Full name : Fasoli Francesca
First name : Francesca
Mail : CNR, Istituto di Neuroscienze, and Dipartimento di Biotecnologie Mediche e Medicina Traslazionale, Universit degli Studi di Milano, Via Vanvitelli 32, Milano, I-20129
Zip Code :
City :
Country : Italy
Email :
Phone :
Fax :
Website :
Directory :
Comment
                    
| Title : From pyrrolidinyl-benzodioxane to pyrrolidinyl-pyridodioxanes, or from unselective antagonism to selective partial agonism at alpha4beta2 nicotinic acetylcholine receptor - Bolchi_2017_Eur.J.Med.Chem_125_1132 | 
| Author(s) : Bolchi C , Bavo F , Gotti C , Fumagalli L , Fasoli F , Binda M , Mucchietto V , Sciaccaluga M , Plutino S , Fucile S , Pallavicini M | 
| Ref : Eur Journal of Medicinal Chemistry , 125 :1132 , 2017 | 
| Abstract : | 
| PubMedSearch : Bolchi_2017_Eur.J.Med.Chem_125_1132 | 
| PubMedID: 27810599 | 
| Title : Novel 5-substituted 3-hydroxyphenyl and 3-nitrophenyl ethers of S-prolinol as alpha4beta2-nicotinic acetylcholine receptor ligands - Bolchi_2016_Bioorg.Med.Chem.Lett_26_5613 | 
| Author(s) : Bolchi C , Bavo F , Fumagalli L , Gotti C , Fasoli F , Moretti M , Pallavicini M | 
| Ref : Bioorganic & Medicinal Chemistry Lett , 26 :5613 , 2016 | 
| Abstract : | 
| PubMedSearch : Bolchi_2016_Bioorg.Med.Chem.Lett_26_5613 | 
| PubMedID: 27818109 | 
| Title : In vivo chronic nicotine exposure differentially and reversibly affects upregulation and stoichiometry of alpha4beta2 nicotinic receptors in cortex and thalamus - Fasoli_2016_Neuropharmacol_108_324 | 
| Author(s) : Fasoli F , Moretti M , Zoli M , Pistillo F , Crespi A , Clementi F , Mc Clure-Begley T , Marks MJ , Gotti C | 
| Ref : Neuropharmacology , 108 :324 , 2016 | 
| Abstract : | 
| PubMedSearch : Fasoli_2016_Neuropharmacol_108_324 | 
| PubMedID: 27157710 | 
| Title : Modification of the anabaseine pyridine nucleus allows achieving binding and functional selectivity for the alpha3beta4 nicotinic acetylcholine receptor subtype - Matera_2016_Eur.J.Med.Chem_108_392 | 
| Author(s) : Matera C , Quadri M , Sciaccaluga M , Pome DY , Fasoli F , De Amici M , Fucile S , Gotti C , Dallanoce C , Grazioso G | 
| Ref : Eur Journal of Medicinal Chemistry , 108 :392 , 2016 | 
| Abstract : | 
| PubMedSearch : Matera_2016_Eur.J.Med.Chem_108_392 | 
| PubMedID: 26706350 | 
| Title : Neuronal Acetylcholine Nicotinic Receptors as New Targets for Lung Cancer Treatment - Mucchietto_2016_Curr.Pharm.Des_22_2160 | 
| Author(s) : Mucchietto V , Crespi A , Fasoli F , Clementi F , Gotti C | 
| Ref : Curr Pharm Des , 22 :2160 , 2016 | 
| Abstract : | 
| PubMedSearch : Mucchietto_2016_Curr.Pharm.Des_22_2160 | 
| PubMedID: 26845123 | 
| Title : Chemistry and Pharmacology of a Series of Unichiral Analogues of 2-(2-Pyrrolidinyl)-1,4-benzodioxane, Prolinol Phenyl Ether, and Prolinol 3-Pyridyl Ether Designed as alpha4beta2-Nicotinic Acetylcholine Receptor Agonists - Bolchi_2015_J.Med.Chem_58_6665 | 
| Author(s) : Bolchi C , Valoti E , Gotti C , Fasoli F , Ruggeri P , Fumagalli L , Binda M , Mucchietto V , Sciaccaluga M , Budriesi R , Fucile S , Pallavicini M | 
| Ref : Journal of Medicinal Chemistry , 58 :6665 , 2015 | 
| Abstract : | 
| PubMedSearch : Bolchi_2015_J.Med.Chem_58_6665 | 
| PubMedID: 26225816 | 
| Title : Design of novel 3,6-diazabicyclo[3.1.1]heptane derivatives with potent and selective affinities for alpha4beta2 neuronal nicotinic acetylcholine receptors - Deligia_2015_Eur.J.Med.Chem_103_429 | 
| Author(s) : Deligia F , Deiana V , Gotti C , Lazzari P , Bottazzi ME , Pucci L , Fasoli F , Ragusa G , Pinna GA , Murineddu G | 
