Nikolsky EE

General

Full name : Nikolsky Evgeny E

First name : Evgeny E

Mail : Kazan State Medical University\; Department of Medical and Biological Physics\; 15\; Butlerova st.\; 420053

Zip Code :

City :

Country : Russia

Email : eenik1947@mail.ru

Phone : +78432387547

Fax :

Website :

Directory :

Comment
Professor Evgeny E. Nikolsky passed away in June 2018 at 71. He was member of the Russian Academy of Science, Professor of physiology at the Medical School of Kazan and director of the Neuropharmacology laboratory of the Federal University of Kazan. Among other events he co-organized the 11th International Meeting on Cholinesterases in Kazan (RU) in 2012

References (29)

Title : Specific inhibition of acetylcholinesterase as an approach to decrease muscarinic side effects during myasthenia gravis treatment - Petrov_2018_Sci.Rep_8_304
Author(s) : Petrov KA , Kharlamova AD , Lenina OA , Nurtdinov AR , Sitdykova ME , Ilyin VI , Zueva IV , Nikolsky EE
Ref : Sci Rep , 8 :304 , 2018
Abstract :
PubMedSearch : Petrov_2018_Sci.Rep_8_304
PubMedID: 29321572

Title : C-547, a 6-methyluracil derivative with long-lasting binding and rebinding on acetylcholinesterase: Pharmacokinetic and pharmacodynamic studies - Petrov_2018_Neuropharmacol_131_304
Author(s) : Petrov KA , Zueva IV , Kovyazina IV , Sedov I , Lushchekina SV , Kharlamova AD , Lenina O , Koshkin S , Shtyrlin Y , Nikolsky EE , Masson P
Ref : Neuropharmacology , 131 :304 , 2018
Abstract :
PubMedSearch : Petrov_2018_Neuropharmacol_131_304
PubMedID: 29277489

Title : Autoregulation of Acetylcholine Release and Micro-Pharmacodynamic Mechanisms at Neuromuscular Junction: Selective Acetylcholinesterase Inhibitors for Therapy of Myasthenic Syndromes - Petrov_2018_Front.Pharmacol_9_766
Author(s) : Petrov KA , Nikolsky EE , Masson P
Ref : Front Pharmacol , 9 :766 , 2018
Abstract :
PubMedSearch : Petrov_2018_Front.Pharmacol_9_766
PubMedID: 30050445

Title : Cholinergic Nociceptive Mechanisms in Rat Meninges and Trigeminal Ganglia: Potential Implications for Migraine Pain - Shelukhina_2017_Front.Neurol_8_163
Author(s) : Shelukhina I , Mikhailov N , Abushik P , Nurullin LF , Nikolsky EE , Giniatullin R
Ref : Front Neurol , 8 :163 , 2017
Abstract :
PubMedSearch : Shelukhina_2017_Front.Neurol_8_163
PubMedID: 28496430

Title : Nanoparticle-Delivered 2-PAM for Rat Brain Protection against Paraoxon Central Toxicity - Pashirova_2017_ACS.Appl.Mater.Interfaces_9_16922
Author(s) : Pashirova TN , Zueva IV , Petrov KA , Babaev VM , Lukashenko SS , Rizvanov IK , Souto EB , Nikolsky EE , Zakharova LY , Masson P , Sinyashin OG
Ref : ACS Appl Mater Interfaces , 9 :16922 , 2017
Abstract :
PubMedSearch : Pashirova_2017_ACS.Appl.Mater.Interfaces_9_16922
PubMedID: 28504886

Title : Slow-binding inhibition of acetylcholinesterase by an alkylammonium derivative of 6-methyluracil: mechanism and possible advantages for myasthenia gravis treatment - Kharlamova_2016_Biochem.J_473_1225
Author(s) : Kharlamova AD , Lushchekina SV , Petrov KA , Kots ED , Nachon F , Villard-Wandhammer M , Zueva IV , Krejci E , Reznik VS , Zobov VV , Nikolsky EE , Masson P
Ref : Biochemical Journal , 473 :1225 , 2016
Abstract :
PubMedSearch : Kharlamova_2016_Biochem.J_473_1225
PubMedID: 26929400
Gene_locus related to this paper: mouse-ACHE

