| Title : Discovery of non-covalent dipeptidyl peptidase IV inhibitors which induce a conformational change in the active site - Sheehan_2007_Bioorg.Med.Chem.Lett_17_1765 |
| Author(s) : Sheehan SM , Mest HJ , Watson BM , Klimkowski VJ , Timm DE , Cauvin A , Parsons SH , Shi Q , Canada EJ , Wiley MR , Ruehter G , Evers B , Petersen S , Blaszczak LC , Pulley SR , Margolis BJ , Wishart GN , Renson B , Hankotius D , Mohr M , Zechel JC , Michael Kalbfleisch J , Dingess-Hammond EA , Boelke A , Weichert AG |
| Ref : Bioorganic & Medicinal Chemistry Lett , 17 :1765 , 2007 |
| Abstract : |
| PubMedSearch : Sheehan_2007_Bioorg.Med.Chem.Lett_17_1765 |
| PubMedID: 17239592 |
| Gene_locus related to this paper: human-DPP4 |
| Title : Poster: Synthesis and structure-activity relationship of 3-(pyrazinyl)- 1, 2, 5, 6-tetrahydro-1-methylpyridines. Construction of a molecular model for the M-1 pharmacophore - |
| Author(s) : Ward JS , Merritt L , Klimkowski VJ , Lamb ML , Mitch CH , Bymaster FP , Sawyer BD , Shannon HE , Olesen PH , Honore T , Sheardown MJ , Sauerberg P |
| Ref : Life Sciences , 52(5-6) :549 , 1993 |
| PubMedID: |
| Title : Structure\/function relationships of muscarinic acetylcholine receptors - Brann_1993_Life.Sci_52(5-6)_405 |
| Author(s) : Brann MR , Klimkowski VJ , Ellis J |
| Ref : Life Sciences , 52 :405 , 1993 |
| Abstract : |
| PubMedSearch : Brann_1993_Life.Sci_52(5-6)_405 |
| PubMedID: 7680090 |
| Title : Novel functional M1 selective muscarinic agonists. 2. Synthesis and structure-activity relationships of 3-pyrazinyl-1,2,5,6-tetrahydro-1-methylpyridines. Construction of a molecular model for the M1 pharmacophore - Ward_1992_J.Med.Chem_35_4011 |
| Author(s) : Ward JS , Merritt L , Klimkowski VJ , Lamb ML , Mitch CH , Bymaster FP , Sawyer BD , Shannon HE , Olesen PH , Honore T , Sheardown MJ , Sauerberg P |
| Ref : Journal of Medicinal Chemistry , 35 :4011 , 1992 |
| Abstract : |
| PubMedSearch : Ward_1992_J.Med.Chem_35_4011 |
| PubMedID: 1433209 |