Title : The discovery of non-benzimidazole and brain-penetrant prolylcarboxypeptidase inhibitors - Graham_2012_Bioorg.Med.Chem.Lett_22_658 |
Author(s) : Graham TH , Shen HC , Liu W , Xiong Y , Verras A , Bleasby K , Bhatt UR , Chabin RM , Chen D , Chen Q , Garcia-Calvo M , Geissler WM , He H , Lassman ME , Shen Z , Tong X , Tung EC , Xie D , Xu S , Colletti SL , Tata JR , Hale JJ , Pinto S , Shen DM |
Ref : Bioorganic & Medicinal Chemistry Lett , 22 :658 , 2012 |
Abstract : Graham_2012_Bioorg.Med.Chem.Lett_22_658 |
ESTHER : Graham_2012_Bioorg.Med.Chem.Lett_22_658 |
PubMedSearch : Graham_2012_Bioorg.Med.Chem.Lett_22_658 |
PubMedID: 22079761 |
Gene_locus related to this paper: human-PRCP |
Title : Discovery of benzimidazole pyrrolidinyl amides as prolylcarboxypeptidase inhibitors - Shen_2011_Bioorg.Med.Chem.Lett_21_1299 |
Author(s) : Shen HC , Ding FX , Zhou C , Xiong Y , Verras A , Chabin RM , Xu S , Tong X , Xie D , Lassman ME , Bhatt UR , Garcia-Calvo MM , Geissler W , Shen Z , Chen D , SinhaRoy R , Hale JJ , Tata JR , Pinto S , Shen DM , Colletti SL |
Ref : Bioorganic & Medicinal Chemistry Lett , 21 :1299 , 2011 |
Abstract : Shen_2011_Bioorg.Med.Chem.Lett_21_1299 |
ESTHER : Shen_2011_Bioorg.Med.Chem.Lett_21_1299 |
PubMedSearch : Shen_2011_Bioorg.Med.Chem.Lett_21_1299 |
PubMedID: 21315588 |
Gene_locus related to this paper: human-PRCP |
Title : Design and synthesis of prolylcarboxypeptidase (PrCP) inhibitors to validate PrCP as a potential target for obesity - Zhou_2010_J.Med.Chem_53_7251 |
Author(s) : Zhou C , Garcia-Calvo M , Pinto S , Lombardo M , Feng Z , Bender K , Pryor KD , Bhatt UR , Chabin RM , Geissler WM , Shen Z , Tong X , Zhang Z , Wong KK , Roy RS , Chapman KT , Yang L , Xiong Y |
Ref : Journal of Medicinal Chemistry , 53 :7251 , 2010 |
Abstract : Zhou_2010_J.Med.Chem_53_7251 |
ESTHER : Zhou_2010_J.Med.Chem_53_7251 |
PubMedSearch : Zhou_2010_J.Med.Chem_53_7251 |
PubMedID: 20857914 |
Gene_locus related to this paper: human-PRCP |