Name : Crystal structure of Dipeptidyl Peptidase IV in complex with a pyrimidinone inhibitor
Revelation date : 16-Feb-2010
Family : DPP4N_Peptidase_S9
Gene_locus : human-DPP4
PDB file : ESTHER: header of PDB entry RCSB: Full entry
Comment
Zhang, Zhiyuan, Wallace, Michael B., Feng, Jun, Stafford, Jeffrey A., Kaldor, Stephen W., Lihong, Shi, Skene, Robert J., Aertgeerts, Kathleen, Lee, Bumsup, Jennings, Andy, Xu, Rongda, Kassel, Daniel, Webb, David R., Gwaltney, Stephen L.
Ligand : Inhibitor Pyrimidinone-inhibitor3 Ligand in structure: Ligplot
Title : Design and synthesis of pyrimidinone and pyrimidinedione inhibitors of dipeptidyl peptidase IV - Zhang_2011_J.Med.Chem_54_510 |
Author(s) : Zhang Z , Wallace MB , Feng J , Stafford JA , Skene RJ , Shi L , Lee B , Aertgeerts K , Jennings A , Xu R , Kassel DB , Kaldor SW , Navre M , Webb DR , Gwaltney SL |
Ref : Journal of Medicinal Chemistry , 54 :510 , 2011 |
Abstract : |
PubMedSearch : Zhang_2011_J.Med.Chem_54_510 |
PubMedID: 21186796 |
Gene_locus related to this paper: human-DPP4 |
PDB-Sum : 3G0G Previously Class, Architecture, Topology and Homologous superfamily - PDB-Sum server
FSSP : 3G0G Fold classification based on Structure-Structure alignment of Proteins - FSSP server
SCOP : 3G0G Structural Classification Of Protein - SCOP server
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