Title : Modulating the selectivity of inhibitors for prolyl oligopeptidase inhibitors and fibroblast activation protein-alpha for different indications - Plescia_2022_Eur.J.Med.Chem_240_114543 |
Author(s) : Plescia J , Hedou D , Pousse ME , Labarre A , Dufresne C , Mittermaier A , Moitessier N |
Ref : Eur Journal of Medicinal Chemistry , 240 :114543 , 2022 |
Abstract : |
PubMedSearch : Plescia_2022_Eur.J.Med.Chem_240_114543 |
PubMedID: 35797897 |
Gene_locus related to this paper: human-FAP , human-PREP |
Title : Discovery of covalent prolyl oligopeptidase boronic ester inhibitors - Plescia_2020_Eur.J.Med.Chem_185_111783 |
Author(s) : Plescia J , Dufresne C , Janmamode N , Wahba AS , Mittermaier AK , Moitessier N |
Ref : Eur Journal of Medicinal Chemistry , 185 :111783 , 2020 |
Abstract : |
PubMedSearch : Plescia_2020_Eur.J.Med.Chem_185_111783 |
PubMedID: 31732257 |
Gene_locus related to this paper: human-PREP |
Title : Integrated Synthetic, Biophysical, and Computational Investigations of Covalent Inhibitors of Prolyl Oligopeptidase and Fibroblast Activation Protein alpha - Plescia_2019_J.Med.Chem_62_7874 |
Author(s) : Plescia J , De Cesco S , Patrascu MB , Kurian J , Di Trani J , Dufresne C , Wahba AS , Janmamode N , Mittermaier AK , Moitessier N |
Ref : Journal of Medicinal Chemistry , 62 :7874 , 2019 |
Abstract : |
PubMedSearch : Plescia_2019_J.Med.Chem_62_7874 |
PubMedID: 31393718 |