Title : A Comparison of Polysorbates and Alternative Surfactants for Interfacial Stress Protection and Mitigation of Fatty Acid Particle Formation in the Presence of an Esterase - Roy_2024_J.Pharm.Sci__ |
Author(s) : Roy I , Wuchner K , Stahl P , Tran T , Yaragudi N |
Ref : J Pharm Sci , : , 2024 |
Abstract : |
PubMedSearch : Roy_2024_J.Pharm.Sci__ |
PubMedID: 39009347 |
Title : A Comparison of Polysorbates and Alternative Surfactants for Interfacial Stress Protection and Mitigation of Fatty Acid Particle Formation in the Presence of an Esterase - Roy_2024_J.Pharm.Sci__ |
Author(s) : Roy I , Wuchner K , Stahl P , Tran T , Yaragudi N |
Ref : J Pharm Sci , : , 2024 |
Abstract : |
PubMedSearch : Roy_2024_J.Pharm.Sci__ |
PubMedID: 39009347 |
Title : An enolase inhibitor for the targeted treatment of ENO1-deleted cancers - Lin_2020_Nat.Metab_2_1413 |
Author(s) : Lin YH , Satani N , Hammoudi N , Yan VC , Barekatain Y , Khadka S , Ackroyd JJ , Georgiou DK , Pham CD , Arthur K , Maxwell D , Peng Z , Leonard PG , Czako B , Pisaneschi F , Mandal P , Sun Y , Zielinski R , Pando SC , Wang X , Tran T , Xu Q , Wu Q , Jiang Y , Kang Z , Asara JM , Priebe W , Bornmann W , Marszalek JR , DePinho RA , Muller FL |
Ref : Nat Metab , 2 :1413 , 2020 |
Abstract : |
PubMedSearch : Lin_2020_Nat.Metab_2_1413 |
PubMedID: 33230295 |
Title : An enolase inhibitor for the targeted treatment of ENO1-deleted cancers - Lin_2020_Nat.Metab_2_1413 |
Author(s) : Lin YH , Satani N , Hammoudi N , Yan VC , Barekatain Y , Khadka S , Ackroyd JJ , Georgiou DK , Pham CD , Arthur K , Maxwell D , Peng Z , Leonard PG , Czako B , Pisaneschi F , Mandal P , Sun Y , Zielinski R , Pando SC , Wang X , Tran T , Xu Q , Wu Q , Jiang Y , Kang Z , Asara JM , Priebe W , Bornmann W , Marszalek JR , DePinho RA , Muller FL |
Ref : Nat Metab , 2 :1413 , 2020 |
Abstract : |
PubMedSearch : Lin_2020_Nat.Metab_2_1413 |
PubMedID: 33230295 |
Title : Understanding the Enzyme-Ligand Complex: Insights from All-Atom Simulations of Butyrylcholinesterase Inhibition - Alvarado_2019_J.Biomol.Struct.Dyn__1 |
Author(s) : Alvarado W , Ladd Bremer P , Choy A , Dinh HN , Eung A , Gonzalez J , Ly P , Tran T , Nakayama K , Schwans JP , Sorin EJ |
Ref : J Biomol Struct Dyn , :1 , 2019 |
Abstract : |
PubMedSearch : Alvarado_2019_J.Biomol.Struct.Dyn__1 |
PubMedID: 30909811 |
Title : Understanding the Enzyme-Ligand Complex: Insights from All-Atom Simulations of Butyrylcholinesterase Inhibition - Alvarado_2019_J.Biomol.Struct.Dyn__1 |
Author(s) : Alvarado W , Ladd Bremer P , Choy A , Dinh HN , Eung A , Gonzalez J , Ly P , Tran T , Nakayama K , Schwans JP , Sorin EJ |
Ref : J Biomol Struct Dyn , :1 , 2019 |
Abstract : |
PubMedSearch : Alvarado_2019_J.Biomol.Struct.Dyn__1 |
PubMedID: 30909811 |
Title : Synthesis, biochemical evaluation, and molecular modeling studies of aryl and arylalkyl di-n-butyl phosphates, effective butyrylcholinesterase inhibitors - Nakayama_2017_Bioorg.Med.Chem_25_3171 |
Author(s) : Nakayama K , Schwans JP , Sorin EJ , Tran T , Gonzalez J , Arteaga E , McCoy S , Alvarado W |
