Title : First demonstration of a functional role for central nervous system betaine\/{gamma}-aminobutyric acid transporter (mGAT2) based on synergistic anticonvulsant action among inhibitors of mGAT1 and mGAT2 - White_2005_J.Pharmacol.Exp.Ther_312_866 |
Author(s) : White HS , Watson WP , Hansen SL , Slough S , Perregaard J , Sarup A , Bolvig T , Petersen G , Larsson OM , Clausen RP , Frolund B , Falch E , Krogsgaard-Larsen P , Schousboe A |
Ref : Journal of Pharmacology & Experimental Therapeutics , 312 :866 , 2005 |
Abstract : |
PubMedSearch : White_2005_J.Pharmacol.Exp.Ther_312_866 |
PubMedID: 15550575 |
Title : Carbamoylcholine homologs: synthesis and pharmacology at nicotinic acetylcholine receptors - Jensen_2004_Eur.J.Pharmacol_497_125 |
Author(s) : Jensen AA , Mikkelsen I , Frolund B , Frydenvang K , Brehm L , Jaroszewski JW , Brauner-Osborne H , Falch E , Krogsgaard-Larsen P |
Ref : European Journal of Pharmacology , 497 :125 , 2004 |
Abstract : |
PubMedSearch : Jensen_2004_Eur.J.Pharmacol_497_125 |
PubMedID: 15306197 |
Title : Carbamoylcholine homologs: novel and potent agonists at neuronal nicotinic acetylcholine receptors - Jensen_2003_Mol.Pharmacol_64_865 |
Author(s) : Jensen AA , Mikkelsen I , Frolund B , Brauner-Osborne H , Falch E , Krogsgaard-Larsen P |
Ref : Molecular Pharmacology , 64 :865 , 2003 |
Abstract : |
PubMedSearch : Jensen_2003_Mol.Pharmacol_64_865 |
PubMedID: 14500743 |
Title : Functional partial agonism at cloned human muscarinic acetylcholine receptors - Brauner-Osborne_1996_Eur.J.Pharmacol_313_145 |
Author(s) : Brauner-Osborne H , Ebert B , Brann MR , Falch E , Krogsgaard-Larsen P |
Ref : European Journal of Pharmacology , 313 :145 , 1996 |
Abstract : |
PubMedSearch : Brauner-Osborne_1996_Eur.J.Pharmacol_313_145 |
PubMedID: 8905341 |
Title : Analogues of carbacholine: synthesis and relationship between structure and affinity for muscarinic and nicotinic acetylcholine receptors - Sokilde_1996_Arch.Pharm.(Weinheim)_329_95 |
Author(s) : Sokilde B , Mikkelsen I , Stensbol TB , Andersen B , Ebdrup S , Krogsgaard-Larsen P , Falch E |
Ref : Arch Pharm (Weinheim) , 329 :95 , 1996 |
Abstract : |
PubMedSearch : Sokilde_1996_Arch.Pharm.(Weinheim)_329_95 |
PubMedID: 8851473 |
Title : Poster: Molecular pharmacology of O-alkyl-thao compounds using the five cloned muscarinic acetylcholine receptors - |
Author(s) : Jorgensen HB , Ebert B , Krogsgaard-Larsen P , Brann MR , Falch E |
Ref : Life Sciences , 56(11-12) :1007 , 1995 |
PubMedID: |
Title : Annulated heterocyclic bioisosteres of norarecoline. Synthesis and molecular pharmacology at five recombinant human muscarinic acetylcholine receptors - Brauner-Osborne_1995_J.Med.Chem_38_2188 |
Author(s) : Brauner-Osborne H , Ebert B , Brann MR , Falch E , Krogsgaard-Larsen P |
Ref : Journal of Medicinal Chemistry , 38 :2188 , 1995 |
Abstract : |
PubMedSearch : Brauner-Osborne_1995_J.Med.Chem_38_2188 |
PubMedID: 7783150 |
Title : Conformational aspects of the muscarinic receptor interactions of bicyclic isoxazole ester bioisosteres of arecoline - Lagersted_1993_Drug.Des.Discov_9_237 |
Author(s) : Lagersted A , Falch E , Ebert B , Krogsgaard-Larsen P |
Ref : Drug Des Discov , 9 :237 , 1993 |
Abstract : |
PubMedSearch : Lagersted_1993_Drug.Des.Discov_9_237 |
PubMedID: 8400005 |
Title : Poster: Heterocyclic muscarinic agonists as experimental tools and potentIal therapeutic agents - |
Author(s) : Byrholt Hansen A , Falch E , Jorgensen FS , Krogsgaard-Larsen P |
Ref : Trends in Pharmacological Sciences , Suppl :112 , 1989 |
PubMedID: |
Title : Heterocyclic muscarinic agonists. Synthesis and biological activity of some bicyclic sulfonium arecoline bioisosteres - Sauerberg_1988_J.Med.Chem_31_1312 |
Author(s) : Sauerberg P , Falch E , Meier E , Lembol HL , Krogsgaard-Larsen P |
Ref : Journal of Medicinal Chemistry , 31 :1312 , 1988 |
Abstract : |
PubMedSearch : Sauerberg_1988_J.Med.Chem_31_1312 |
PubMedID: 3385727 |
Title : Bioisosteres of arecoline as novel CNS-active muscarinic agonists - |
Author(s) : Krogsgaard-Larsen P , Falch E , Sauerberg P , Freedman SB , Lembol HL , Meier E |
Ref : Trends in Pharmacological Sciences , Suppl :69 , 1988 |
PubMedID: 3074541 |
Title : GABA uptake inhibitors. Synthesis and effects on audiogenic seizures of ester prodrugs of nipecotic acid, guvacine and cis-4-hydroxynipecotic acid - Falch_1987_Drug.Des.Deliv_2_9 |
Author(s) : Falch E , Meldrum BS , Krogsgaard-Larsen P |
Ref : Drug Des Deliv , 2 :9 , 1987 |
Abstract : |
PubMedSearch : Falch_1987_Drug.Des.Deliv_2_9 |
PubMedID: 3509345 |
Title : Pharmacological profile of a novel class of muscarinic acetylcholine receptor agonists - Sauerberg_1986_Eur.J.Pharmacol_130_125 |
Author(s) : Sauerberg P , Fjalland B , Larsen JJ , Bach-Lauritsen T , Falch E , Krogsgaard-Larsen P |
Ref : European Journal of Pharmacology , 130 :125 , 1986 |
Abstract : |
PubMedSearch : Sauerberg_1986_Eur.J.Pharmacol_130_125 |
PubMedID: 3780854 |
Title : A novel class of conformationally restricted heterocyclic muscarinic agonists - Sauerberg_1986_J.Med.Chem_29_1004 |
Author(s) : Sauerberg P , Larsen JJ , Falch E , Krogsgaard-Larsen P |
Ref : Journal of Medicinal Chemistry , 29 :1004 , 1986 |
Abstract : |
PubMedSearch : Sauerberg_1986_J.Med.Chem_29_1004 |
PubMedID: 3712371 |