Title : Extended structure-activity relationship and pharmacokinetic investigation of (4-quinolinoyl)glycyl-2-cyanopyrrolidine inhibitors of fibroblast activation protein (FAP) - Jansen_2014_J.Med.Chem_57_3053 |
Author(s) : Jansen K , Heirbaut L , Verkerk R , Cheng JD , Joossens J , Cos P , Maes L , Lambeir AM , De Meester I , Augustyns K , Van der Veken P |
Ref : Journal of Medicinal Chemistry , 57 :3053 , 2014 |
Abstract : |
PubMedSearch : Jansen_2014_J.Med.Chem_57_3053 |
PubMedID: 24617858 |
Title : Selective Inhibitors of Fibroblast Activation Protein (FAP) with a (4-Quinolinoyl)-glycyl-2-cyanopyrrolidine Scaffold - Jansen_2013_ACS.Med.Chem.Lett_4_491 |
Author(s) : Jansen K , Heirbaut L , Cheng JD , Joossens J , Ryabtsova O , Cos P , Maes L , Lambeir AM , De Meester I , Augustyns K , Van der Veken P |
Ref : ACS Med Chem Lett , 4 :491 , 2013 |
Abstract : |
PubMedSearch : Jansen_2013_ACS.Med.Chem.Lett_4_491 |
PubMedID: 24900696 |
Title : Acylated Gly-(2-cyano)pyrrolidines as inhibitors of fibroblast activation protein (FAP) and the issue of FAP\/prolyl oligopeptidase (PREP)-selectivity - Ryabtsova_2012_Bioorg.Med.Chem.Lett_22_3412 |
Author(s) : Ryabtsova O , Jansen K , Van Goethem S , Joossens J , Cheng JD , Lambeir AM , De Meester I , Augustyns K , Van der Veken P |
Ref : Bioorganic & Medicinal Chemistry Lett , 22 :3412 , 2012 |
Abstract : |
PubMedSearch : Ryabtsova_2012_Bioorg.Med.Chem.Lett_22_3412 |
PubMedID: 22525314 |
Title : The toxicity of mixtures of specific organophosphate compounds is modulated by paraoxonase 1 status - Cole_2010_Adv.Exp.Med.Biol_660_47 |
Author(s) : Cole TB , Jansen K , Park S , Li WF , Furlong CE , Costa LG |
Ref : Advances in Experimental Medicine & Biology , 660 :47 , 2010 |
Abstract : |
PubMedSearch : Cole_2010_Adv.Exp.Med.Biol_660_47 |
PubMedID: 20221870 |