| Ref : Eur Journal of Medicinal Chemistry , 103 :429 , 2015 | 
| Abstract : | 
| PubMedSearch : Deligia_2015_Eur.J.Med.Chem_103_429 | 
| PubMedID: 26383127 | 
| Title : Structure of neuronal nicotinic receptors - Fasoli_2015_Curr.Top.Behav.Neurosci_23_1 | 
| Author(s) : Fasoli F , Gotti C | 
| Ref : Curr Top Behavioral Neuroscience , 23 :1 , 2015 | 
| Abstract : | 
| PubMedSearch : Fasoli_2015_Curr.Top.Behav.Neurosci_23_1 | 
| PubMedID: 25655885 | 
| Title : Different physiological and behavioural effects of e-cigarette vapour and cigarette smoke in mice - Ponzoni_2015_Eur.Neuropsychopharmacol_25_1775 | 
| Author(s) : Ponzoni L , Moretti M , Sala M , Fasoli F , Mucchietto V , Lucini V , Cannazza G , Gallesi G , Castellana CN , Clementi F , Zoli M , Gotti C , Braida D | 
| Ref : European Neuropsychopharmacology , 25 :1775 , 2015 | 
| Abstract : | 
| PubMedSearch : Ponzoni_2015_Eur.Neuropsychopharmacol_25_1775 | 
| PubMedID: 26141510 | 
| Title : Synthesis and Pharmacological Evaluation of alpha4beta2 Nicotinic Ligands with a 3-Fluoropyrrolidine Nucleus - Tamborini_2015_ChemMedChem_10_1071 | 
| Author(s) : Tamborini L , Pinto A , Ettari R , Gotti C , Fasoli F , Conti P , De Micheli C | 
| Ref : ChemMedChem , 10 :1071 , 2015 | 
| Abstract : | 
| PubMedSearch : Tamborini_2015_ChemMedChem_10_1071 | 
| PubMedID: 25882435 | 
| Title : Poster: Nicotinic receptors increase cell proliferation and tumour progression in non-small cell lung cancer cell line - | 
| Author(s) : Mucchietto V , Fasoli F , Benfante R , Maroli A , Cattaneo MG , Pistillo F , Moretti M , Bolchi C , Pallavicini M , Clementi F , Gotti C | 
| Ref : Biochemical Pharmacology , 97 :631 , 2015 | 
| PubMedID: | 
| Title : The cytisine derivatives, CC4 and CC26, reduce nicotine-induced conditioned place preference in zebrafish by acting on heteromeric neuronal nicotinic acetylcholine receptors - Ponzoni_2014_Psychopharmacology.(Berl)_231_4681 | 
| Author(s) : Ponzoni L , Braida D , Pucci L , Andrea D , Fasoli F , Manfredi I , Papke RL , Stokes C , Cannazza G , Clementi F , Gotti C , Sala M | 
| Ref : Psychopharmacology (Berl) , 231 :4681 , 2014 | 
| Abstract : | 
| PubMedSearch : Ponzoni_2014_Psychopharmacology.(Berl)_231_4681 | 
| PubMedID: 24862365 | 
| Title : (+)-Laburnamine, a natural selective ligand and partial agonist for the alpha4beta2 nicotinic receptor subtype - Tasso_2013_J.Nat.Prod_76_727 | 
| Author(s) : Tasso B , Novelli F , Sparatore F , Fasoli F , Gotti C | 
| Ref : Journal of Natural Products , 76 :727 , 2013 | 
| Abstract : | 
| PubMedSearch : Tasso_2013_J.Nat.Prod_76_727 | 
| PubMedID: 23461628 | 
| Title : Design, synthesis and binding affinity of acetylcholine carbamoyl analogues - Bolchi_2013_Bioorg.Med.Chem.Lett_23_6481 | 
| Author(s) : Bolchi C , Valoti E , Binda M , Fasoli F , Ferrara R , Fumagalli L , Gotti C , Matucci R , Vistoli G , Pallavicini M | 
| Ref : Bioorganic & Medicinal Chemistry Lett , 23 :6481 , 2013 | 
| Abstract : | 
| PubMedSearch : Bolchi_2013_Bioorg.Med.Chem.Lett_23_6481 | 
| PubMedID: 24128660 | 
| Title : CC4, a dimer of cytisine, is a selective partial agonist at alpha4beta2\/alpha6beta2 nAChR with improved selectivity for tobacco smoking cessation - Sala_2013_Br.J.Pharmacol_168_835 | 
| Author(s) : Sala M , Braida D , Pucci L , Manfredi I , Marks MJ , Wageman CR , Grady SR , Loi B , Fucile S , Fasoli F , Zoli M , Tasso B , Sparatore F , Clementi F , Gotti C | 
| Ref : British Journal of Pharmacology , 168 :835 , 2013 | 
| Abstract : | 
| PubMedSearch : Sala_2013_Br.J.Pharmacol_168_835 | 
| PubMedID: 22957729 |