| Title : Synthesis and structure-activity relationships for some novel diflapolin derivatives with benzimidazole subunit - Vieider_2022_J.Enzyme.Inhib.Med.Chem_37_1752 |
| Author(s) : Vieider L , Zoeller E , Romp E , Schoenthaler M , Hernandez-Olmos V , Temml V , Hasenoehrl T , Schuster D , Werz O , Garscha U , Matuszczak B |
| Ref : J Enzyme Inhib Med Chem , 37 :1752 , 2022 |
| Abstract : Vieider_2022_J.Enzyme.Inhib.Med.Chem_37_1752 |
| ESTHER : Vieider_2022_J.Enzyme.Inhib.Med.Chem_37_1752 |
| PubMedSearch : Vieider_2022_J.Enzyme.Inhib.Med.Chem_37_1752 |
| PubMedID: 36124840 |
| Title : Combined Cardioprotective and Adipocyte Browning Effects Promoted by the Eutomer of Dual sEH\/PPARgamma Modulator - Hartmann_2021_J.Med.Chem_64_2815 |
| Author(s) : Hartmann M , Bibli SI , Tews D , Ni X , Kircher T , Kramer JS , Kilu W , Heering J , Hernandez-Olmos V , Weizel L , Scriba GKE , Krait S , Knapp S , Chaikuad A , Merk D , Fleming I , Fischer-Posovszky P , Proschak E |
| Ref : Journal of Medicinal Chemistry , 64 :2815 , 2021 |
| Abstract : Hartmann_2021_J.Med.Chem_64_2815 |
| ESTHER : Hartmann_2021_J.Med.Chem_64_2815 |
| PubMedSearch : Hartmann_2021_J.Med.Chem_64_2815 |
| PubMedID: 33620196 |
| Title : Structure-Based Design of Dual Partial Peroxisome Proliferator-Activated Receptor gamma Agonists\/Soluble Epoxide Hydrolase Inhibitors - Lillich_2021_J.Med.Chem_64_17259 |
| Author(s) : Lillich FF , Willems S , Ni X , Kilu W , Borkowsky C , Brodsky M , Kramer JS , Brunst S , Hernandez-Olmos V , Heering J , Schierle S , Kestner RI , Mayser FM , Helmstadter M , Gobel T , Weizel L , Namgaladze D , Kaiser A , Steinhilber D , Pfeilschifter W , Kahnt AS , Proschak A , Chaikuad A , Knapp S , Merk D , Proschak E |
| Ref : Journal of Medicinal Chemistry , : , 2021 |
| Abstract : Lillich_2021_J.Med.Chem_64_17259 |
| ESTHER : Lillich_2021_J.Med.Chem_64_17259 |
| PubMedSearch : Lillich_2021_J.Med.Chem_64_17259 |
| PubMedID: 34818007 |
| Gene_locus related to this paper: human-EPHX2 |
| Title : Discovery of the First in Vivo Active Inhibitors of the Soluble Epoxide Hydrolase Phosphatase Domain - Kramer_2019_J.Med.Chem_62_8443 |
| Author(s) : Kramer JS , Woltersdorf S , Duflot T , Hiesinger K , Lillich FF , Knoll F , Wittmann SK , Klingler FM , Brunst S , Chaikuad A , Morisseau C , Hammock BD , Buccellati C , Sala A , Rovati GE , Leuillier M , Fraineau S , Rondeaux J , Hernandez-Olmos V , Heering J , Merk D , Pogoryelov D , Steinhilber D , Knapp S , Bellien J , Proschak E |
| Ref : Journal of Medicinal Chemistry , 62 :8443 , 2019 |
| Abstract : Kramer_2019_J.Med.Chem_62_8443 |
| ESTHER : Kramer_2019_J.Med.Chem_62_8443 |
| PubMedSearch : Kramer_2019_J.Med.Chem_62_8443 |
| PubMedID: 31436984 |
| Title : Synthesis, Biological Evaluation and Structure-Activity Relationships of Diflapolin Analogues as Dual sEH\/FLAP Inhibitors - Vieider_2019_ACS.Med.Chem.Lett_10_62 |
| Author(s) : Vieider L , Romp E , Temml V , Fischer J , Kretzer C , Schoenthaler M , Taha A , Hernandez-Olmos V , Sturm S , Schuster D , Werz O , Garscha U , Matuszczak B |
| Ref : ACS Med Chem Lett , 10 :62 , 2019 |
| Abstract : Vieider_2019_ACS.Med.Chem.Lett_10_62 |
| ESTHER : Vieider_2019_ACS.Med.Chem.Lett_10_62 |
| PubMedSearch : Vieider_2019_ACS.Med.Chem.Lett_10_62 |
| PubMedID: 30655948 |
| Title : Discovery of polar spirocyclic orally bioavailable urea inhibitors of soluble epoxide hydrolase - Lukin_2018_Bioorg.Chem_80_655 |
| Author(s) : Lukin A , Kramer J , Hartmann M , Weizel L , Hernandez-Olmos V , Falahati K , Burghardt I , Kalinchenkova N , Bagnyukova D , Zhurilo N , Rautio J , Forsberg M , Ihalainen J , Auriola S , Leppanen J , Konstantinov I , Pogoryelov D , Proschak E , Dar'in D , Krasavin M |
| Ref : Bioorg Chem , 80 :655 , 2018 |
| Abstract : Lukin_2018_Bioorg.Chem_80_655 |
| ESTHER : Lukin_2018_Bioorg.Chem_80_655 |
| PubMedSearch : Lukin_2018_Bioorg.Chem_80_655 |
| PubMedID: 30059891 |
| Gene_locus related to this paper: human-EPHX2 |