Overkleeft HS

References (19)

Title : Identification of fungal lignocellulose-degrading biocatalysts secreted by Phanerochaete chrysosporium via activity-based protein profiling - Schmerling_2022_Commun.Biol_5_1254
Author(s) : Schmerling C , Sewald L , Heilmann G , Witfeld F , Begerow D , Jensen K , Brsen C , Kaschani F , Overkleeft HS , Siebers B , Kaiser M
Ref : Commun Biol , 5 :1254 , 2022
Abstract :
PubMedSearch : Schmerling_2022_Commun.Biol_5_1254
PubMedID: 36385496

Title : Detecting and identifying glycoside hydrolases using cyclophellitol-derived activity-based probes - McGregor_2022_Methods.Enzymol_664_103
Author(s) : McGregor NGS , Overkleeft HS , Davies GJ
Ref : Methods Enzymol , 664 :103 , 2022
Abstract :
PubMedSearch : McGregor_2022_Methods.Enzymol_664_103
PubMedID: 35331370

Title : ABHD2 Inhibitor Identified by Activity-Based Protein Profiling Reduces Acrosome Reaction - Baggelaar_2019_ACS.Chem.Biol_14_2295
Author(s) : Baggelaar MP , den Dulk H , Florea BI , Fazio D , Perruzza D , Bernabo N , Raspa M , Janssen APA , Scavizzi F , Barboni B , Overkleeft HS , Maccarrone M , van der Stelt M
Ref : ACS Chemical Biology , 14 :2295 , 2019
Abstract :
PubMedSearch : Baggelaar_2019_ACS.Chem.Biol_14_2295
PubMedID: 31525885
Gene_locus related to this paper: human-ABHD2 , human-ABHD3

Title : Identification of alpha,beta-Hydrolase Domain Containing Protein 6 as a Diacylglycerol Lipase in Neuro-2a Cells - van Esbroeck_2019_Front.Mol.Neurosci_12_286
Author(s) : van Esbroeck ACM , Kantae V , Di X , van der Wel T , den Dulk H , Stevens AF , Singh S , Bakker AT , Florea BI , Stella N , Overkleeft HS , Hankemeier T , van der Stelt M
Ref : Front Mol Neurosci , 12 :286 , 2019
Abstract :
PubMedSearch : van Esbroeck_2019_Front.Mol.Neurosci_12_286
PubMedID: 31849602
Gene_locus related to this paper: human-ABHD6

Title : Activity-Based Protein Profiling Identifies alpha-Ketoamides as Inhibitors for Phospholipase A2 Group XVI - Zhou_2019_ACS.Chem.Biol_14_164
Author(s) : Zhou J , Mock ED , Martella A , Kantae V , Di X , Burggraaff L , Baggelaar MP , Al-Ayed K , Bakker A , Florea BI , Grimm SH , den Dulk H , Li CT , Mulder L , Overkleeft HS , Hankemeier T , van Westen GJP , van der Stelt M
Ref : ACS Chemical Biology , 14 :164 , 2019
Abstract :
PubMedSearch : Zhou_2019_ACS.Chem.Biol_14_164
PubMedID: 30620559

Title : Mapping in vivo target interaction profiles of covalent inhibitors using chemical proteomics with label-free quantification - van Rooden_2018_Nat.Protoc_13_752
Author(s) : van Rooden EJ , Florea BI , Deng H , Baggelaar MP , van Esbroeck ACM , Zhou J , Overkleeft HS , van der Stelt M
Ref : Nat Protoc , 13 :752 , 2018
Abstract :
PubMedSearch : van Rooden_2018_Nat.Protoc_13_752
PubMedID: 29565900

Title : Design and Synthesis of Quenched Activity-based Probes for Diacylglycerol Lipase and alpha,beta-Hydrolase Domain Containing Protein 6 - van Rooden_2018_Chem.Asian.J_13_3491
Author(s) : van Rooden EJ , Kohsiek M , Kreekel R , van Esbroeck ACM , van den Nieuwendijk A , Janssen APA , van den Berg R , Overkleeft HS , van der Stelt M
Ref : Chem Asian J , 13 :3491 , 2018
Abstract :
PubMedSearch : van Rooden_2018_Chem.Asian.J_13_3491
PubMedID: 29901868

