Title : Poster: Profile of A-716096, a novel thiazolylidine positive allosteric modulator of the alpha7 nicotinic acetylcholine receptor - |
Author(s) : Donnelly-Roberts D , Malysz J , Faghih R , Gronlien H , Haakerud M , Thorin-Hagne K , Ween H , Gopalakrishnan SM , Hu M , Li J , Anderson DJ , Kohlhaas KL , Namovic M , Radek R , Robb H , Briggs CA , Bitner RS , Bunnelle WH , Gopalakrishnan M |
Ref : Biochemical Pharmacology , 78 :912 , 2009 |
PubMedID: |
Title : Discovery of 4-(5-(4-chlorophenyl)-2-methyl-3-propionyl-1H-pyrrol-1-yl)benzenesulfonamide (A-867744) as a novel positive allosteric modulator of the alpha7 nicotinic acetylcholine receptor - Faghih_2009_J.Med.Chem_52_3377 |
Author(s) : Faghih R , Gopalakrishnan SM , Gronlien JH , Malysz J , Briggs CA , Wetterstrand C , Ween H , Curtis MP , Sarris KA , Gfesser GA , El-Kouhen R , Robb HM , Radek RJ , Marsh KC , Bunnelle WH , Gopalakrishnan M |
Ref : Journal of Medicinal Chemistry , 52 :3377 , 2009 |
Abstract : |
PubMedSearch : Faghih_2009_J.Med.Chem_52_3377 |
PubMedID: 19419141 |
Title : In vitro pharmacological characterization of a novel allosteric modulator of alpha 7 neuronal acetylcholine receptor, 4-(5-(4-chlorophenyl)-2-methyl-3-propionyl-1H-pyrrol-1-yl)benzenesulfonamide (A-867744), exhibiting unique pharmacological profile - Malysz_2009_J.Pharmacol.Exp.Ther_330_257 |
Author(s) : Malysz J , Gronlien JH , Anderson DJ , Hakerud M , Thorin-Hagene K , Ween H , Wetterstrand C , Briggs CA , Faghih R , Bunnelle WH , Gopalakrishnan M |
Ref : Journal of Pharmacology & Experimental Therapeutics , 330 :257 , 2009 |
Abstract : |
PubMedSearch : Malysz_2009_J.Pharmacol.Exp.Ther_330_257 |
PubMedID: 19389923 |
Title : Allosteric modulators of the alpha7 nicotinic acetylcholine receptor - |
Author(s) : Faghih R , Gopalakrishnan M , Briggs CA |
Ref : Journal of Medicinal Chemistry , 51 :701 , 2008 |
PubMedID: 18198823 |
Title : Advances in the discovery of novel positive allosteric modulators of the alpha7 nicotinic acetylcholine receptor - Faghih_2007_Recent.Pat.CNS.Drug.Discov_2_99 |
Author(s) : Faghih R , Gfesser GA , Gopalakrishnan M |
Ref : Recent Pat CNS Drug Discov , 2 :99 , 2007 |
Abstract : |
PubMedSearch : Faghih_2007_Recent.Pat.CNS.Drug.Discov_2_99 |
PubMedID: 18221220 |