Ref : Bioorganic & Medicinal Chemistry , 25 :3171 , 2017 |
Abstract : |
PubMedSearch : Nakayama_2017_Bioorg.Med.Chem_25_3171 |
PubMedID: 28416102 |
Title : Synthesis, biochemical evaluation, and molecular modeling studies of aryl and arylalkyl di-n-butyl phosphates, effective butyrylcholinesterase inhibitors - Nakayama_2017_Bioorg.Med.Chem_25_3171 |
Author(s) : Nakayama K , Schwans JP , Sorin EJ , Tran T , Gonzalez J , Arteaga E , McCoy S , Alvarado W |
Ref : Bioorganic & Medicinal Chemistry , 25 :3171 , 2017 |
Abstract : |
PubMedSearch : Nakayama_2017_Bioorg.Med.Chem_25_3171 |
PubMedID: 28416102 |
Title : 18F-ASEM, a radiolabeled antagonist for imaging the alpha7-nicotinic acetylcholine receptor with PET - Horti_2014_J.Nucl.Med_55_672 |
Author(s) : Horti AG , Gao Y , Kuwabara H , Wang Y , Abazyan S , Yasuda RP , Tran T , Xiao Y , Sahibzada N , Holt DP , Kellar KJ , Pletnikov MV , Pomper MG , Wong DF , Dannals RF |
Ref : J Nucl Med , 55 :672 , 2014 |
Abstract : |
PubMedSearch : Horti_2014_J.Nucl.Med_55_672 |
PubMedID: 24556591 |
Title : 18F-ASEM, a radiolabeled antagonist for imaging the alpha7-nicotinic acetylcholine receptor with PET - Horti_2014_J.Nucl.Med_55_672 |
Author(s) : Horti AG , Gao Y , Kuwabara H , Wang Y , Abazyan S , Yasuda RP , Tran T , Xiao Y , Sahibzada N , Holt DP , Kellar KJ , Pletnikov MV , Pomper MG , Wong DF , Dannals RF |
Ref : J Nucl Med , 55 :672 , 2014 |
Abstract : |
PubMedSearch : Horti_2014_J.Nucl.Med_55_672 |
PubMedID: 24556591 |
Title : Derivatives of dibenzothiophene for positron emission tomography imaging of alpha7-nicotinic acetylcholine receptors - Gao_2013_J.Med.Chem_56_7574 |
Author(s) : Gao Y , Kellar KJ , Yasuda RP , Tran T , Xiao Y , Dannals RF , Horti AG |
Ref : Journal of Medicinal Chemistry , 56 :7574 , 2013 |
Abstract : |
PubMedSearch : Gao_2013_J.Med.Chem_56_7574 |
PubMedID: 24050653 |
Title : Design, synthesis and discovery of picomolar selective alpha4beta2 nicotinic acetylcholine receptor ligands - Yenugonda_2013_J.Med.Chem_56_8404 |
Author(s) : Yenugonda VM , Xiao Y , Levin ED , Rezvani AH , Tran T , Al-Muhtasib N , Sahibzada N , Xie T , Wells C , Slade S , Johnson JE , Dakshanamurthy S , Kong HS , Tomita Y , Liu Y , Paige M , Kellar KJ , Brown ML |
Ref : Journal of Medicinal Chemistry , 56 :8404 , 2013 |
Abstract : |
PubMedSearch : Yenugonda_2013_J.Med.Chem_56_8404 |
PubMedID: 24047231 |
Title : Chemistry and pharmacological studies of 3-alkoxy-2,5-disubstituted-pyridinyl compounds as novel selective alpha4beta2 nicotinic acetylcholine receptor ligands that reduce alcohol intake in rats - Liu_2013_J.Med.Chem_56_3000 |
Author(s) : Liu Y , Richardson J , Tran T , Al-Muhtasib N , Xie T , Yenugonda VM , Sexton HG , Rezvani AH , Levin ED , Sahibzada N , Kellar KJ , Brown ML , Xiao Y , Paige M |
Ref : Journal of Medicinal Chemistry , 56 :3000 , 2013 |
Abstract : |
PubMedSearch : Liu_2013_J.Med.Chem_56_3000 |
PubMedID: 23540678 |
Title : Design, synthesis and discovery of picomolar selective alpha4beta2 nicotinic acetylcholine receptor ligands - Yenugonda_2013_J.Med.Chem_56_8404 |
