| PubMedID: 30959739 |
| Title : Investigation of salicylanilide and 4-chlorophenol-based N-monosubstituted carbamates as potential inhibitors of acetyl- and butyrylcholinesterase - Kratky_2018_Bioorg.Chem_80_668 |
| Author(s) : Kratky M , Stepankova S , Vorcakova K , Vinsova J |
| Ref : Bioorg Chem , 80 :668 , 2018 |
| Abstract : |
| PubMedSearch : Kratky_2018_Bioorg.Chem_80_668 |
| PubMedID: 30059892 |
| Title : Synthesis and characterization of new inhibitors of cholinesterases based on N-phenylcarbamates: In vitro study of inhibitory effect, type of inhibition, lipophilicity and molecular docking - Vorcakova_2018_Bioorg.Chem_78_280 |
| Author(s) : Vorcakova K , Majekova M , Horakova E , Drabina P , Sedlak M , Stepankova S |
| Ref : Bioorg Chem , 78 :280 , 2018 |
| Abstract : |
| PubMedSearch : Vorcakova_2018_Bioorg.Chem_78_280 |
| PubMedID: 29621640 |
| Title : Proline-Based Carbamates as Cholinesterase Inhibitors - Pizova_2017_Molecules_22_ |
| Author(s) : Pizova H , Havelkova M , Stepankova S , Bak A , Kauerova T , Kozik V , Oravec M , Imramovsky A , Kollar P , Bobal P , Jampilek J |
| Ref : Molecules , 22 : , 2017 |
| Abstract : |
| PubMedSearch : Pizova_2017_Molecules_22_ |
| PubMedID: 29135926 |
| Title : Synthesis of readily available fluorophenylalanine derivatives and investigation of their biological activity - Kratky_2017_Bioorg.Chem_71_244 |
| Author(s) : Kratky M , Stepankova S , Vorcakova K , Navratilova L , Trejtnar F , Stolarikova J , Vinsova J |
| Ref : Bioorg Chem , 71 :244 , 2017 |
| Abstract : |
| PubMedSearch : Kratky_2017_Bioorg.Chem_71_244 |
| PubMedID: 28245905 |
| Title : Cholinesterase-based biosensors - Stepankova_2016_J.Enzyme.Inhib.Med.Chem__1 |
| Author(s) : Stepankova S , Vorcakova K |
| Ref : J Enzyme Inhib Med Chem , :1 , 2016 |
| Abstract : |
| PubMedSearch : Stepankova_2016_J.Enzyme.Inhib.Med.Chem__1 |
| PubMedID: 27405024 |
| Title : Novel Cholinesterase Inhibitors Based on O-Aromatic N,N-Disubstituted Carbamates and Thiocarbamates - Kratky_2016_Molecules_21_ |
| Author(s) : Kratky M , Stepankova S , Vorcakova K , Svarcova M , Vinsova J |
| Ref : Molecules , 21 : , 2016 |
| Abstract : |
| PubMedSearch : Kratky_2016_Molecules_21_ |
| PubMedID: 26875979 |
| Title : Synthesis, characterization and in vitro evaluation of substituted N-(2-phenylcyclopropyl)carbamates as acetyl- and butyrylcholinesterase inhibitors - Horakova_2016_J.Enzyme.Inhib.Med.Chem__1 |
| Author(s) : Horakova E , Drabina P , Broz B , Stepankova S , Vorcakova K , Kralovec K , Havelek R , Sedlak M |
| Ref : J Enzyme Inhib Med Chem , :1 , 2016 |
| Abstract : |
| PubMedSearch : Horakova_2016_J.Enzyme.Inhib.Med.Chem__1 |
| PubMedID: 27476673 |
| Title : Synthesis and in vitro evaluation of novel rhodanine derivatives as potential cholinesterase inhibitors - Kratky_2016_Bioorg.Chem_68_23 |
| Author(s) : Kratky M , Stepankova S , Vorcakova K , Vinsova J |
| Ref : Bioorg Chem , 68 :23 , 2016 |
| Abstract : |
| PubMedSearch : Kratky_2016_Bioorg.Chem_68_23 |
| PubMedID: 27428597 |
