| Title : Integrated Synthetic, Biophysical, and Computational Investigations of Covalent Inhibitors of Prolyl Oligopeptidase and Fibroblast Activation Protein alpha - Plescia_2019_J.Med.Chem_62_7874 |
| Author(s) : Plescia J , De Cesco S , Patrascu MB , Kurian J , Di Trani J , Dufresne C , Wahba AS , Janmamode N , Mittermaier AK , Moitessier N |
| Ref : Journal of Medicinal Chemistry , 62 :7874 , 2019 |
| Abstract : |
| PubMedSearch : Plescia_2019_J.Med.Chem_62_7874 |
| PubMedID: 31393718 |
| Title : 3-Oxo-hexahydro-1H-isoindole-4-carboxylic Acid as a Drug Chiral Bicyclic Scaffold: Structure-Based Design and Preparation of Conformationally Constrained Covalent and Noncovalent Prolyl Oligopeptidase Inhibitors - Mariaule_2016_J.Med.Chem_59_4221 |
| Author(s) : Mariaule G , De Cesco S , Airaghi F , Kurian J , Schiavini P , Rocheleau S , Huskic I , Auclair K , Mittermaier A , Moitessier N |
| Ref : Journal of Medicinal Chemistry , 59 :4221 , 2016 |
| Abstract : |
| PubMedSearch : Mariaule_2016_J.Med.Chem_59_4221 |
| PubMedID: 26619267 |
| Gene_locus related to this paper: human-PREP |
| Title : Virtual screening and computational optimization for the discovery of covalent prolyl oligopeptidase inhibitors with activity in human cells - De Cesco_2012_J.Med.Chem_55_6306 |
| Author(s) : De Cesco S , Deslandes S , Therrien E , Levan D , Cueto M , Schmidt R , Cantin LD , Mittermaier A , Juillerat-Jeanneret L , Moitessier N |
| Ref : Journal of Medicinal Chemistry , 55 :6306 , 2012 |
| Abstract : |
| PubMedSearch : De Cesco_2012_J.Med.Chem_55_6306 |
| PubMedID: 22765237 |