Title : Synthesis and biological evaluation of novel hybrids of highly potent and selective alpha4beta2-Nicotinic acetylcholine receptor (nAChR) partial agonists - Zhang_2016_Eur.J.Med.Chem_124_689 |
Author(s) : Zhang HK , Eaton JB , Fedolak A , Gunosewoyo H , Onajole OK , Brunner D , Lukas RJ , Yu LF , Kozikowski AP |
Ref : Eur Journal of Medicinal Chemistry , 124 :689 , 2016 |
Abstract : Zhang_2016_Eur.J.Med.Chem_124_689 |
ESTHER : Zhang_2016_Eur.J.Med.Chem_124_689 |
PubMedSearch : Zhang_2016_Eur.J.Med.Chem_124_689 |
PubMedID: 27639361 |
Title : Chemistry and behavioral studies identify chiral cyclopropanes as selective alpha4beta2-nicotinic acetylcholine receptor partial agonists exhibiting an antidepressant profile - Zhang_2012_J.Med.Chem_55_717 |
Author(s) : Zhang H , Tuckmantel W , Eaton JB , Yuen PW , Yu LF , Bajjuri KM , Fedolak A , Wang D , Ghavami A , Caldarone B , Paterson NE , Lowe DA , Brunner D , Lukas RJ , Kozikowski AP |
Ref : Journal of Medicinal Chemistry , 55 :717 , 2012 |
Abstract : Zhang_2012_J.Med.Chem_55_717 |
ESTHER : Zhang_2012_J.Med.Chem_55_717 |
PubMedSearch : Zhang_2012_J.Med.Chem_55_717 |
PubMedID: 22171543 |
Title : Discovery of isoxazole analogues of sazetidine-A as selective alpha4beta2-nicotinic acetylcholine receptor partial agonists for the treatment of depression - Liu_2011_J.Med.Chem_54_7280 |
Author(s) : Liu J , Yu LF , Eaton JB , Caldarone B , Cavino K , Ruiz C , Terry M , Fedolak A , Wang D , Ghavami A , Lowe DA , Brunner D , Lukas RJ , Kozikowski AP |
Ref : Journal of Medicinal Chemistry , 54 :7280 , 2011 |
Abstract : Liu_2011_J.Med.Chem_54_7280 |
ESTHER : Liu_2011_J.Med.Chem_54_7280 |
PubMedSearch : Liu_2011_J.Med.Chem_54_7280 |
PubMedID: 21905669 |
Title : Dissociation between duration of action in the forced swim test in mice and nicotinic acetylcholine receptor occupancy with sazetidine, varenicline, and 5-I-A85380 - Caldarone_2011_Psychopharmacology.(Berl)_217_199 |
Author(s) : Caldarone BJ , Wang D , Paterson NE , Manzano M , Fedolak A , Cavino K , Kwan M , Hanania T , Chellappan SK , Kozikowski AP , Olivier B , Picciotto MR , Ghavami A |
Ref : Psychopharmacology (Berl) , 217 :199 , 2011 |
Abstract : Caldarone_2011_Psychopharmacology.(Berl)_217_199 |
ESTHER : Caldarone_2011_Psychopharmacology.(Berl)_217_199 |
PubMedSearch : Caldarone_2011_Psychopharmacology.(Berl)_217_199 |
PubMedID: 21487659 |