Title : Novel potent pyridoxine-based inhibitors of AChE and BChE, structural analogs of pyridostigmine, with improved in vivo safety profile - Strelnik_2016_Bioorg.Med.Chem.Lett_26_4092
Author(s) : Strelnik AD , Petukhov AS , Zueva IV , Zobov VV , Petrov KA , Nikolsky EE , Balakin KV , Bachurin SO , Shtyrlin YG
Ref : Bioorganic & Medicinal Chemistry Lett , 26 :4092 , 2016
Abstract :
PubMedSearch : Strelnik_2016_Bioorg.Med.Chem.Lett_26_4092
PubMedID: 27377327

Title : 6-Methyluracil Derivatives as Bifunctional Acetylcholinesterase Inhibitors for the Treatment of Alzheimer's Disease - Semenov_2015_ChemMedChem_10_1863
Author(s) : Semenov VE , Zueva IV , Mukhamedyarov MA , Lushchekina SV , Kharlamova AD , Petukhova EO , Mikhailov AS , Podyachev SN , Saifina LF , Petrov KA , Minnekhanova OA , Zobov VV , Nikolsky EE , Masson P , Reznik VS
Ref : ChemMedChem , 10 :1863 , 2015
Abstract :
PubMedSearch : Semenov_2015_ChemMedChem_10_1863
PubMedID: 26412714

Title : 6-Methyluracil derivatives as acetylcholinesterase inhibitors for treatment of Alzheimer's disease - Zueva_2015_Int.J.Risk.Saf.Med_27 Suppl 1_S69
Author(s) : Zueva IV , Semenov VE , Mukhamedyarov MA , Lushchekina SV , Kharlamova AD , Petukhova EO , Mikhailov AS , Podyachev SN , Saifina LF , Petrov KA , Minnekhanova OA , Zobov VV , Nikolsky EE , Masson P , Reznik VS
Ref : Int J Risk Saf Med , 27 Suppl 1 :S69 , 2015
Abstract :
PubMedSearch : Zueva_2015_Int.J.Risk.Saf.Med_27 Suppl 1_S69
PubMedID: 26639718

Title : Schwann Cells Sense and Control Acetylcholine Spillover at the Neuromuscular Junction by alpha7 Nicotinic Receptors and Butyrylcholinesterase - Petrov_2014_J.Neurosci_34_11870
Author(s) : Petrov KA , Girard E , Nikitashina AD , Colasante C , Bernard V , Nurullin LF , Leroy J , Samigullin D , Colak O , Nikolsky EE , Plaud B , Krejci E
Ref : Journal of Neuroscience , 34 :11870 , 2014
Abstract :
PubMedSearch : Petrov_2014_J.Neurosci_34_11870
PubMedID: 25186736

Title : Specific inhibitory effects of the alkylammonium derivative 6-methyluracil on acetylcholinesterase of smooth and striated muscles in rats -
Author(s) : Nikitashina AD , Petrov KA , Zobov VV , Reznik VS , Nikolsky EE
Ref : Dokl Biol Sci , 449 :82 , 2013
PubMedID: 23652433

Title : Regulation of acetylcholinesterase activity by nitric oxide in rat neuromuscular junction via N-methyl-d-aspartate receptor activation - Petrov_2013_Eur.J.Neurosci_37_181
Author(s) : Petrov KA , Malomouzh AI , Kovyazina IV , Krejci E , Nikitashina AD , Proskurina SE , Zobov VV , Nikolsky EE
Ref : European Journal of Neuroscience , 37 :181 , 2013
Abstract :
PubMedSearch : Petrov_2013_Eur.J.Neurosci_37_181
PubMedID: 23121214

Title : Effect of tissue-specific acetylcholinesterase inhibitor C-547 on alpha3beta4 and alphabetaepsilondelta acetylcholine receptors in COS cells - Lindovsky_2012_Eur.J.Pharmacol_688_22
Author(s) : Lindovsky J , Petrov KA , Krusek J , Reznik VS , Nikolsky EE , Vyskocil F
Ref : European Journal of Pharmacology , 688 :22 , 2012
Abstract :
PubMedSearch : Lindovsky_2012_Eur.J.Pharmacol_688_22
PubMedID: 22634638

