Title : Three-dimensional rational approach to the discovery of potent substituted cyclopropyl urea soluble epoxide hydrolase inhibitors - Takai_2015_Bioorg.Med.Chem.Lett_25_1705 |
Author(s) : Takai K , Chiyo N , Nakajima T , Nariai T , Ishikawa C , Nakatani S , Ikeno A , Yamamoto S , Sone T |
Ref : Bioorganic & Medicinal Chemistry Lett , 25 :1705 , 2015 |
Abstract : |
PubMedSearch : Takai_2015_Bioorg.Med.Chem.Lett_25_1705 |
PubMedID: 25800114 |
Gene_locus related to this paper: human-EPHX2 |
Title : Structure-based optimization of cyclopropyl urea derivatives as potent soluble epoxide hydrolase inhibitors for potential decrease of renal injury without hypotensive action - Takai_2014_Bioorg.Med.Chem_22_1548 |
Author(s) : Takai K , Nakajima T , Takanashi Y , Sone T , Nariai T , Chiyo N , Nakatani S , Ishikawa C , Yamaguchi N , Fujita K , Yamada K |
Ref : Bioorganic & Medicinal Chemistry , 22 :1548 , 2014 |
Abstract : |
PubMedSearch : Takai_2014_Bioorg.Med.Chem_22_1548 |
PubMedID: 24530032 |
Title : Anti-inflammatory action of donepezil ameliorates tau pathology, synaptic loss, and neurodegeneration in a tauopathy mouse model - Yoshiyama_2010_J.Alzheimers.Dis_22_295 |
Author(s) : Yoshiyama Y , Kojima A , Ishikawa C , Arai K |
Ref : J Alzheimers Dis , 22 :295 , 2010 |
Abstract : |
PubMedSearch : Yoshiyama_2010_J.Alzheimers.Dis_22_295 |
PubMedID: 20847440 |
Title : The p75 neurotrophin receptor promotes amyloid-beta(1-42)-induced neuritic dystrophy in vitro and in vivo - Knowles_2009_J.Neurosci_29_10627 |
Author(s) : Knowles JK , Rajadas J , Nguyen TV , Yang T , LeMieux MC , Vander Griend L , Ishikawa C , Massa SM , Wyss-Coray T , Longo FM |
Ref : Journal of Neuroscience , 29 :10627 , 2009 |
Abstract : |
PubMedSearch : Knowles_2009_J.Neurosci_29_10627 |
PubMedID: 19710315 |