| Title : Structure and Dynamics of an Archeal Monoglyceride Lipase from Palaeococcus ferrophilus as Revealed by Crystallography and In Silico Analysis - Labar_2021_Biomolecules_11_533 |
| Author(s) : Labar G , Brandt N , Flaba A , Wouters J , Leherte L |
| Ref : Biomolecules , 11 :533 , 2021 |
| Abstract : |
| PubMedSearch : Labar_2021_Biomolecules_11_533 |
| PubMedID: 33916727 |
| Gene_locus related to this paper: 9eury-6QE2 |
| Title : (S)-1-(Pent-4'-enoyl)-4-(hydroxymethyl)-azetidin-2-one derivatives as inhibitors of human fatty acid amide hydrolase (hFAAH): synthesis, biological evaluation and molecular modelling - Caruano_2014_J.Enzyme.Inhib.Med.Chem_29_654 |
| Author(s) : Caruano J , Feledziak M , Labar G , Michaux C , Perpete EA , Muccioli GG , Robiette R , Marchand-Brynaert J |
| Ref : Journal of enzyme inhibition and medicinal chemistry , 29 :654 , 2014 |
| Abstract : |
| PubMedSearch : Caruano_2014_J.Enzyme.Inhib.Med.Chem_29_654 |
| PubMedID: 24102523 |
| Title : Development and characterization of endocannabinoid hydrolases FAAH and MAGL inhibitors bearing a benzotriazol-1-yl carboxamide scaffold - Morera_2012_Bioorg.Med.Chem_20_6260 |
| Author(s) : Morera L , Labar G , Ortar G , Lambert DM |
| Ref : Bioorganic & Medicinal Chemistry , 20 :6260 , 2012 |
| Abstract : |
| PubMedSearch : Morera_2012_Bioorg.Med.Chem_20_6260 |
| PubMedID: 23036333 |
| Title : Synthesis and pharmacological evaluation of 2,4-dinitroaryldithiocarbamate derivatives as novel monoacylglycerol lipase inhibitors - Kapanda_2012_J.Med.Chem_55_5774 |
| Author(s) : Kapanda CN , Masquelier J , Labar G , Muccioli GG , Poupaert JH , Lambert DM |
| Ref : Journal of Medicinal Chemistry , 55 :5774 , 2012 |
| Abstract : |
| PubMedSearch : Kapanda_2012_J.Med.Chem_55_5774 |
| PubMedID: 22651858 |
| Title : Benzisothiazolinone as a useful template for the design of new monoacylglycerol lipase inhibitors: investigation of the target residues and comparison with octhilinone - Matuszak_2011_Bioorg.Med.Chem.Lett_21_7321 |
| Author(s) : Matuszak N , Es Saadi B , Labar G , Marchand-Brynaert J , Lambert DM |
| Ref : Bioorganic & Medicinal Chemistry Lett , 21 :7321 , 2011 |
| Abstract : |
| PubMedSearch : Matuszak_2011_Bioorg.Med.Chem.Lett_21_7321 |
| PubMedID: 22056744 |
| Gene_locus related to this paper: human-ABHD6 |
| Title : Crystal structure of the human monoacylglycerol lipase, a key actor in endocannabinoid signaling - Labar_2010_Chembiochem_11_218 |
| Author(s) : Labar G , Bauvois C , Borel F , Ferrer JL , Wouters J , Lambert DM |
| Ref : Chembiochem , 11 :218 , 2010 |
| Abstract : |
| PubMedSearch : Labar_2010_Chembiochem_11_218 |
| PubMedID: 19957260 |
| Gene_locus related to this paper: human-MGLL |
| Title : A review on the monoacylglycerol lipase: at the interface between fat and endocannabinoid signalling - Labar_2010_Curr.Med.Chem_17_2588 |
| Author(s) : Labar G , Wouters J , Lambert DM |
| Ref : Curr Med Chem , 17 :2588 , 2010 |
| Abstract : |
| PubMedSearch : Labar_2010_Curr.Med.Chem_17_2588 |
| PubMedID: 20491633 |
| Title : Bis(dialkylaminethiocarbonyl)disulfides as potent and selective monoglyceride lipase inhibitors - Kapanda_2009_J.Med.Chem_52_7310 |
| Author(s) : Kapanda CN , Muccioli GG , Labar G , Poupaert JH , Lambert DM |
| Ref : Journal of Medicinal Chemistry , 52 :7310 , 2009 |
| Abstract : |
| PubMedSearch : Kapanda_2009_J.Med.Chem_52_7310 |
| PubMedID: 19883085 |
| Title : Synthesis and in vitro evaluation of N-substituted maleimide derivatives as selective monoglyceride lipase inhibitors - Matuszak_2009_J.Med.Chem_52_7410 |
| Author(s) : Matuszak N , Muccioli GG , Labar G , Lambert DM |
| Ref : Journal of Medicinal Chemistry , 52 :7410 , 2009 |
| Abstract : |
| PubMedSearch : Matuszak_2009_J.Med.Chem_52_7410 |
| PubMedID: 19583260 |
| Title : beta-Lactams derived from a carbapenem chiron are selective inhibitors of human fatty acid amide hydrolase versus human monoacylglycerol lipase - Feledziak_2009_J.Med.Chem_52_7054 |
| Author(s) : Feledziak M , Michaux C , Urbach A , Labar G , Muccioli GG , Lambert DM , Marchand-Brynaert J |
| Ref : Journal of Medicinal Chemistry , 52 :7054 , 2009 |
| Abstract : |
| PubMedSearch : Feledziak_2009_J.Med.Chem_52_7054 |
| PubMedID: 19877691 |
| Title : CAY10499, a novel monoglyceride lipase inhibitor evidenced by an expeditious MGL assay - Muccioli_2008_Chembiochem_9_2704 |
| Author(s) : Muccioli GG , Labar G , Lambert DM |
| Ref : Chembiochem , 9 :2704 , 2008 |
| Abstract : |
| PubMedSearch : Muccioli_2008_Chembiochem_9_2704 |
| PubMedID: 18855964 |
| Gene_locus related to this paper: human-MGLL |
| Title : A MBP-FAAH fusion protein as a tool to produce human and rat fatty acid amide hydrolase: expression and pharmacological comparison - Labar_2008_Amino.Acids_34_127 |
| Author(s) : Labar G , Vliet FV , Wouters J , Lambert DM |
| Ref : Amino Acids , 34 :127 , 2008 |
| Abstract : |
| PubMedSearch : Labar_2008_Amino.Acids_34_127 |
| PubMedID: 17476568 |
| Title : Disulfiram is an inhibitor of human purified monoacylglycerol lipase, the enzyme regulating 2-arachidonoylglycerol signaling - Labar_2007_Chembiochem_8_1293 |
| Author(s) : Labar G , Bauvois C , Muccioli GG , Wouters J , Lambert DM |
| Ref : Chembiochem , 8 :1293 , 2007 |
| Abstract : |
| PubMedSearch : Labar_2007_Chembiochem_8_1293 |
| PubMedID: 17579916 |
| Gene_locus related to this paper: human-MGLL |
| Title : Lack of selectivity of URB602 for 2-oleoylglycerol compared to anandamide hydrolysis in vitro - Vandevoorde_2007_Br.J.Pharmacol_150_186 |
| Author(s) : Vandevoorde S , Jonsson KO , Labar G , Persson E , Lambert DM , Fowler CJ |
| Ref : British Journal of Pharmacology , 150 :186 , 2007 |
| Abstract : |
| PubMedSearch : Vandevoorde_2007_Br.J.Pharmacol_150_186 |
| PubMedID: 17143303 |