Title : Both neuronal and non-neuronal acetylcholine take part in non-quantal acetylcholine release in the rat atrium - Abramochkin_2012_Life.Sci_91_1023
Author(s) : Abramochkin DV , Borodinova AA , Rosenshtraukh LV , Nikolsky EE
Ref : Life Sciences , 91 :1023 , 2012
Abstract :
PubMedSearch : Abramochkin_2012_Life.Sci_91_1023
PubMedID: 23289117

Title : Different sensitivities of rat skeletal muscles and brain to novel anti-cholinesterase agents, alkylammonium derivatives of 6-methyluracil (ADEMS) - Petrov_2011_Br.J.Pharmacol_163_732
Author(s) : Petrov KA , Yagodina LO , Valeeva GR , Lannik NI , Nikitashina AD , Rizvanov AA , Zobov VV , Bukharaeva EA , Reznik VS , Nikolsky EE , Vyskocil F
Ref : British Journal of Pharmacology , 163 :732 , 2011
Abstract :
PubMedSearch : Petrov_2011_Br.J.Pharmacol_163_732
PubMedID: 21232040

Title : Non-quantal release of acetylcholine from parasympathetic nerve terminals in the right atrium of rats - Abramochkin_2010_Exp.Physiol_95_265
Author(s) : Abramochkin DV , Nurullin LF , Borodinova AA , Tarasova NV , Sukhova GS , Nikolsky EE , Rosenshtraukh LV
Ref : Exp Physiol , 95 :265 , 2010
Abstract :
PubMedSearch : Abramochkin_2010_Exp.Physiol_95_265
PubMedID: 19767403

Title : Mechanisms of cardiac muscle insensitivity to a novel acetylcholinesterase inhibitor C-547 - Abramochkin_2009_J.Cardiovasc.Pharmacol_53_162
Author(s) : Abramochkin DV , Petrov KA , Zobov VV , Yagodina LO , Nikolsky EE , Rosenshtraukh LV
Ref : J Cardiovasc Pharmacol , 53 :162 , 2009
Abstract :
PubMedSearch : Abramochkin_2009_J.Cardiovasc.Pharmacol_53_162
PubMedID: 19188831

Title : Different sensitivity of miniature endplate currents in rat external and internal intercostal muscles to the acetylcholinesterase inhibitor C-547 as compared with diaphragm and extensor digitorum longus - Petrov_2009_Physiol.Res_58_149
Author(s) : Petrov KA , Kovyazina IV , Zobov VV , Bukharaeva EA , Nikolsky EE , Vyskocil F
Ref : Physiol Res , 58 :149 , 2009
Abstract :
PubMedSearch : Petrov_2009_Physiol.Res_58_149
PubMedID: 19331513

Title : Effect of a tetraalkylammonium derivative of 6-methyluracil from a new class of acetylcholinesterase inhibitors on the endplate potential amplitude in muscles of different function types under high-frequency nerve stimulation -
Author(s) : Petrov KA , Kovyazina IV , Zobov VV , Bukharaeva EA , Reznik VS , Nikolsky EE
Ref : Dokl Biol Sci , 415 :261 , 2007
PubMedID: 17929660

Title : Different sensitivity of miniature endplate currents of the rat extensor digitorum longus, soleus and diaphragm muscles to a novel acetylcholinesterase inhibitor C-547 - Petrov_2006_Physiol.Res_55_585
Author(s) : Petrov KA , Kovyazina LV , Zobov VV , Bukharaeva EA , Nikolsky EE , Vyskocil F
Ref : Physiol Res , 55 :585 , 2006
Abstract :
PubMedSearch : Petrov_2006_Physiol.Res_55_585
PubMedID: 16792471

