Title : Exploration of novel triazolo-thiadiazine hybrids of deferasirox as multi-target-directed anti-neuroinflammatory agents with structure-activity relationship (SAR): a new treatment opportunity for Alzheimer's disease - Shakir_2025_RSC.Adv_15_101 |
Author(s) : Shakir SA , Rashid U , Marryum , Fatima N , Ejaz SA , Fayyaz A , Ullah MZ , Saeed A , Khan A , Al Harrasi A , Mumtaz A |
Ref : RSC Adv , 15 :101 , 2025 |
Abstract : |
PubMedSearch : Shakir_2025_RSC.Adv_15_101 |
PubMedID: 39758929 |
Title : Plant extracts as emerging modulators of neuroinflammation and immune receptors in Alzheimer's pathogenesis - Mohamed_2024_Heliyon_10_e35943 |
Author(s) : Mohamed IE , Osman EE , Saeed A , Ming LC , Goh KW , Razi P , Abdullah ADI , Dahab M |
Ref : Heliyon , 10 :e35943 , 2024 |
Abstract : |
PubMedSearch : Mohamed_2024_Heliyon_10_e35943 |
PubMedID: 39229544 |
Title : Design, Synthesis, QSAR studies, and Molecular Modeling of Some Novel Bis Methyl 2-[3-(benzo[d]thiazol-2-yl)-2-terephthaloyl-bis-4-oxo-thiazolidin-5-ylidene]acetates and Screening of their Antioxidant and Enzyme Inhibition Properties - Naseem_2023_Curr.Org.Synth__ |
Author(s) : Naseem M , Rafique H , Tayyab M , Saeed A , Mumtaz A |
Ref : Curr Org Synth , : , 2023 |
Abstract : |
PubMedSearch : Naseem_2023_Curr.Org.Synth__ |
PubMedID: 37670713 |
Title : Synthesis and evaluation of novel xanthene-based thiazoles as potential antidiabetic agents - Naseem_2022_Arch.Pharm.(Weinheim)__e2200356 |
Author(s) : Naseem S , Shafiq Z , Taslimi P , Hussain S , Taskin-Tok T , Kisa D , Saeed A , Temirak A , Tahir MN , Rauf K , El-Gokha A |
Ref : Arch Pharm (Weinheim) , :e2200356 , 2022 |
Abstract : |
PubMedSearch : Naseem_2022_Arch.Pharm.(Weinheim)__e2200356 |
PubMedID: 36220614 |
Title : Facile synthesis, crystal structure, biological evaluation, and molecular modeling studies of N-((4-acetyl phenyl) carbamothioyl) pivalamide as the multitarget-directed ligand - Saeed_2022_Front.Chem_10_992701 |
Author(s) : Saeed A , Ejaz SA , Khalid A , Channar PA , Aziz M , Wani TA , Zargar S , Hassan S , Ismail H , Khalid D , Hashmi MZ , Hokelek T , Aborode AT |
Ref : Front Chem , 10 :992701 , 2022 |
Abstract : |
PubMedSearch : Saeed_2022_Front.Chem_10_992701 |
PubMedID: 36226116 |
Title : Synthesis, bioactivity and binding energy calculations of novel 3-ethoxysalicylaldehyde based thiosemicarbazone derivatives - Ishaq_2020_Bioorg.Chem_100_103924 |
Author(s) : Ishaq M , Taslimi P , Shafiq Z , Khan S , Ekhteiari Salmas R , Zangeneh MM , Saeed A , Zangeneh A , Sadeghian N , Asari A , Mohamad H |
Ref : Bioorg Chem , 100 :103924 , 2020 |
Abstract : |
PubMedSearch : Ishaq_2020_Bioorg.Chem_100_103924 |
PubMedID: 32442818 |
Title : Drug-1,3,4-Thiadiazole Conjugates as Novel Mixed-Type Inhibitors of Acetylcholinesterase: Synthesis, Molecular Docking, Pharmacokinetics, and ADMET Evaluation - Ujan_2019_Molecules_24_ |
Author(s) : Ujan R , Saeed A , Channar PA , Larik FA , Abbas Q , Alajmi MF , El-Seedi HR , Rind MA , Hassan M , Raza H , Seo SY |
Ref : Molecules , 24 : , 2019 |
Abstract : |
PubMedSearch : Ujan_2019_Molecules_24_ |
PubMedID: 30823444 |
Title : Investigation of potent inhibitors of cholinesterase based on thiourea and pyrazoline derivatives: Synthesis, inhibition assay and molecular modeling studies - Mumtaz_2019_Bioorg.Chem_90_103036 |
Author(s) : Mumtaz A , Majeed A , Zaib S , Ur Rahman S , Hameed S , Saeed A , Rafique H , Mughal E , Maalik A , Hussain I , Iqbal J |
Ref : Bioorg Chem , 90 :103036 , 2019 |
Abstract : |
PubMedSearch : Mumtaz_2019_Bioorg.Chem_90_103036 |
PubMedID: 31271943 |
Title : Synthesis, molecular modelling and biological evaluation of tetrasubstituted thiazoles towards cholinesterase enzymes and cytotoxicity studies - Mumtaz_2018_Bioorg.Chem_78_141 |
Author(s) : Mumtaz A , Shoaib M , Zaib S , Shah MS , Bhatti HA , Saeed A , Hussain I , Iqbal J |
Ref : Bioorg Chem , 78 :141 , 2018 |
Abstract : |
PubMedSearch : Mumtaz_2018_Bioorg.Chem_78_141 |
