| Title : A novel approach for modeling in vivo enzyme turnover in the presence of a suicide inhibitor drug: A proof-of-concept brain PET study on MAG lipase - Volpi_2025_J.Cereb.Blood.Flow.Metab__271678x251329254 |
| Author(s) : Volpi T , Holden D , Gallezot JD , Nabulsi N , Lim K , Labaree D , Gao H , Kapinos M , Keliher EJ , Fonseca KR , Trapa P , Varrone A , Halldin C , Maresca KP , Huang Y , Carson RE |
| Ref : Journal of Cerebral Blood Flow & Metabolism , :271678x251329254 , 2025 |
| Abstract : |
| PubMedSearch : Volpi_2025_J.Cereb.Blood.Flow.Metab__271678x251329254 |
| PubMedID: 40370302 |
| Title : Identification and Development of an Irreversible Monoacylglycerol Lipase (MAGL) Positron Emission Tomography (PET) Radioligand with High Specificity - Zhang_2019_J.Med.Chem_62_8532 |
| Author(s) : Zhang L , Butler CR , Maresca KP , Takano A , Nag S , Jia Z , Arakawa R , Piro JR , Samad T , Smith DL , Nason DM , O'Neil S , McAllister L , Schildknegt K , Trapa P , McCarthy TJ , Villalobos A , Halldin C |
| Ref : Journal of Medicinal Chemistry , 62 :8532 , 2019 |
| Abstract : |
| PubMedSearch : Zhang_2019_J.Med.Chem_62_8532 |
| PubMedID: 31483137 |
| Title : Liver-Targeted Small-Molecule Inhibitors of Proprotein Convertase Subtilisin\/Kexin Type 9 Synthesis - McClure_2017_Angew.Chem.Int.Ed.Engl_56_16218 |
| Author(s) : McClure KF , Piotrowski DW , Petersen D , Wei L , Xiao J , Londregan AT , Kamlet AS , Dechert-Schmitt AM , Raymer B , Ruggeri RB , Canterbury D , Limberakis C , Liras S , DaSilva-Jardine P , Dullea RG , Loria PM , Reidich B , Salatto CT , Eng H , Kimoto E , Atkinson K , King-Ahmad A , Scott D , Beaumont K , Chabot JR , Bolt MW , Maresca K , Dahl K , Arakawa R , Takano A , Halldin C |
| Ref : Angew Chem Int Ed Engl , 56 :16218 , 2017 |
| Abstract : |
| PubMedSearch : McClure_2017_Angew.Chem.Int.Ed.Engl_56_16218 |
| PubMedID: 29073340 |
| Title : PET study of the M1-agonists [11C]xanomeline and [11C]butylthio-TZTP in monkey and man - Farde_1996_Dementia_7_187 |
| Author(s) : Farde L , Suhara T , Halldin C , Nyback H , Nakashima Y , Swahn CG , Karlsson P , Ginovart N , Bymaster FP , Shannon HE , Foged C , Suzdak PD , Sauerberg P |
| Ref : Dementia , 7 :187 , 1996 |
| Abstract : |
| PubMedSearch : Farde_1996_Dementia_7_187 |
| PubMedID: 8835881 |