Author(s) : Yenugonda VM , Xiao Y , Levin ED , Rezvani AH , Tran T , Al-Muhtasib N , Sahibzada N , Xie T , Wells C , Slade S , Johnson JE , Dakshanamurthy S , Kong HS , Tomita Y , Liu Y , Paige M , Kellar KJ , Brown ML |
Ref : Journal of Medicinal Chemistry , 56 :8404 , 2013 |
Abstract : |
PubMedSearch : Yenugonda_2013_J.Med.Chem_56_8404 |
PubMedID: 24047231 |
Title : Derivatives of dibenzothiophene for positron emission tomography imaging of alpha7-nicotinic acetylcholine receptors - Gao_2013_J.Med.Chem_56_7574 |
Author(s) : Gao Y , Kellar KJ , Yasuda RP , Tran T , Xiao Y , Dannals RF , Horti AG |
Ref : Journal of Medicinal Chemistry , 56 :7574 , 2013 |
Abstract : |
PubMedSearch : Gao_2013_J.Med.Chem_56_7574 |
PubMedID: 24050653 |
Title : Chemistry and pharmacological studies of 3-alkoxy-2,5-disubstituted-pyridinyl compounds as novel selective alpha4beta2 nicotinic acetylcholine receptor ligands that reduce alcohol intake in rats - Liu_2013_J.Med.Chem_56_3000 |
Author(s) : Liu Y , Richardson J , Tran T , Al-Muhtasib N , Xie T , Yenugonda VM , Sexton HG , Rezvani AH , Levin ED , Sahibzada N , Kellar KJ , Brown ML , Xiao Y , Paige M |
Ref : Journal of Medicinal Chemistry , 56 :3000 , 2013 |
Abstract : |
PubMedSearch : Liu_2013_J.Med.Chem_56_3000 |
PubMedID: 23540678 |
Title : Identification and pharmacological characterization of multiple allosteric binding sites on the free fatty acid 1 receptor - Lin_2012_Mol.Pharmacol_82_843 |
Author(s) : Lin DC , Guo Q , Luo J , Zhang J , Nguyen K , Chen M , Tran T , Dransfield PJ , Brown SP , Houze J , Vimolratana M , Jiao XY , Wang Y , Birdsall NJ , Swaminath G |
Ref : Molecular Pharmacology , 82 :843 , 2012 |
Abstract : |
PubMedSearch : Lin_2012_Mol.Pharmacol_82_843 |
PubMedID: 22859723 |
Title : Identification and pharmacological characterization of multiple allosteric binding sites on the free fatty acid 1 receptor - Lin_2012_Mol.Pharmacol_82_843 |
Author(s) : Lin DC , Guo Q , Luo J , Zhang J , Nguyen K , Chen M , Tran T , Dransfield PJ , Brown SP , Houze J , Vimolratana M , Jiao XY , Wang Y , Birdsall NJ , Swaminath G |
Ref : Molecular Pharmacology , 82 :843 , 2012 |
Abstract : |
PubMedSearch : Lin_2012_Mol.Pharmacol_82_843 |
PubMedID: 22859723 |
Title : Poster: Pharmacological properties of sazetidine A, a selective ligand of alpha4\/beta2 nicotinic acetylcholine receptors - |
Author(s) : Xiao Y , Tuan E , Yasuda RP , Sahibzada N , Wolfe BB , Horton L , Tran T , Al-Muhtasib N , Iwueze AF , Dipietro JR , Xie T , Paige M , Brown ML , Kellar KJ |
Ref : Biochemical Pharmacology , 82 :1029 , 2011 |
PubMedID: |
Title : Poster: Pharmacological properties of sazetidine A, a selective ligand of alpha4\/beta2 nicotinic acetylcholine receptors - |
Author(s) : Xiao Y , Tuan E , Yasuda RP , Sahibzada N , Wolfe BB , Horton L , Tran T , Al-Muhtasib N , Iwueze AF , Dipietro JR , Xie T , Paige M , Brown ML , Kellar KJ |
Ref : Biochemical Pharmacology , 82 :1029 , 2011 |
PubMedID: |
Title : Activity-dependent changes in cholinergic innervation of the mouse olfactory bulb - Salcedo_2011_PLoS.One_6_e25441 |
