Title : Chemistry and Pharmacology of a Series of Unichiral Analogues of 2-(2-Pyrrolidinyl)-1,4-benzodioxane, Prolinol Phenyl Ether, and Prolinol 3-Pyridyl Ether Designed as alpha4beta2-Nicotinic Acetylcholine Receptor Agonists - Bolchi_2015_J.Med.Chem_58_6665 |
Author(s) : Bolchi C , Valoti E , Gotti C , Fasoli F , Ruggeri P , Fumagalli L , Binda M , Mucchietto V , Sciaccaluga M , Budriesi R , Fucile S , Pallavicini M |
Ref : Journal of Medicinal Chemistry , 58 :6665 , 2015 |
Abstract : |
PubMedSearch : Bolchi_2015_J.Med.Chem_58_6665 |
PubMedID: 26225816 |
Title : Design, synthesis, and biological evaluation of symmetrically and unsymmetrically substituted methoctramine-related polyamines as muscular nicotinic receptor noncompetitive antagonists - Rosini_1999_J.Med.Chem_42_5212 |
Author(s) : Rosini M , Budriesi R , Bixel MG , Bolognesi ML , Chiarini A , Hucho F , Krogsgaard-Larsen P , Mellor IR , Minarini A , Tumiatti V , Usherwood PN , Melchiorre C |
Ref : Journal of Medicinal Chemistry , 42 :5212 , 1999 |
Abstract : |
PubMedSearch : Rosini_1999_J.Med.Chem_42_5212 |
PubMedID: 10602706 |
Title : Acetylcholinesterase Noncovalent Inhibitors Based on a Polyamine Backbone for Potential Use against Alzheimer's Disease - |
Author(s) : Melchiorre C , Andrisano V , Bolognesi ML , Budriesi R , Cavalli A , Cavrini V , Rosini M , Tumiatti V , Recanatini M |
Ref : Journal of Medicinal Chemistry , 41 :4186 , 1998 |
PubMedID: 9784091 |
Title : Universal template approach to drug design: polyamines as selective muscarinic receptor antagonists - Bolognesi_1998_J.Med.Chem_41_4150 |
Author(s) : Bolognesi ML , Minarini A , Budriesi R , Cacciaguerra S , Chiarini A , Spampinato S , Tumiatti V , Melchiorre C |
Ref : Journal of Medicinal Chemistry , 41 :4150 , 1998 |
Abstract : |
PubMedSearch : Bolognesi_1998_J.Med.Chem_41_4150 |
PubMedID: 9767650 |
Title : The design of novel methoctramine-related tetraamines as muscarinic receptor subtype selective antagonists - Melchiorre_1995_Life.Sci_56(11-12)_837 |
Author(s) : Melchiorre C , Minarini A , Budriesi R , Chiarini A , Spampinato S , Tumiatti V |
Ref : Life Sciences , 56(11-12) :837 , 1995 |
Abstract : |
PubMedSearch : Melchiorre_1995_Life.Sci_56(11-12)_837 |
PubMedID: 10188783 |