Title : A novel mechanism of G protein-coupled receptor functional selectivity. Muscarinic partial agonist McN-A-343 as a bitopic orthosteric\/allosteric ligand - Valant_2008_J.Biol.Chem_283_29312 |
Author(s) : Valant C , Gregory KJ , Hall NE , Scammells PJ , Lew MJ , Sexton PM , Christopoulos A |
Ref : Journal of Biological Chemistry , 283 :29312 , 2008 |
Abstract : |
PubMedSearch : Valant_2008_J.Biol.Chem_283_29312 |
PubMedID: 18723515 |
Title : The assessment of antagonist potency under conditions of transient response kinetics - Christopoulos_1999_Eur.J.Pharmacol_382_217 |
Author(s) : Christopoulos A , Parsons AM , Lew MJ , El-Fakahany EE |
Ref : European Journal of Pharmacology , 382 :217 , 1999 |
Abstract : |
PubMedSearch : Christopoulos_1999_Eur.J.Pharmacol_382_217 |
PubMedID: 10556673 |