Author(s) : Salcedo E , Tran T , Ly X , Lopez R , Barbica C , Restrepo D , Vijayaraghavan S |
Ref : PLoS ONE , 6 :e25441 , 2011 |
Abstract : |
PubMedSearch : Salcedo_2011_PLoS.One_6_e25441 |
PubMedID: 22053179 |
Title : Activity-dependent changes in cholinergic innervation of the mouse olfactory bulb - Salcedo_2011_PLoS.One_6_e25441 |
Author(s) : Salcedo E , Tran T , Ly X , Lopez R , Barbica C , Restrepo D , Vijayaraghavan S |
Ref : PLoS ONE , 6 :e25441 , 2011 |
Abstract : |
PubMedSearch : Salcedo_2011_PLoS.One_6_e25441 |
PubMedID: 22053179 |
Title : Synthesis and structure-activity relationship of N-acyl-Gly-, N-acyl-Sar- and N-blocked-boroPro inhibitors of FAP, DPP4, and POP - Tran_2007_Bioorg.Med.Chem.Lett_17_1438 |
Author(s) : Tran T , Quan C , Edosada CY , Mayeda M , Wiesmann C , Sutherlin D , Wolf BB |
Ref : Bioorganic & Medicinal Chemistry Lett , 17 :1438 , 2007 |
Abstract : |
PubMedSearch : Tran_2007_Bioorg.Med.Chem.Lett_17_1438 |
PubMedID: 17174090 |
Title : Ala657 and conserved active site residues promote fibroblast activation protein endopeptidase activity via distinct mechanisms of transition state stabilization - Meadows_2007_Biochemistry_46_4598 |
Author(s) : Meadows SA , Edosada CY , Mayeda M , Tran T , Quan C , Raab H , Wiesmann C , Wolf BB |
Ref : Biochemistry , 46 :4598 , 2007 |
Abstract : |
PubMedSearch : Meadows_2007_Biochemistry_46_4598 |
PubMedID: 17381073 |
Title : Synthesis and structure-activity relationship of N-acyl-Gly-, N-acyl-Sar- and N-blocked-boroPro inhibitors of FAP, DPP4, and POP - Tran_2007_Bioorg.Med.Chem.Lett_17_1438 |
Author(s) : Tran T , Quan C , Edosada CY , Mayeda M , Wiesmann C , Sutherlin D , Wolf BB |
Ref : Bioorganic & Medicinal Chemistry Lett , 17 :1438 , 2007 |
Abstract : |
PubMedSearch : Tran_2007_Bioorg.Med.Chem.Lett_17_1438 |
PubMedID: 17174090 |
Title : Ala657 and conserved active site residues promote fibroblast activation protein endopeptidase activity via distinct mechanisms of transition state stabilization - Meadows_2007_Biochemistry_46_4598 |
Author(s) : Meadows SA , Edosada CY , Mayeda M , Tran T , Quan C , Raab H , Wiesmann C , Wolf BB |
Ref : Biochemistry , 46 :4598 , 2007 |
Abstract : |
PubMedSearch : Meadows_2007_Biochemistry_46_4598 |
PubMedID: 17381073 |
Title : Selective inhibition of fibroblast activation protein protease based on dipeptide substrate specificity - Edosada_2006_J.Biol.Chem_281_7437 |
Author(s) : Edosada CY , Quan C , Wiesmann C , Tran T , Sutherlin D , Reynolds M , Elliott JM , Raab H , Fairbrother W , Wolf BB |
Ref : Journal of Biological Chemistry , 281 :7437 , 2006 |
Abstract : |
PubMedSearch : Edosada_2006_J.Biol.Chem_281_7437 |
PubMedID: 16410248 |
Title : Selective inhibition of fibroblast activation protein protease based on dipeptide substrate specificity - Edosada_2006_J.Biol.Chem_281_7437 |
Author(s) : Edosada CY , Quan C , Wiesmann C , Tran T , Sutherlin D , Reynolds M , Elliott JM , Raab H , Fairbrother W , Wolf BB |
Ref : Journal of Biological Chemistry , 281 :7437 , 2006 |
Abstract : |
PubMedSearch : Edosada_2006_J.Biol.Chem_281_7437 |
PubMedID: 16410248 |