| Title : Novel thiazolopyridine derivatives of diflapolin as dual sEH\/FLAP inhibitors with improved solubility - Schoenthaler_2023_Bioorg.Chem_139_106685 |
| Author(s) : Schoenthaler M , Waltl L , Hasenoehrl T , Seher D , Lutz A , Aulinger L , Temml V , Konig S , Siller A , Braun DE , Garscha U , Werz O , Schuster D , Schennach H , Koeberle A , Matuszczak B |
| Ref : Bioorg Chem , 139 :106685 , 2023 |
| Abstract : |
| PubMedSearch : Schoenthaler_2023_Bioorg.Chem_139_106685 |
| PubMedID: 37418786 |
| Title : Synthesis and structure-activity relationships for some novel diflapolin derivatives with benzimidazole subunit - Vieider_2022_J.Enzyme.Inhib.Med.Chem_37_1752 |
| Author(s) : Vieider L , Zoeller E , Romp E , Schoenthaler M , Hernandez-Olmos V , Temml V , Hasenoehrl T , Schuster D , Werz O , Garscha U , Matuszczak B |
| Ref : J Enzyme Inhib Med Chem , 37 :1752 , 2022 |
| Abstract : |
| PubMedSearch : Vieider_2022_J.Enzyme.Inhib.Med.Chem_37_1752 |
| PubMedID: 36124840 |
| Title : N-methylated diazabicyclo[3.2.2]nonane substituted triterpenoic acids are excellent, hyperbolic and selective inhibitors for butyrylcholinesterase - Heise_2021_Eur.J.Med.Chem_227_113947 |
| Author(s) : Heise N , Friedrich S , Temml V , Schuster D , Siewert B , Csuk R |
| Ref : Eur Journal of Medicinal Chemistry , 227 :113947 , 2021 |
| Abstract : |
| PubMedSearch : Heise_2021_Eur.J.Med.Chem_227_113947 |
| PubMedID: 34731766 |
| Title : Synthesis, Biological Evaluation and Structure-Activity Relationships of Diflapolin Analogues as Dual sEH\/FLAP Inhibitors - Vieider_2019_ACS.Med.Chem.Lett_10_62 |
| Author(s) : Vieider L , Romp E , Temml V , Fischer J , Kretzer C , Schoenthaler M , Taha A , Hernandez-Olmos V , Sturm S , Schuster D , Werz O , Garscha U , Matuszczak B |
| Ref : ACS Med Chem Lett , 10 :62 , 2019 |
| Abstract : |
| PubMedSearch : Vieider_2019_ACS.Med.Chem.Lett_10_62 |
| PubMedID: 30655948 |
| Title : Discovery of the first dual inhibitor of the 5-lipoxygenase-activating protein and soluble epoxide hydrolase using pharmacophore-based virtual screening - Temml_2017_Sci.Rep_7_42751 |
| Author(s) : Temml V , Garscha U , Romp E , Schubert G , Gerstmeier J , Kutil Z , Matuszczak B , Waltenberger B , Stuppner H , Werz O , Schuster D |
| Ref : Sci Rep , 7 :42751 , 2017 |
| Abstract : |
| PubMedSearch : Temml_2017_Sci.Rep_7_42751 |
| PubMedID: 28218273 |
| Title : Pharmacological profile and efficiency in vivo of diflapolin, the first dual inhibitor of 5-lipoxygenase-activating protein and soluble epoxide hydrolase - Garscha_2017_Sci.Rep_7_9398 |
| Author(s) : Garscha U , Romp E , Pace S , Rossi A , Temml V , Schuster D , Konig S , Gerstmeier J , Liening S , Werner M , Atze H , Wittmann S , Weinigel C , Rummler S , Scriba GK , Sautebin L , Werz O |
| Ref : Sci Rep , 7 :9398 , 2017 |
| Abstract : |
| PubMedSearch : Garscha_2017_Sci.Rep_7_9398 |
| PubMedID: 28839250 |