Title : Chemoproteomics-Enabled Identification of 4-Oxo-beta-Lactams as Inhibitors of Dipeptidyl Peptidases 8 and 9 - Carvalho_2022_Angew.Chem.Int.Ed.Engl_61_e202210498 |
Author(s) : Carvalho LAR , Ross B , Fehr L , Bolgi O , Wohrle S , Lum KM , Podlesainski D , Vieira AC , Kiefersauer R , Felix R , Rodrigues T , Lucas SD , Gross O , Geiss-Friedlander R , Cravatt BF , Huber R , Kaiser M , Moreira R |
Ref : Angew Chem Int Ed Engl , : , 2022 |
Abstract : |
PubMedSearch : Carvalho_2022_Angew.Chem.Int.Ed.Engl_61_e202210498 |
PubMedID: 36089535 |
Gene_locus related to this paper: human-DPP8 , human-DPP9 |
Title : Repeated Administration of Clinical Doses of Tramadol and Tapentadol Causes Hepato- and Nephrotoxic Effects in Wistar Rats - Barbosa_2020_Pharmaceuticals.(Basel)_13_ |
Author(s) : Barbosa J , Faria J , Garcez F , Leal S , Afonso LP , Nascimento AV , Moreira R , Queiros O , Carvalho F , Dinis-Oliveira RJ |
Ref : Pharmaceuticals (Basel) , 13 : , 2020 |
Abstract : |
PubMedSearch : Barbosa_2020_Pharmaceuticals.(Basel)_13_ |
PubMedID: 32664348 |
Title : 3-Oxo-beta-sultam as a Sulfonylating Chemotype for Inhibition of Serine Hydrolases and Activity-Based Protein Profiling - Carvalho_2020_ACS.Chem.Biol_15_878 |
Author(s) : Carvalho LAR , Almeida VT , Brito JA , Lum KM , Oliveira TF , Guedes RC , Goncalves LM , Lucas SD , Cravatt BF , Archer M , Moreira R |
Ref : ACS Chemical Biology , 15 :878 , 2020 |
Abstract : |
PubMedSearch : Carvalho_2020_ACS.Chem.Biol_15_878 |
PubMedID: 32176480 |
Title : Acute administration of tramadol and tapentadol at effective analgesic and maximum tolerated doses causes hepato- and nephrotoxic effects in Wistar rats - Barbosa_2017_Toxicology_389_118 |
Author(s) : Barbosa J , Faria J , Leal S , Afonso LP , Lobo J , Queiros O , Moreira R , Carvalho F , Dinis-Oliveira RJ |
Ref : Toxicology , 389 :118 , 2017 |
Abstract : |
PubMedSearch : Barbosa_2017_Toxicology_389_118 |
PubMedID: 28689766 |
Title : A carbamate-based approach to primaquine prodrugs: antimalarial activity, chemical stability and enzymatic activation - Mata_2012_Bioorg.Med.Chem_20_886 |
Author(s) : Mata G , do Rosario VE , Iley J , Constantino L , Moreira R |
Ref : Bioorganic & Medicinal Chemistry , 20 :886 , 2012 |
Abstract : |
PubMedSearch : Mata_2012_Bioorg.Med.Chem_20_886 |
PubMedID: 22189276 |
Title : Acyloxymethyl as a drug protecting group. Part 6: N-acyloxymethyl- and N-[(aminocarbonyloxy)methyl]sulfonamides as prodrugs of agents containing a secondary sulfonamide group - Lopes_2000_Bioorg.Med.Chem_8_707 |
Author(s) : Lopes F , Moreira R , Iley J |
Ref : Bioorganic & Medicinal Chemistry , 8 :707 , 2000 |
Abstract : |
PubMedSearch : Lopes_2000_Bioorg.Med.Chem_8_707 |
PubMedID: 10819159 |