Name : X-ray Structure of Novel Biaryl-Based Dipeptidyl peptidase IV inhibitor
Revelation date : 08-Nov-2005
Family : DPP4N_Peptidase_S9
Gene_locus : human-DPP4
PDB file : ESTHER: header of PDB entry RCSB: Full entry
Comment
Qiao, L., Baumann, C.A., Crysler, C.S., Ninan, N.S., Abad, M.C., Spurlino, J.C., Desjarlais, R.L., Kervinen, J., Neeper, M.P., Bayoumy, S.S., Williams, R., Deckman, I.C., Dasgupta, M., Reed, R.L., Huebert, N.D., Tomczuk, B.E., Moriarty, K.J.
Ligand :
Title : Discovery, SAR, and X-ray structure of novel biaryl-based dipeptidyl peptidase IV inhibitors - Qiao_2006_Bioorg.Med.Chem.Lett_16_123 |
Author(s) : Qiao L , Baumann CA , Crysler CS , Ninan NS , Abad MC , Spurlino JC , Desjarlais RL , Kervinen J , Neeper MP , Bayoumy SS , Williams R , Deckman IC , Dasgupta M , Reed RL , Huebert ND , Tomczuk BE , Moriarty KJ |
Ref : Bioorganic & Medicinal Chemistry Lett , 16 :123 , 2006 |
Abstract : Qiao_2006_Bioorg.Med.Chem.Lett_16_123 |
ESTHER : Qiao_2006_Bioorg.Med.Chem.Lett_16_123 |
PubMedSearch : Qiao_2006_Bioorg.Med.Chem.Lett_16_123 |
PubMedID: 16236500 |
Gene_locus related to this paper: human-DPP4 |
PDB-Sum : 2AJL Previously Class, Architecture, Topology and Homologous superfamily - PDB-Sum server
FSSP : 2AJL Fold classification based on Structure-Structure alignment of Proteins - FSSP server
SCOP : 2AJL Structural Classification Of Protein - SCOP server
PROTEOPEDIA : 2AJL 3D, interactive encyclopedia of proteins - PROTEOPEDIA server