Title : Novel Uracil-Based Inhibitors of Acetylcholinesterase with Potency for Treating Memory Impairment in an Animal Model of Alzheimer's Disease - Semenov_2022_Molecules_27_ |
Author(s) : Semenov VE , Zueva IV , Lushchekina SV , Suleimanov EG , Gubaidullina LM , Shulaeva MM , Lenina OA , Petrov KA |
Ref : Molecules , 27 : , 2022 |
Abstract : Semenov_2022_Molecules_27_ |
ESTHER : Semenov_2022_Molecules_27_ |
PubMedSearch : Semenov_2022_Molecules_27_ |
PubMedID: 36431954 |
Title : Novel slow-binding reversible acetylcholinesterase inhibitors based on uracil moieties for possible treatment of myasthenia gravis and protection from organophosphate poisoning - Saifina_2022_Eur.J.Med.Chem_246_114949 |
Author(s) : Saifina LF , Abdalla M , Gubaidullina LM , Zueva IV , Eltayb WA , El-Arabey AA , Kharlamova AD , Lenina OA , Semenov VE , Petrov KA |
Ref : Eur Journal of Medicinal Chemistry , 246 :114949 , 2022 |
Abstract : Saifina_2022_Eur.J.Med.Chem_246_114949 |
ESTHER : Saifina_2022_Eur.J.Med.Chem_246_114949 |
PubMedSearch : Saifina_2022_Eur.J.Med.Chem_246_114949 |
PubMedID: 36462442 |
Title : Balanced modulation of neuromuscular synaptic transmission via M1 and M2 muscarinic receptors during inhibition of cholinesterases - Lenina_2022_Sci.Rep_12_1688 |
Author(s) : Lenina OA , Petrov KA |
Ref : Sci Rep , 12 :1688 , 2022 |
Abstract : Lenina_2022_Sci.Rep_12_1688 |
ESTHER : Lenina_2022_Sci.Rep_12_1688 |
PubMedSearch : Lenina_2022_Sci.Rep_12_1688 |
PubMedID: 35105922 |
Title : Protective effects of m-(tert-butyl) trifluoroacetophenone, a transition state analogue of acetylcholine, against paraoxon toxicity and memory impairments - Zueva_2021_Chem.Biol.Interact_345_109558 |
Author(s) : Zueva IV , Lenina OA , Kayumova RM , Petrov KA , Masson P |
Ref : Chemico-Biological Interactions , 345 :109558 , 2021 |
Abstract : Zueva_2021_Chem.Biol.Interact_345_109558 |
ESTHER : Zueva_2021_Chem.Biol.Interact_345_109558 |
PubMedSearch : Zueva_2021_Chem.Biol.Interact_345_109558 |
PubMedID: 34147486 |
Title : Slow-binding reversible inhibitor of acetylcholinesterase with long-lasting action for prophylaxis of organophosphate poisoning - Lenina_2020_Sci.Rep_10_16611 |
Author(s) : Lenina OA , Zueva IV , Zobov VV , Semenov VE , Masson P , Petrov KA |
Ref : Sci Rep , 10 :16611 , 2020 |
Abstract : Lenina_2020_Sci.Rep_10_16611 |
ESTHER : Lenina_2020_Sci.Rep_10_16611 |
PubMedSearch : Lenina_2020_Sci.Rep_10_16611 |
PubMedID: 33024231 |
Title : Novel Acetylcholinesterase Inhibitors Based on Uracil Moiety for Possible Treatment of Alzheimer Disease - Semenov_2020_Molecules_25_ |
Author(s) : Semenov VE , Zueva IV , Mukhamedyarov MA , Lushchekina SV , Petukhova EO , Gubaidullina LM , Krylova ES , Saifina LF , Lenina OA , Petrov KA |
Ref : Molecules , 25 : , 2020 |
Abstract : Semenov_2020_Molecules_25_ |
ESTHER : Semenov_2020_Molecules_25_ |
PubMedSearch : Semenov_2020_Molecules_25_ |
PubMedID: 32932702 |
Title : Water-soluble betaines and amines based on thiacalix[4]arene scaffold as new cholinesterase inhibitors - Padnya_2019_Bioorg.Chem__103455 |
Author(s) : Padnya PL , Bayarashov EE , Zueva IV , Lushchekina SV , Lenina OA , Evtugyn VG , Osin YN , Petrov KA , Stoikov, II |
Ref : Bioorg Chem , :103455 , 2019 |
Abstract : Padnya_2019_Bioorg.Chem__103455 |
ESTHER : Padnya_2019_Bioorg.Chem__103455 |
PubMedSearch : Padnya_2019_Bioorg.Chem__103455 |
PubMedID: 31791680 |
Title : 6-Methyluracil derivatives as peripheral site ligand-hydroxamic acid conjugates: Reactivation for paraoxon-inhibited acetylcholinesterase - Semenov_2019_Eur.J.Med.Chem_185_111787 |
Author(s) : Semenov VE , Zueva IV , Lushchekina SV , Lenina OA , Gubaidullina LM , Saifina LF , Shulaeva MM , Kayumova RM , Saifina AF , Gubaidullin AT , Kondrashova SA , Latypov SK , Masson P , Petrov KA |
Ref : Eur Journal of Medicinal Chemistry , 185 :111787 , 2019 |
Abstract : Semenov_2019_Eur.J.Med.Chem_185_111787 |
ESTHER : Semenov_2019_Eur.J.Med.Chem_185_111787 |
PubMedSearch : Semenov_2019_Eur.J.Med.Chem_185_111787 |
PubMedID: 31675511 |
Title : Specific inhibition of acetylcholinesterase as an approach to decrease muscarinic side effects during myasthenia gravis treatment - Petrov_2018_Sci.Rep_8_304 |
Author(s) : Petrov KA , Kharlamova AD , Lenina OA , Nurtdinov AR , Sitdykova ME , Ilyin VI , Zueva IV , Nikolsky EE |
Ref : Sci Rep , 8 :304 , 2018 |
Abstract : Petrov_2018_Sci.Rep_8_304 |
ESTHER : Petrov_2018_Sci.Rep_8_304 |
PubMedSearch : Petrov_2018_Sci.Rep_8_304 |
PubMedID: 29321572 |