Title : Effect of N-acetylaspartylglutamate (NAAG) on non-quantal and spontaneous quantal release of acetylcholine at the neuromuscular synapse of rat - Malomouzh_2005_J.Neurochem_94_257
Author(s) : Malomouzh AI , Nikolsky EE , Lieberman EM , Sherman JA , Lubischer JL , Grossfeld RM , Urazaev A
Ref : Journal of Neurochemistry , 94 :257 , 2005
Abstract :
PubMedSearch : Malomouzh_2005_J.Neurochem_94_257
PubMedID: 15953368

Title : Dependence of miniature endplate current on kinetic parameters of acetylcholine receptors activation: a model study - Kovyazina_2003_Neurochem.Res_28_443
Author(s) : Kovyazina IV , Nikolsky EE , Giniatullin RA , Adamek S , Vyskocil F
Ref : Neurochem Res , 28 :443 , 2003
Abstract :
PubMedSearch : Kovyazina_2003_Neurochem.Res_28_443
PubMedID: 12675129

Title : Glutamate regulation of non-quantal release of acetylcholine in the rat neuromuscular junction - Malomouzh_2003_J.Neurochem_85_206
Author(s) : Malomouzh AI , Mukhtarov MR , Nikolsky EE , Vyskocil F , Lieberman EM , Urazaev AK
Ref : Journal of Neurochemistry , 85 :206 , 2003
Abstract :
PubMedSearch : Malomouzh_2003_J.Neurochem_85_206
PubMedID: 12641742

Title : Modulation by nitric oxide (NO) of the intensity of non-quantum mediator secretion in neuromuscular junctions in rats - Mukhtarov_2001_Neurosci.Behav.Physiol_31_451
Author(s) : Mukhtarov MR , Urazaev AK , Nikolsky EE , Vyskocil F
Ref : Neurosci Behav Physiol , 31 :451 , 2001
Abstract :
PubMedSearch : Mukhtarov_2001_Neurosci.Behav.Physiol_31_451
PubMedID: 11508498

Title : Effect of tetraalkylammonium derivative of 6-methyluracil on amplitude and temporal parameters of miniature endplate potentials in frog neuromuscular junction - Gorshkova_2001_Bull.Exp.Biol.Med_131_446
Author(s) : Gorshkova OV , Zobov VV , Bukharaeva EA , Nikolsky EE , Akamsin VD , Galyametdinova IV , Reznik VS
Ref : Bulletin of Experimental Biology & Medicine , 131 :446 , 2001
Abstract :
PubMedSearch : Gorshkova_2001_Bull.Exp.Biol.Med_131_446
PubMedID: 11550049

Title : Non-quantal acetylcholine release is increased after nitric oxide synthase inhibition - Mukhtarov_1999_Physiol.Res_48_315
Author(s) : Mukhtarov MR , Vyskocil F , Urazaev AK , Nikolsky EE
Ref : Physiol Res , 48 :315 , 1999
Abstract :
PubMedSearch : Mukhtarov_1999_Physiol.Res_48_315
PubMedID: 10638684

Title : The NO-mediated effect of carbachol and glutamate on postdenervation decrease of membrane potential in rat diaphragm is directed towards furosemide-sensitive chloride transport -
Author(s) : Vyskocil F , Urazaev AK , Naumenko NV , Nikolsky EE
Ref : Journal de Physiologie (Paris) , 92 :507 , 1998
PubMedID:

Title : Role of non-quantal acetylcholine release in surplus polarization of mouse diaphragm fibres at the endplate zone - Nikolsky_1994_J.Physiol_477_497
Author(s) : Nikolsky EE , Zemkova H , Voronin VA , Vyskocil F
Ref : The Journal of Physiology , 477 :497 , 1994
Abstract :
PubMedSearch : Nikolsky_1994_J.Physiol_477_497
PubMedID: 7932237

Title : Functional role of cholinesterase in different types of neuro-muscular junction -
Author(s) : Magazanik LG , Fedorov VV , Giniatullin RA , Nikolsky EE , Snetkov VA
Ref : In: Cholinesterases, fundamental and applied aspects : proceedings of the Second International Meeting on Cholinesterases , (Brzin M, Barnard EA, Sket D, Eds) De Gruyter :229 , 1984
PubMedID: