| Title : The preparation, in vitro screening and molecular docking of symmetrical bisquaternary cholinesterase inhibitors containing a but-(2E)-en-1,4-diyl connecting linkage - Musilek_2011_J.Enzyme.Inhib.Med.Chem_26_245 |
| Author(s) : Musilek K , Pavlikova R , Marek J , Komloova M , Holas O , Hrabinova M , Pohanka M , Dohnal V , Dolezal M , Gunn-Moore F , Kuca K |
| Ref : J Enzyme Inhib Med Chem , 26 :245 , 2011 |
| Abstract : |
| PubMedSearch : Musilek_2011_J.Enzyme.Inhib.Med.Chem_26_245 |
| PubMedID: 21406034 |
| Title : Design, evaluation and structure-activity relationship studies of the AChE reactivators against organophosphorus pesticides - Musilek_2011_Med.Res.Rev_31_548 |
| Author(s) : Musilek K , Dolezal M , Gunn-Moore F , Kuca K |
| Ref : Med Res Rev , 31 :548 , 2011 |
| Abstract : |
| PubMedSearch : Musilek_2011_Med.Res.Rev_31_548 |
| PubMedID: 20027669 |
| Title : The preparation, in vitro screening and molecular docking of symmetrical bisquaternary cholinesterase inhibitors containing a but-(2E)-en-1,4-diyl connecting linkage - Musilek_2011_J.Enzyme.Inhib.Med.Chem_26_245 |
| Author(s) : Musilek K , Pavlikova R , Marek J , Komloova M , Holas O , Hrabinova M , Pohanka M , Dohnal V , Dolezal M , Gunn-Moore F , Kuca K |
| Ref : J Enzyme Inhib Med Chem , 26 :245 , 2011 |
| Abstract : |
| PubMedSearch : Musilek_2011_J.Enzyme.Inhib.Med.Chem_26_245 |
| PubMedID: 21406034 |
| Title : Preparation, in vitro screening and molecular modelling of symmetrical bis-quinolinium cholinesterase inhibitors--implications for early myasthenia gravis treatment - Komloova_2011_Bioorg.Med.Chem.Lett_21_2505 |
| Author(s) : Komloova M , Musilek K , Horova A , Holas O , Dohnal V , Gunn-Moore F , Kuca K |
| Ref : Bioorganic & Medicinal Chemistry Lett , 21 :2505 , 2011 |
| Abstract : |
| PubMedSearch : Komloova_2011_Bioorg.Med.Chem.Lett_21_2505 |
| PubMedID: 21397501 |
| Title : Design, evaluation and structure-activity relationship studies of the AChE reactivators against organophosphorus pesticides - Musilek_2011_Med.Res.Rev_31_548 |
| Author(s) : Musilek K , Dolezal M , Gunn-Moore F , Kuca K |
| Ref : Med Res Rev , 31 :548 , 2011 |
| Abstract : |
| PubMedSearch : Musilek_2011_Med.Res.Rev_31_548 |
| PubMedID: 20027669 |
| Title : Mono-oxime bisquaternary acetylcholinesterase reactivators with prop-1,3-diyl linkage-Preparation, in vitro screening and molecular docking - Musilek_2011_Bioorg.Med.Chem_19_754 |
| Author(s) : Musilek K , Komloova M , Holas O , Horova A , Pohanka M , Gunn-Moore F , Dohnal V , Dolezal M , Kuca K |
| Ref : Bioorganic & Medicinal Chemistry , 19 :754 , 2011 |
| Abstract : |
| PubMedSearch : Musilek_2011_Bioorg.Med.Chem_19_754 |
| PubMedID: 21215642 |
| Title : Preparation, in vitro screening and molecular modelling of symmetrical bis-quinolinium cholinesterase inhibitors--implications for early myasthenia gravis treatment - Komloova_2011_Bioorg.Med.Chem.Lett_21_2505 |
| Author(s) : Komloova M , Musilek K , Horova A , Holas O , Dohnal V , Gunn-Moore F , Kuca K |
| Ref : Bioorganic & Medicinal Chemistry Lett , 21 :2505 , 2011 |
| Abstract : |
| PubMedSearch : Komloova_2011_Bioorg.Med.Chem.Lett_21_2505 |
| PubMedID: 21397501 |
| Title : Mono-oxime bisquaternary acetylcholinesterase reactivators with prop-1,3-diyl linkage-Preparation, in vitro screening and molecular docking - Musilek_2011_Bioorg.Med.Chem_19_754 |
| Author(s) : Musilek K , Komloova M , Holas O , Horova A , Pohanka M , Gunn-Moore F , Dohnal V , Dolezal M , Kuca K |
| Ref : Bioorganic & Medicinal Chemistry , 19 :754 , 2011 |
| Abstract : |
