Name : Dipepdyl peptidase IV in complex with inhibitor PZF
Revelation date : 29-Jul-2008
Family : DPP4N_Peptidase_S9
Gene_locus : human-DPP4
PDB file : ESTHER: header of PDB entry RCSB: Full entry
Comment
Wright SW, Ammirati MJ, Andrews KM, Brodeur AM, Danley DE, Doran SD, Lillquist JS, Liu S, McClure LD, McPherson RK, Olson TV, Orena SJ, Parker JC, Rocke BN, Soeller WC, Soglia CB, Treadway JL, Vanvolkenburg MA, Zhao Z, Cox ED
Ligand :
Title : (3R,4S)-4-(2,4,5-Trifluorophenyl)-pyrrolidin-3-ylamine inhibitors of dipeptidyl peptidase IV: synthesis, in vitro, in vivo, and X-ray crystallographic characterization - Wright_2007_Bioorg.Med.Chem.Lett_17_5638 |
Author(s) : Wright SW , Ammirati MJ , Andrews KM , Brodeur AM , Danley DE , Doran SD , Lillquist JS , Liu S , McClure LD , McPherson RK , Olson TV , Orena SJ , Parker JC , Rocke BN , Soeller WC , Soglia CB , Treadway JL , VanVolkenburg MA , Zhao Z , Cox ED |
Ref : Bioorganic & Medicinal Chemistry Lett , 17 :5638 , 2007 |
Abstract : Wright_2007_Bioorg.Med.Chem.Lett_17_5638 |
ESTHER : Wright_2007_Bioorg.Med.Chem.Lett_17_5638 |
PubMedSearch : Wright_2007_Bioorg.Med.Chem.Lett_17_5638 |
PubMedID: 17822893 |
Gene_locus related to this paper: human-DPP4 |
PDB-Sum : 2QJR Previously Class, Architecture, Topology and Homologous superfamily - PDB-Sum server
FSSP : 2QJR Fold classification based on Structure-Structure alignment of Proteins - FSSP server
SCOP : 2QJR Structural Classification Of Protein - SCOP server
PROTEOPEDIA : 2QJR 3D, interactive encyclopedia of proteins - PROTEOPEDIA server