Title : A novel approach for modeling in vivo enzyme turnover in the presence of a suicide inhibitor drug: A proof-of-concept brain PET study on MAG lipase - Volpi_2025_J.Cereb.Blood.Flow.Metab__271678x251329254 |
Author(s) : Volpi T , Holden D , Gallezot JD , Nabulsi N , Lim K , Labaree D , Gao H , Kapinos M , Keliher EJ , Fonseca KR , Trapa P , Varrone A , Halldin C , Maresca KP , Huang Y , Carson RE |
Ref : Journal of Cerebral Blood Flow & Metabolism , :271678x251329254 , 2025 |
Abstract : |
PubMedSearch : Volpi_2025_J.Cereb.Blood.Flow.Metab__271678x251329254 |
PubMedID: 40370302 |
Title : Identification and Development of an Irreversible Monoacylglycerol Lipase (MAGL) Positron Emission Tomography (PET) Radioligand with High Specificity - Zhang_2019_J.Med.Chem_62_8532 |
Author(s) : Zhang L , Butler CR , Maresca KP , Takano A , Nag S , Jia Z , Arakawa R , Piro JR , Samad T , Smith DL , Nason DM , O'Neil S , McAllister L , Schildknegt K , Trapa P , McCarthy TJ , Villalobos A , Halldin C |
Ref : Journal of Medicinal Chemistry , 62 :8532 , 2019 |
Abstract : |
PubMedSearch : Zhang_2019_J.Med.Chem_62_8532 |
PubMedID: 31483137 |