| Title : Synthesis, structural characterization, docking, lipophilicity and cytotoxicity of 1-[(1R)-1-(6-fluoro-1,3-benzothiazol-2-yl)ethyl]-3-alkyl carbamates, novel acetylcholinesterase and butyrylcholinesterase pseudo-irreversible inhibitors - Pejchal_2016_Bioorg.Med.Chem_24_1560 |
| Author(s) : Pejchal V , Stepankova S , Pejchalova M , Kralovec K , Havelek R , Ruzickova Z , Ajani H , Lo R , Lepsik M |
| Ref : Bioorganic & Medicinal Chemistry , 24 :1560 , 2016 |
| Abstract : |
| PubMedSearch : Pejchal_2016_Bioorg.Med.Chem_24_1560 |
| PubMedID: 26947959 |
| Title : In Vitro Inhibitory Effects of 8-O-Demethylmaritidine and Undulatine on Acetylcholinesterase and Their Predicted Penetration across the Blood-Brain Barrier - Cahlikova_2015_J.Nat.Prod_78_1189 |
| Author(s) : Cahlikova L , Perez DI , Stepankova S , Chlebek J , Safratova M , Host'alkova A , Opletal L |
| Ref : Journal of Natural Products , 78 :1189 , 2015 |
| Abstract : |
| PubMedSearch : Cahlikova_2015_J.Nat.Prod_78_1189 |
| PubMedID: 26030662 |
| Title : Salicylanilide diethyl phosphates as cholinesterases inhibitors - Kratky_2014_Bioorg.Chem_58C_48 |
| Author(s) : Kratky M , Stepankova S , Vorcakova K , Vinsova J |
| Ref : Bioorg Chem , 58C :48 , 2014 |
| Abstract : |
| PubMedSearch : Kratky_2014_Bioorg.Chem_58C_48 |
| PubMedID: 25462625 |
| Title : Diethyl 2-(Phenylcarbamoyl)phenyl Phosphorothioates: Synthesis, Antimycobacterial Activity and Cholinesterase Inhibition - Vinsova_2014_Molecules_19_7152 |
| Author(s) : Vinsova J , Kratky M , Komloova M , Dadapeer E , Stepankova S , Vorcakova K , Stolarikova J |
| Ref : Molecules , 19 :7152 , 2014 |
| Abstract : |
| PubMedSearch : Vinsova_2014_Molecules_19_7152 |
| PubMedID: 24886941 |
| Title : Chemical composition of bioactive alkaloid extracts from some Narcissus species and varieties and their biological activity - Havlasova_2014_Nat.Prod.Commun_9_1151 |
| Author(s) : Havlasova J , Safratova M , Siatka T , Stepankova S , Novak Z , Locarek M , Opletal L , Hrabinova M , Jun D , Benesova N , Kunes J , Cahlikova L |
| Ref : Nat Prod Commun , 9 :1151 , 2014 |
| Abstract : |
| PubMedSearch : Havlasova_2014_Nat.Prod.Commun_9_1151 |
| PubMedID: 25233595 |
| Title : New method for the determination of the half inhibition concentration (IC50) of cholinesterase inhibitors - Kovarova_2013_Z.Naturforsch.C_68_133 |
| Author(s) : Kovarova M , Komers K , Stepankova S , Parik P , Cegan A |
| Ref : Z Naturforsch C , 68 :133 , 2013 |
| Abstract : |
| PubMedSearch : Kovarova_2013_Z.Naturforsch.C_68_133 |
| PubMedID: 23819309 |
| Title : Synthesis and in vitro evaluation of new derivatives of 2-substituted-6-fluorobenzo[d]thiazoles as cholinesterase inhibitors - Imramovsky_2013_Bioorg.Med.Chem_21_1735 |
| Author(s) : Imramovsky A , Pejchal V , Stepankova S , Vorcakova K , Jampilek J , Vanco J , Simunek P , Kralovec K , Bruckova L , Mandikova J , Trejtnar F |
| Ref : Bioorganic & Medicinal Chemistry , 21 :1735 , 2013 |
| Abstract : |
| PubMedSearch : Imramovsky_2013_Bioorg.Med.Chem_21_1735 |
| PubMedID: 23462716 |