PubMedID: 29567428 |
Title : One-pot four-component synthesis of thiazolidin-2-imines using Cu(I)\/Zn(II) dual catalysis: A new class of acetylcholinesterase inhibitors - Shehzadi_2018_Bioorg.Chem_84_518 |
Author(s) : Shehzadi SA , Khan I , Saeed A , Larik FA , Channar PA , Hassan M , Raza H , Abbas Q , Seo SY |
Ref : Bioorg Chem , 84 :518 , 2018 |
Abstract : |
PubMedSearch : Shehzadi_2018_Bioorg.Chem_84_518 |
PubMedID: 30610971 |
Title : New cholinesterase inhibitors for Alzheimer's disease: Structure activity relationship, kinetics and molecular docking studies of 1-butanoyl-3-arylthiourea derivatives - Larik_2018_Int.J.Biol.Macromol_116_144 |
Author(s) : Larik FA , Shah MS , Saeed A , Shah HS , Channar PA , Bolte M , Iqbal J |
Ref : Int J Biol Macromol , 116 :144 , 2018 |
Abstract : |
PubMedSearch : Larik_2018_Int.J.Biol.Macromol_116_144 |
PubMedID: 29729344 |
Title : Synthesis, Characterization and Cholinesterase Inhibition Studies of New Arylidene Aminothiazolylethanone Derivatives - Channar_2017_Med.Chem_13_648 |
Author(s) : Channar PA , Shah MS , Saeed A , Khan SU , Larik FA , Shabir G , Iqbal J |
Ref : Med Chem , 13 :648 , 2017 |
Abstract : |
PubMedSearch : Channar_2017_Med.Chem_13_648 |
PubMedID: 28266279 |
Title : Design and synthesis of 2,6-di(substituted phenyl)thiazolo[3,2-b]-1,2,4-triazoles as alpha-glucosidase and alpha-amylase inhibitors, co-relative Pharmacokinetics and 3D QSAR and risk analysis - Channar_2017_Biomed.Pharmacother_94_499 |
Author(s) : Channar PA , Saeed A , Larik FA , Rashid S , Iqbal Q , Rozi M , Younis S , Mahar J |
Ref : Biomed Pharmacother , 94 :499 , 2017 |
Abstract : |
PubMedSearch : Channar_2017_Biomed.Pharmacother_94_499 |
PubMedID: 28780468 |
Title : Biological Evaluation of Azomethine-dihydroquinazolinone Conjugates as Cancer and Cholinesterase Inhibitors - Iqbal_2016_Med.Chem_12_74 |
Author(s) : Iqbal J , Saeed A , Shah SJ , Al-Rashida M , Mahmood SU |
Ref : Med Chem , 12 :74 , 2016 |
Abstract : |
PubMedSearch : Iqbal_2016_Med.Chem_12_74 |
PubMedID: 26152145 |
Title : Synthesis, cholinesterase inhibition and molecular modelling studies of coumarin linked thiourea derivatives - Saeed_2015_Bioorg.Chem_63_58 |
Author(s) : Saeed A , Zaib S , Ashraf S , Iftikhar J , Muddassar M , Zhang KY , Iqbal J |
Ref : Bioorg Chem , 63 :58 , 2015 |
Abstract : |
PubMedSearch : Saeed_2015_Bioorg.Chem_63_58 |
PubMedID: 26440714 |
Title : Synthesis of brominated 2-phenitidine derivatives as valuable inhibitors of cholinesterases for the treatment of Alzheimer's disease - Abbasi_2014_Iran.J.Pharm.Res_13_87 |
Author(s) : Abbasi MA , Saeed A , Aziz Ur R , Mohmmed Khan K , Ashraf M , Ejaz SA |
Ref : Iran J Pharm Res , 13 :87 , 2014 |
Abstract : |
PubMedSearch : Abbasi_2014_Iran.J.Pharm.Res_13_87 |
PubMedID: 24734059 |
Title : Synthesis, cytotoxicity and molecular modelling studies of new phenylcinnamide derivatives as potent inhibitors of cholinesterases - Saeed_2014_Eur.J.Med.Chem_78C_43 |
Author(s) : Saeed A , Mahesar PA , Zaib S , Khan MS , Matin A , Shahid M , Iqbal J |
Ref : Eur Journal of Medicinal Chemistry , 78C :43 , 2014 |
Abstract : |
PubMedSearch : Saeed_2014_Eur.J.Med.Chem_78C_43 |
PubMedID: 24675179 |
Title : Synthesis and Biological Evaluation of 3-thiazolocoumarinyl Schiff-base Derivatives as Cholinesterase Inhibitors - Raza_2012_Chem.Biol.Drug.Des_80_605 |
Author(s) : Raza R , Saeed A , Arif M , Mahmood S , Muddassar M , Raza A , Iqbal J |
Ref : Chemical Biology Drug Des , 80 :605 , 2012 |
Abstract : |
PubMedSearch : Raza_2012_Chem.Biol.Drug.Des_80_605 |
PubMedID: 22726458 |
Title : Pharmacological Evaluation and Docking Studies of 3-Thiadiazolyl- and Thioxo-1,2,4-triazolylcoumarin Derivatives as Cholinesterase Inhibitors - Raza_2012_ISRN.Pharmacol_2012_707932 |
Author(s) : Raza A , Saeed A , Ibrar A , Muddassar M , Khan AA , Iqbal J |
Ref : ISRN Pharmacol , 2012 :707932 , 2012 |
Abstract : |
PubMedSearch : Raza_2012_ISRN.Pharmacol_2012_707932 |
PubMedID: 22966467 |