Title : Discovery and preclinical profile of teneligliptin (3-[(2S,4S)-4-[4-(3-methyl-1-phenyl-1H-pyrazol-5-yl)piperazin-1-yl]pyrrolidin-2-y lcarbonyl]thiazolidine): a highly potent, selective, long-lasting and orally active dipeptidyl peptidase IV inhibitor for the treatment of type 2 diabetes - Yoshida_2012_Bioorg.Med.Chem_20_5705 |
Author(s) : Yoshida T , Akahoshi F , Sakashita H , Kitajima H , Nakamura M , Sonda S , Takeuchi M , Tanaka Y , Ueda N , Sekiguchi S , Ishige T , Shima K , Nabeno M , Abe Y , Anabuki J , Soejima A , Yoshida K , Takashina Y , Ishii S , Kiuchi S , Fukuda S , Tsutsumiuchi R , Kosaka K , Murozono T , Nakamaru Y , Utsumi H , Masutomi N , Kishida H , Miyaguchi I , Hayashi Y |
Ref : Bioorganic & Medicinal Chemistry , 20 :5705 , 2012 |
Abstract : |
PubMedSearch : Yoshida_2012_Bioorg.Med.Chem_20_5705 |
PubMedID: 22959556 |
Gene_locus related to this paper: human-DPP4 |
Title : Fused bicyclic heteroarylpiperazine-substituted L-prolylthiazolidines as highly potent DPP-4 inhibitors lacking the electrophilic nitrile group - Yoshida_2012_Bioorg.Med.Chem_20_5033 |
Author(s) : Yoshida T , Akahoshi F , Sakashita H , Sonda S , Takeuchi M , Tanaka Y , Nabeno M , Kishida H , Miyaguchi I , Hayashi Y |
Ref : Bioorganic & Medicinal Chemistry , 20 :5033 , 2012 |
Abstract : |
PubMedSearch : Yoshida_2012_Bioorg.Med.Chem_20_5033 |
PubMedID: 22824762 |
Gene_locus related to this paper: human-DPP4 |
Title : Sequence completion, identification and definition of the fengycin operon in Bacillus subtilis 168 - Tosato_1997_Microbiology_143 ( Pt 11)_3443 |
Author(s) : Tosato V , Albertini AM , Zotti M , Sonda S , Bruschi CV |
Ref : Microbiology , 143 ( Pt 11) :3443 , 1997 |
Abstract : |
PubMedSearch : Tosato_1997_Microbiology_143 ( Pt 11)_3443 |
PubMedID: 9387222 |
Gene_locus related to this paper: bacsu-PPSE |