| Title : Acetylcholinesterase-inhibiting activity of salicylanilide N-alkylcarbamates and their molecular docking - Imramovsky_2012_Molecules_17_10142 |
| Author(s) : Imramovsky A , Stepankova S , Vanco J , Pauk K , Monreal-Ferriz J , Vinsova J , Jampilek J |
| Ref : Molecules , 17 :10142 , 2012 |
| Abstract : |
| PubMedSearch : Imramovsky_2012_Molecules_17_10142 |
| PubMedID: 22922284 |
| Title : 1,3-substituted imidazolidine-2,4,5-triones: synthesis and inhibition of cholinergic enzymes - Pejchal_2011_Molecules_16_7565 |
| Author(s) : Pejchal V , Stepankova S , Padelkova Z , Imramovsky A , Jampilek J |
| Ref : Molecules , 16 :7565 , 2011 |
| Abstract : |
| PubMedSearch : Pejchal_2011_Molecules_16_7565 |
| PubMedID: 21894089 |
| Title : Inhibition of acetylcholinesterase by 14 achiral and five chiral imidazole derivates - Kovarova_2010_Bioresour.Technol_101_6281 |
| Author(s) : Kovarova M , Komers K , Stepankova S , Cegan A |
| Ref : Bioresour Technol , 101 :6281 , 2010 |
| Abstract : |
| PubMedSearch : Kovarova_2010_Bioresour.Technol_101_6281 |
| PubMedID: 20335028 |
| Title : Inhibition of cholinesterase by dialkylcarbamates - Stepankova_2007_Z.Naturforsch.C_62_308 |
| Author(s) : Stepankova S , Komers K , Komersova A , Masopustova M , Cegan A |
| Ref : Z Naturforsch C , 62 :308 , 2007 |
| Abstract : |
| PubMedSearch : Stepankova_2007_Z.Naturforsch.C_62_308 |
| PubMedID: 17542500 |
| Title : In vitro inhibition of cholinesterases by carbamates--a kinetic study - Komersova_2007_Z.Naturforsch.C_62_305 |
| Author(s) : Komersova A , Masopustova M , Komers K , Stepankova S , Cegan A |
| Ref : Z Naturforsch C , 62 :305 , 2007 |
| Abstract : |
| PubMedSearch : Komersova_2007_Z.Naturforsch.C_62_305 |
| PubMedID: 17542499 |
| Title : Kinetics of 13 new cholinesterase inhibitors - Zdrazilova_2006_Z.Naturforsch.C_61_611 |
| Author(s) : Zdrazilova P , Stepankova S , Komersova A , Vranova M , Komers K , Cegan A |
| Ref : Z Naturforsch C , 61 :611 , 2006 |
| Abstract : |
| PubMedSearch : Zdrazilova_2006_Z.Naturforsch.C_61_611 |
| PubMedID: 16989325 |
| Title : Kinetics of total enzymatic hydrolysis of acetylcholine and acetylthiocholine - Zdrazilova_2006_Z.Naturforsch.C_61_289 |
| Author(s) : Zdrazilova P , Stepankova S , Vranova M , Komers K , Komersova A , Cegan A |
| Ref : Z Naturforsch C , 61 :289 , 2006 |
| Abstract : |
| PubMedSearch : Zdrazilova_2006_Z.Naturforsch.C_61_289 |
| PubMedID: 16729592 |
| Title : Two new methods monitoring kinetics of hydrolysis of acetylcholine and acetylthiocholine - Stepankova_2005_Z.Naturforsch.C_60_943 |
| Author(s) : Stepankova S , Vranova M , Zdrazilova P , Komers K , Komersova A , Cegan A |
| Ref : Z Naturforsch C , 60 :943 , 2005 |
| Abstract : |
| PubMedSearch : Stepankova_2005_Z.Naturforsch.C_60_943 |
| PubMedID: 16402558 |
| Title : Half-inhibition concentrations of new cholinesterase inhibitors - Zdrazilova_2004_Z.Naturforsch.C_59_293 |
| Author(s) : Zdrazilova P , Stepankova S , Komers K , Ventura K , Cegan A |
| Ref : Z Naturforsch C , 59 :293 , 2004 |
| Abstract : |
| PubMedSearch : Zdrazilova_2004_Z.Naturforsch.C_59_293 |
| PubMedID: 15241943 |