| PubMedSearch : Musilek_2011_Bioorg.Med.Chem_19_754 |
| PubMedID: 21215642 |
| Title : The preparation, in vitro screening and molecular docking of symmetrical bisquaternary cholinesterase inhibitors containing a but-(2E)-en-1,4-diyl connecting linkage - Musilek_2011_J.Enzyme.Inhib.Med.Chem_26_245 |
| Author(s) : Musilek K , Pavlikova R , Marek J , Komloova M , Holas O , Hrabinova M , Pohanka M , Dohnal V , Dolezal M , Gunn-Moore F , Kuca K |
| Ref : J Enzyme Inhib Med Chem , 26 :245 , 2011 |
| Abstract : |
| PubMedSearch : Musilek_2011_J.Enzyme.Inhib.Med.Chem_26_245 |
| PubMedID: 21406034 |
| Title : Preparation, in vitro screening and molecular modelling of symmetrical bis-quinolinium cholinesterase inhibitors--implications for early myasthenia gravis treatment - Komloova_2011_Bioorg.Med.Chem.Lett_21_2505 |
| Author(s) : Komloova M , Musilek K , Horova A , Holas O , Dohnal V , Gunn-Moore F , Kuca K |
| Ref : Bioorganic & Medicinal Chemistry Lett , 21 :2505 , 2011 |
| Abstract : |
| PubMedSearch : Komloova_2011_Bioorg.Med.Chem.Lett_21_2505 |
| PubMedID: 21397501 |
| Title : Design, evaluation and structure-activity relationship studies of the AChE reactivators against organophosphorus pesticides - Musilek_2011_Med.Res.Rev_31_548 |
| Author(s) : Musilek K , Dolezal M , Gunn-Moore F , Kuca K |
| Ref : Med Res Rev , 31 :548 , 2011 |
| Abstract : |
| PubMedSearch : Musilek_2011_Med.Res.Rev_31_548 |
| PubMedID: 20027669 |
| Title : Mono-oxime bisquaternary acetylcholinesterase reactivators with prop-1,3-diyl linkage-Preparation, in vitro screening and molecular docking - Musilek_2011_Bioorg.Med.Chem_19_754 |
| Author(s) : Musilek K , Komloova M , Holas O , Horova A , Pohanka M , Gunn-Moore F , Dohnal V , Dolezal M , Kuca K |
| Ref : Bioorganic & Medicinal Chemistry , 19 :754 , 2011 |
| Abstract : |
| PubMedSearch : Musilek_2011_Bioorg.Med.Chem_19_754 |
| PubMedID: 21215642 |
| Title : Structure-activity relationship of quaternary acetylcholinesterase inhibitors - outlook for early myasthenia gravis treatment - Komloova_2010_Curr.Med.Chem_17_1810 |
| Author(s) : Komloova M , Musilek K , Dolezal M , Gunn-Moore F , Kuca K |
| Ref : Curr Med Chem , 17 :1810 , 2010 |
| Abstract : |
| PubMedSearch : Komloova_2010_Curr.Med.Chem_17_1810 |
| PubMedID: 20345342 |
| Title : Structure-activity relationship of quaternary acetylcholinesterase inhibitors - outlook for early myasthenia gravis treatment - Komloova_2010_Curr.Med.Chem_17_1810 |
| Author(s) : Komloova M , Musilek K , Dolezal M , Gunn-Moore F , Kuca K |
| Ref : Curr Med Chem , 17 :1810 , 2010 |
| Abstract : |
| PubMedSearch : Komloova_2010_Curr.Med.Chem_17_1810 |
| PubMedID: 20345342 |
| Title : Structure-activity relationship of quaternary acetylcholinesterase inhibitors - outlook for early myasthenia gravis treatment - Komloova_2010_Curr.Med.Chem_17_1810 |
| Author(s) : Komloova M , Musilek K , Dolezal M , Gunn-Moore F , Kuca K |
| Ref : Curr Med Chem , 17 :1810 , 2010 |
| Abstract : |
| PubMedSearch : Komloova_2010_Curr.Med.Chem_17_1810 |
| PubMedID: 20345342 |
| Title : RP-HPLC determination of the lipophilicity of bispyridinium reactivators of acetylcholinesterase bearing a but-2-ene connecting linker - Musilek_2008_Anal.Bioanal.Chem_391_367 |
| Author(s) : Musilek K , Jampilek J , Dohnal J , Jun D , Gunn-Moore F , Dolezal M , Kuca K |
| Ref : Anal Bioanal Chem , 391 :367 , 2008 |
| Abstract : |
| PubMedSearch : Musilek_2008_Anal.Bioanal.Chem_391_367 |
| PubMedID: 18369602 |