Title : Chemical Proteomic Analysis of Serine Hydrolase Activity in Niemann-Pick Type C Mouse Brain - van Rooden_2018_Front.Neurosci_12_440
Author(s) : van Rooden EJ , van Esbroeck ACM , Baggelaar MP , Deng H , Florea BI , Marques ARA , Ottenhoff R , Boot RG , Overkleeft HS , Aerts J , van der Stelt M
Ref : Front Neurosci , 12 :440 , 2018
Abstract :
PubMedSearch : van Rooden_2018_Front.Neurosci_12_440
PubMedID: 30018533

Title : Chemical Proteomics Maps Brain Region Specific Activity of Endocannabinoid Hydrolases - Baggelaar_2017_ACS.Chem.Biol_12_852
Author(s) : Baggelaar MP , van Esbroeck AC , van Rooden EJ , Florea BI , Overkleeft HS , Marsicano G , Chaouloff F , van der Stelt M
Ref : ACS Chemical Biology , 12 :852 , 2017
Abstract :
PubMedSearch : Baggelaar_2017_ACS.Chem.Biol_12_852
PubMedID: 28106377
Gene_locus related to this paper: human-ABHD4 , human-ABHD6 , human-ABHD12 , human-DAGLA , human-MGLL

Title : Chiral disubstituted piperidinyl ureas: a class of dual diacylglycerol lipase-alpha and ABHD6 inhibitors - Deng_2017_Medchemcomm_8_982
Author(s) : Deng H , van der Wel T , van den Berg R , van den Nieuwendijk A , Janssen FJ , Baggelaar MP , Overkleeft HS , van der Stelt M
Ref : Medchemcomm , 8 :982 , 2017
Abstract :
PubMedSearch : Deng_2017_Medchemcomm_8_982
PubMedID: 30108813
Gene_locus related to this paper: human-ABHD6

Title : Triazole Ureas Act as Diacylglycerol Lipase Inhibitors and Prevent Fasting-Induced Refeeding - Deng_2017_J.Med.Chem_60_428
Author(s) : Deng H , Kooijman S , van den Nieuwendijk AM , Ogasawara D , van der Wel T , van Dalen F , Baggelaar MP , Janssen FJ , van den Berg RJ , den Dulk H , Cravatt BF , Overkleeft HS , Rensen PC , van der Stelt M
Ref : Journal of Medicinal Chemistry , 60 :428 , 2017
Abstract :
PubMedSearch : Deng_2017_J.Med.Chem_60_428
PubMedID: 27992221

Title : Activity-based protein profiling reveals off-target proteins of the FAAH inhibitor BIA 10-2474 - van Esbroeck_2017_Science_356_1084
Author(s) : van Esbroeck ACM , Janssen APA , Cognetta AB, 3rd , Ogasawara D , Shpak G , van der Kroeg M , Kantae V , Baggelaar MP , de Vrij FMS , Deng H , Allara M , Fezza F , Lin Z , van der Wel T , Soethoudt M , Mock ED , den Dulk H , Baak IL , Florea BI , Hendriks G , De Petrocellis L , Overkleeft HS , Hankemeier T , De Zeeuw CI , Di Marzo V , Maccarrone M , Cravatt BF , Kushner SA , van der Stelt M
Ref : Science , 356 :1084 , 2017
Abstract :
PubMedSearch : van Esbroeck_2017_Science_356_1084
PubMedID: 28596366

Title : Rapid and profound rewiring of brain lipid signaling networks by acute diacylglycerol lipase inhibition - Ogasawara_2016_Proc.Natl.Acad.Sci.U.S.A_113_26
Author(s) : Ogasawara D , Deng H , Viader A , Baggelaar MP , Breman A , den Dulk H , van den Nieuwendijk AM , Soethoudt M , van der Wel T , Zhou J , Overkleeft HS , Sanchez-Alavez M , Mori S , Nguyen W , Conti B , Liu X , Chen Y , Liu QS , Cravatt BF , van der Stelt M
Ref : Proc Natl Acad Sci U S A , 113 :26 , 2016
Abstract :
PubMedSearch : Ogasawara_2016_Proc.Natl.Acad.Sci.U.S.A_113_26
PubMedID: 26668358
Gene_locus related to this paper: human-DAGLA , human-DAGLB

