| Title : Mitigation of Acetylcholine Esterase Activity in the 1,7-Diazacarbazole Series of Inhibitors of Checkpoint Kinase 1 - Gazzard_2015_J.Med.Chem_58_5053 |
| Author(s) : Gazzard L , Williams K , Chen H , Axford L , Blackwood E , Burton B , Chapman K , Crackett P , Drobnick J , Ellwood C , Epler J , Flagella M , Gancia E , Gill M , Goodacre S , Halladay J , Hewitt J , Hunt H , Kintz S , Lyssikatos J , Macleod C , Major S , Medard G , Narukulla R , Ramiscal J , Schmidt S , Seward E , Wiesmann C , Wu P , Yee S , Yen I , Malek S |
| Ref : Journal of Medicinal Chemistry , 58 :5053 , 2015 |
| Abstract : |
| PubMedSearch : Gazzard_2015_J.Med.Chem_58_5053 |
| PubMedID: 25988399 |
| Title : Synthesis and structure-activity relationship of N-acyl-Gly-, N-acyl-Sar- and N-blocked-boroPro inhibitors of FAP, DPP4, and POP - Tran_2007_Bioorg.Med.Chem.Lett_17_1438 |
| Author(s) : Tran T , Quan C , Edosada CY , Mayeda M , Wiesmann C , Sutherlin D , Wolf BB |
| Ref : Bioorganic & Medicinal Chemistry Lett , 17 :1438 , 2007 |
| Abstract : |
| PubMedSearch : Tran_2007_Bioorg.Med.Chem.Lett_17_1438 |
| PubMedID: 17174090 |
| Title : Ala657 and conserved active site residues promote fibroblast activation protein endopeptidase activity via distinct mechanisms of transition state stabilization - Meadows_2007_Biochemistry_46_4598 |
| Author(s) : Meadows SA , Edosada CY , Mayeda M , Tran T , Quan C , Raab H , Wiesmann C , Wolf BB |
| Ref : Biochemistry , 46 :4598 , 2007 |
| Abstract : |
| PubMedSearch : Meadows_2007_Biochemistry_46_4598 |
| PubMedID: 17381073 |
| Title : Selective inhibition of fibroblast activation protein protease based on dipeptide substrate specificity - Edosada_2006_J.Biol.Chem_281_7437 |
| Author(s) : Edosada CY , Quan C , Wiesmann C , Tran T , Sutherlin D , Reynolds M , Elliott JM , Raab H , Fairbrother W , Wolf BB |
| Ref : Journal of Biological Chemistry , 281 :7437 , 2006 |
| Abstract : |
| PubMedSearch : Edosada_2006_J.Biol.Chem_281_7437 |
| PubMedID: 16410248 |