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| Title : Design, synthesis and preliminary biological evaluation of rivastigmine-INDY hybrids as multitarget ligands against Alzheimer's disease by targeting butyrylcholinesterase and DYRK1A\/CLK1 kinases - Tintas_2024_RSC.Med.Chem_15_963 |
| Author(s) : Tintas ML , Peauger L , Barre A , Papamical C , Besson T , Sopkova-de Oliveira Santos J , Gembus V , Levacher V |
| Ref : RSC Med Chem , 15 :963 , 2024 |
| Abstract : Tintas_2024_RSC.Med.Chem_15_963 |
| ESTHER : Tintas_2024_RSC.Med.Chem_15_963 |
| PubMedSearch : Tintas_2024_RSC.Med.Chem_15_963 |
| PubMedID: 38516603 |
| Title : Design, Synthesis, and In Vitro Biological Activities of a Bio-Oxidizable Prodrug to Deliver Both ChEs and DYRK1A Inhibitors for AD Therapy - Barre_2019_Molecules_24_ |
| Author(s) : Barre A , Azzouz R , Gembus V , Papamicael C , Levacher V |
| Ref : Molecules , 24 : , 2019 |
| Abstract : Barre_2019_Molecules_24_ |
| ESTHER : Barre_2019_Molecules_24_ |
| PubMedSearch : Barre_2019_Molecules_24_ |
| PubMedID: 30939771 |
| Title : Rational design of carbamate-based dual binding site and central AChE inhibitors by a 'biooxidisable' prodrug approach: Synthesis, invitro evaluation and docking studies - Tintas_2018_Eur.J.Med.Chem_155_171 |
| Author(s) : Tintas ML , Gembus V , Alix F , Barre A , Coadou G , Truong L , Sebban M , Papamical C , Oulyadi H , Levacher V |
| Ref : Eur Journal of Medicinal Chemistry , 155 :171 , 2018 |
| Abstract : Tintas_2018_Eur.J.Med.Chem_155_171 |
| ESTHER : Tintas_2018_Eur.J.Med.Chem_155_171 |
| PubMedSearch : Tintas_2018_Eur.J.Med.Chem_155_171 |
| PubMedID: 29886321 |
| Title : Donepezil-Based Central Acetylcholinesterase Inhibitors by Means of a Bio-Oxidizable Prodrug Strategy: Design, Synthesis, and in Vitro Biological Evaluation - Peauger_2017_J.Med.Chem_60_5909 |
| Author(s) : Peauger L , Azzouz R , Gembus V , Tintas ML , Sopkova-de Oliveira Santos J , Bohn P , Papamicael C , Levacher V |
| Ref : Journal of Medicinal Chemistry , 60 :5909 , 2017 |
| Abstract : Peauger_2017_J.Med.Chem_60_5909 |
| ESTHER : Peauger_2017_J.Med.Chem_60_5909 |
| PubMedSearch : Peauger_2017_J.Med.Chem_60_5909 |
| PubMedID: 28613859 |
| Title : Dihydroquinoline Carbamate Derivatives as Bio-oxidizable Prodrugs for Brain Delivery of Acetylcholinesterase Inhibitors: [(11)C] Radiosynthesis and Biological Evaluation - Bohn_2015_ACS.Chem.Neurosci_6_737 |
| Author(s) : Bohn P , Gourand F , Papamicael C , Ibazizene M , Dhilly M , Gembus V , Alix F , Tintas ML , Marsais F , Barre L , Levacher V |
| Ref : ACS Chem Neurosci , 6 :737 , 2015 |
| Abstract : Bohn_2015_ACS.Chem.Neurosci_6_737 |
| ESTHER : Bohn_2015_ACS.Chem.Neurosci_6_737 |
| PubMedSearch : Bohn_2015_ACS.Chem.Neurosci_6_737 |
| PubMedID: 25695305 |
| Title : New developments in redox chemical delivery systems by means of 1,4-dihydroquinoline-based targetor: Application to galantamine delivery to the brain - Tintas_2014_Eur.J.Med.Chem_81C_218 |
| Author(s) : Tintas ML , Foucout L , Petit S , Oudeyer S , Gourand F , Barre L , Papamicael C , Levacher V |
| Ref : Eur Journal of Medicinal Chemistry , 81C :218 , 2014 |
| Abstract : Tintas_2014_Eur.J.Med.Chem_81C_218 |
| ESTHER : Tintas_2014_Eur.J.Med.Chem_81C_218 |
| PubMedSearch : Tintas_2014_Eur.J.Med.Chem_81C_218 |
| PubMedID: 24852273 |
| Title : Rational design of central selective acetylcholinesterase inhibitors by means of a bio-oxidisable prodrug strategy - Bohn_2009_Org.Biomol.Chem_7_2612 |
| Author(s) : Bohn P , Le Fur N , Hagues G , Costentin J , Torquet N , Papamicael C , Marsais F , Levacher V |
| Ref : Org Biomol Chem , 7 :2612 , 2009 |
| Abstract : Bohn_2009_Org.Biomol.Chem_7_2612 |
| ESTHER : Bohn_2009_Org.Biomol.Chem_7_2612 |
| PubMedSearch : Bohn_2009_Org.Biomol.Chem_7_2612 |
| PubMedID: 19503937 |