McGuire R

Title : Discovery of Glycine Sulfonamides as Dual Inhibitors of sn-1-Diacylglycerol Lipase alpha and alpha\/beta-Hydrolase Domain 6 - Janssen_2014_J.Med.Chem_57_6610

Author(s) : Janssen FJ , Deng H , Baggelaar MP , Allara M , van der Wel T , den Dulk H , Ligresti A , van Esbroeck AC , McGuire R , Di Marzo V , Overkleeft HS , van der Stelt M

Ref : Journal of Medicinal Chemistry , 57 :6610 , 2014

Abstract :

PubMedSearch : Janssen_2014_J.Med.Chem_57_6610

PubMedID: 24988361

Title : Development of an activity-based probe and in silico design reveal highly selective inhibitors for diacylglycerol lipase-alpha in brain - Baggelaar_2013_Angew.Chem.Int.Ed.Engl_52_12081

Author(s) : Baggelaar MP , Janssen FJ , van Esbroeck AC , den Dulk H , Allara M , Hoogendoorn S , McGuire R , Florea BI , Meeuwenoord N , van den Elst H , van der Marel GA , Brouwer J , Di Marzo V , Overkleeft HS , van der Stelt M

Ref : Angew Chem Int Ed Engl , 52 :12081 , 2013

Abstract :

PubMedSearch : Baggelaar_2013_Angew.Chem.Int.Ed.Engl_52_12081

PubMedID: 24173880

Gene_locus related to this paper: human-DAGLA

McGuire R

References (2)

1. Discovery of Glycine Sulfonamides as Dual Inhibitors of sn-1-Diacylglycerol Lipase alpha and alpha\/beta-Hydrolase Domain 6 - Janssen_2014_J.Med.Chem_57_6610

2. Development of an activity-based probe and in silico design reveal highly selective inhibitors for diacylglycerol lipase-alpha in brain - Baggelaar_2013_Angew.Chem.Int.Ed.Engl_52_12081