Title : Comprehensive Analysis of Structure-Activity Relationships of alpha-Ketoheterocycles as sn-1-Diacylglycerol Lipase alpha Inhibitors - Janssen_2015_J.Med.Chem_58_9742
Author(s) : Janssen FJ , Baggelaar MP , Hummel JJ , Overkleeft HS , Cravatt BF , Boger DL , van der Stelt M
Ref : Journal of Medicinal Chemistry , 58 :9742 , 2015
Abstract :
PubMedSearch : Janssen_2015_J.Med.Chem_58_9742
PubMedID: 26584396

Title : Highly Selective, Reversible Inhibitor Identified by Comparative Chemoproteomics Modulates Diacylglycerol Lipase Activity in Neurons - Baggelaar_2015_J.Am.Chem.Soc_137_8851
Author(s) : Baggelaar MP , Chameau PJ , Kantae V , Hummel J , Hsu KL , Janssen F , van der Wel T , Soethoudt M , Deng H , den Dulk H , Allara M , Florea BI , Di Marzo V , Wadman WJ , Kruse CG , Overkleeft HS , Hankemeier T , Werkman TR , Cravatt BF , van der Stelt M
Ref : Journal of the American Chemical Society , 137 :8851 , 2015
Abstract :
PubMedSearch : Baggelaar_2015_J.Am.Chem.Soc_137_8851
PubMedID: 26083464
Gene_locus related to this paper: human-DAGLA , human-DAGLB

Title : A natural substrate-based fluorescence assay for inhibitor screening on diacylglycerol lipase alpha - van der Wel_2015_J.Lipid.Res_56_927
Author(s) : van der Wel T , Janssen FJ , Baggelaar MP , Deng H , den Dulk H , Overkleeft HS , van der Stelt M
Ref : J Lipid Res , 56 :927 , 2015
Abstract :
PubMedSearch : van der Wel_2015_J.Lipid.Res_56_927
PubMedID: 25684760

Title : Discovery of Glycine Sulfonamides as Dual Inhibitors of sn-1-Diacylglycerol Lipase alpha and alpha\/beta-Hydrolase Domain 6 - Janssen_2014_J.Med.Chem_57_6610
Author(s) : Janssen FJ , Deng H , Baggelaar MP , Allara M , van der Wel T , den Dulk H , Ligresti A , van Esbroeck AC , McGuire R , Di Marzo V , Overkleeft HS , van der Stelt M
Ref : Journal of Medicinal Chemistry , 57 :6610 , 2014
Abstract :
PubMedSearch : Janssen_2014_J.Med.Chem_57_6610
PubMedID: 24988361

Title : Development of an activity-based probe and in silico design reveal highly selective inhibitors for diacylglycerol lipase-alpha in brain -
Author(s) : Baggelaar MP , Janssen FJ , van Esbroeck AC , den Dulk H , Allara M , Hoogendoorn S , McGuire R , Florea BI , Meeuwenoord N , van den Elst H , van der Marel GA , Brouwer J , Di Marzo V , Overkleeft HS , van der Stelt M
Ref : Angew Chem Int Ed Engl , 52 :12081 , 2013
PubMedID: 24173880
Gene_locus related to this paper: human-DAGLA

Title : Activity-Based Protein Profiling Reveals Broad Reactivity of the Nerve Agent Sarin - Tuin_2009_Chem.Res.Toxicol_22_683
Author(s) : Tuin AW , Mol MA , van den Berg RM , Fidder A , van der Marel GA , Overkleeft HS , Noort D
Ref : Chemical Research in Toxicology , 22 :683 , 2009
Abstract :
PubMedSearch : Tuin_2009_Chem.Res.Toxicol_22_683
PubMedID: 19226147