Title : Synthesis and SAR of 4-aminocyclopentapyrrolidines as N-type Ca(2)(+) channel blockers with analgesic activity - Beebe_2012_Bioorg.Med.Chem_20_4128 |
Author(s) : Beebe X , Darczak D , Henry RF , Vortherms T , Janis R , Namovic M , Donnelly-Roberts D , Kage KL , Surowy C , Milicic I , Niforatos W , Swensen A , Marsh KC , Wetter JM , Franklin P , Baker S , Zhong C , Simler G , Gomez E , Boyce-Rustay JM , Zhu CZ , Stewart AO , Jarvis MF , Scott VE |
Ref : Bioorganic & Medicinal Chemistry , 20 :4128 , 2012 |
Abstract : |
PubMedSearch : Beebe_2012_Bioorg.Med.Chem_20_4128 |
PubMedID: 22626552 |
Title : Poster: A-582941, a pro-cognitive alpha7 nAChR agonist, differentially modulates mitochondrial membrane potential - |
Author(s) : Namovic M , Hu M , Abraham V , Towne D , Lee C-H , Gopalakrishnan M , Esbenshade T , Donnelly-Roberts D |
Ref : Biochemical Pharmacology , 82 :1027 , 2011 |
PubMedID: |
Title : The antihyperalgesic activity of a selective P2X7 receptor antagonist, A-839977, is lost in IL-1alphabeta knockout mice - Honore_2009_Behav.Brain.Res_204_77 |
Author(s) : Honore P , Donnelly-Roberts D , Namovic M , Zhong C , Wade C , Chandran P , Zhu C , Carroll W , Perez-Medrano A , Iwakura Y , Jarvis MF |
Ref : Behavioural Brain Research , 204 :77 , 2009 |
Abstract : |
PubMedSearch : Honore_2009_Behav.Brain.Res_204_77 |
PubMedID: 19464323 |
Title : Poster: Radioligand binding characterization of [3H]-A-998679: A novel positive allosteric modulator of alpha4\/beta2 nAChRs - |
Author(s) : Anderson DJ , Vaidyanathan S , Namovic M , Donnelly-Roberts D , Lee L , Gopalakrishnan M |
Ref : Biochemical Pharmacology , 78 :903 , 2009 |
PubMedID: |
Title : Poster: Profile of A-716096, a novel thiazolylidine positive allosteric modulator of the alpha7 nicotinic acetylcholine receptor - |
Author(s) : Donnelly-Roberts D , Malysz J , Faghih R , Gronlien H , Haakerud M , Thorin-Hagne K , Ween H , Gopalakrishnan SM , Hu M , Li J , Anderson DJ , Kohlhaas KL , Namovic M , Radek R , Robb H , Briggs CA , Bitner RS , Bunnelle WH , Gopalakrishnan M |
Ref : Biochemical Pharmacology , 78 :912 , 2009 |
PubMedID: |
Title : Synthesis and activity of N-cyanoguanidine-piperazine P2X7 antagonists - Betschmann_2008_Bioorg.Med.Chem.Lett_18_3848 |
Author(s) : Betschmann P , Bettencourt B , Donnelly-Roberts D , Friedman M , George J , Hirst G , Josephsohn N , Konopacki D , Li B , Maull J , Morytko MJ , Moore NS , Namovic M , Rafferty P , Salmeron-Garcia JA , Tarcsa E , Wang L , Woller K |
Ref : Bioorganic & Medicinal Chemistry Lett , 18 :3848 , 2008 |
Abstract : |
PubMedSearch : Betschmann_2008_Bioorg.Med.Chem.Lett_18_3848 |
PubMedID: 18595695 |
Title : Reduced nicotinic receptor-mediated antinociception following in vivo antisense knock-down in rat - Bitner_2000_Brain.Res_871_66 |
Author(s) : Bitner RS , Nikkel AL , Curzon P , Donnelly-Roberts D , Puttfarcken PS , Namovic M , Jacobs IC , Meyer MD , Decker MW |
Ref : Brain Research , 871 :66 , 2000 |
Abstract : |
PubMedSearch : Bitner_2000_Brain.Res_871_66 |
PubMedID: 10882784 |