| Title : RP-HPLC determination of the lipophilicity of bispyridinium reactivators of acetylcholinesterase bearing a but-2-ene connecting linker - Musilek_2008_Anal.Bioanal.Chem_391_367 |
| Author(s) : Musilek K , Jampilek J , Dohnal J , Jun D , Gunn-Moore F , Dolezal M , Kuca K |
| Ref : Anal Bioanal Chem , 391 :367 , 2008 |
| Abstract : |
| PubMedSearch : Musilek_2008_Anal.Bioanal.Chem_391_367 |
| PubMedID: 18369602 |
| Title : RP-HPLC determination of the lipophilicity of bispyridinium reactivators of acetylcholinesterase bearing a but-2-ene connecting linker - Musilek_2008_Anal.Bioanal.Chem_391_367 |
| Author(s) : Musilek K , Jampilek J , Dohnal J , Jun D , Gunn-Moore F , Dolezal M , Kuca K |
| Ref : Anal Bioanal Chem , 391 :367 , 2008 |
| Abstract : |
| PubMedSearch : Musilek_2008_Anal.Bioanal.Chem_391_367 |
| PubMedID: 18369602 |
| Title : Design of a potent reactivator of tabun-inhibited acetylcholinesterase--synthesis and evaluation of (E)-1-(4-carbamoylpyridinium)-4-(4-hydroxyiminomethylpyridinium)-but-2-ene dibromide (K203) - Musilek_2007_J.Med.Chem_50_5514 |
| Author(s) : Musilek K , Jun D , Cabal J , Kassa J , Gunn-Moore F , Kuca K |
| Ref : Journal of Medicinal Chemistry , 50 :5514 , 2007 |
| Abstract : |
| PubMedSearch : Musilek_2007_J.Med.Chem_50_5514 |
| PubMedID: 17924614 |
| Title : Monooxime reactivators of acetylcholinesterase with (E)-but-2-ene linker: preparation and reactivation of tabun- and paraoxon-inhibited acetylcholinesterase - Musilek_2007_Bioorg.Med.Chem_15_6733 |
| Author(s) : Musilek K , Holas O , Jun D , Dohnal V , Gunn-Moore F , Opletalova V , Dolezal M , Kuca K |
| Ref : Bioorganic & Medicinal Chemistry , 15 :6733 , 2007 |
| Abstract : |
| PubMedSearch : Musilek_2007_Bioorg.Med.Chem_15_6733 |
| PubMedID: 17764957 |
| Title : Design of a potent reactivator of tabun-inhibited acetylcholinesterase--synthesis and evaluation of (E)-1-(4-carbamoylpyridinium)-4-(4-hydroxyiminomethylpyridinium)-but-2-ene dibromide (K203) - Musilek_2007_J.Med.Chem_50_5514 |
| Author(s) : Musilek K , Jun D , Cabal J , Kassa J , Gunn-Moore F , Kuca K |
| Ref : Journal of Medicinal Chemistry , 50 :5514 , 2007 |
| Abstract : |
| PubMedSearch : Musilek_2007_J.Med.Chem_50_5514 |
| PubMedID: 17924614 |
| Title : Monooxime reactivators of acetylcholinesterase with (E)-but-2-ene linker: preparation and reactivation of tabun- and paraoxon-inhibited acetylcholinesterase - Musilek_2007_Bioorg.Med.Chem_15_6733 |
| Author(s) : Musilek K , Holas O , Jun D , Dohnal V , Gunn-Moore F , Opletalova V , Dolezal M , Kuca K |
| Ref : Bioorganic & Medicinal Chemistry , 15 :6733 , 2007 |
| Abstract : |
| PubMedSearch : Musilek_2007_Bioorg.Med.Chem_15_6733 |
| PubMedID: 17764957 |
| Title : Design of a potent reactivator of tabun-inhibited acetylcholinesterase--synthesis and evaluation of (E)-1-(4-carbamoylpyridinium)-4-(4-hydroxyiminomethylpyridinium)-but-2-ene dibromide (K203) - Musilek_2007_J.Med.Chem_50_5514 |
| Author(s) : Musilek K , Jun D , Cabal J , Kassa J , Gunn-Moore F , Kuca K |
| Ref : Journal of Medicinal Chemistry , 50 :5514 , 2007 |
| Abstract : |
| PubMedSearch : Musilek_2007_J.Med.Chem_50_5514 |
| PubMedID: 17924614 |
| Title : Monooxime reactivators of acetylcholinesterase with (E)-but-2-ene linker: preparation and reactivation of tabun- and paraoxon-inhibited acetylcholinesterase - Musilek_2007_Bioorg.Med.Chem_15_6733 |
| Author(s) : Musilek K , Holas O , Jun D , Dohnal V , Gunn-Moore F , Opletalova V , Dolezal M , Kuca K |
| Ref : Bioorganic & Medicinal Chemistry , 15 :6733 , 2007 |
| Abstract : |
| PubMedSearch : Musilek_2007_Bioorg.Med.Chem_15_6733 |
| PubMedID: 17764957 |